Patents by Inventor Edward E. Kilbourn

Edward E. Kilbourn has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4310537
    Abstract: Acetyl- and carbalkoxythioureidobenzophenones having a substituted amine adjacent to the thioureido radical are disclosed as having anthelmintic and antifungal activity.
    Type: Grant
    Filed: October 7, 1977
    Date of Patent: January 12, 1982
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, W. David Weir
  • Patent number: 4297342
    Abstract: Novel 3-pyridylmethyl N-(4-substituted-phenyl)thiocarbamates are disclosed. These compounds are useful as single-dose rodenticides, which have high bait acceptance.
    Type: Grant
    Filed: January 17, 1980
    Date of Patent: October 27, 1981
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, Ernest D. Weiler, William D. Weir
  • Patent number: 4276290
    Abstract: This invention relates to novel anthelmintic compounds containing an arylene or divalent heterocyclic ring whose free valences are satisfied by(1) a disubstituted phosphoryl ureido or thioureido group and(2) an amino group or a substituted amido or thioamido group,to compositions containing them, and to methods of using them for the treatment of intestinal parasites in mammals and birds.
    Type: Grant
    Filed: September 6, 1979
    Date of Patent: June 30, 1981
    Assignee: Rohm and Haas Company
    Inventors: W. David Weir, Edward E. Kilbourn
  • Patent number: 4259330
    Abstract: This invention relates to novel phosphoramidates of the formula: ##STR1## wherein R.sup.1 is hydrogen, alkyl, cycloalkyl, or optionally substituted aralkyl, aryl, pyridyl, pyridylmethyl, pyridylethyl or pyrazinyl;R.sup.2 is hydrogen provided R.sup.1 is other than optionally substituted aryl; alkyl; cycloalkyl; alkoxyalkyl; alkylthioalkyl; cyanoalkyl; alkenyl; optionally substituted aralylky; or optionally substituted aryl, provided R.sup.1 is other than hydrogen;R.sup.1 and R.sup.2 taken together with the nitrogen to which they are attached form an optionally substituted morpholino or piperidino group;R.sup.3 is hydrogen, alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.4 is (C.sub.1 -C.sub.6) alkyl;R.sup.5 is (C.sub.3 -C.sub.4) alkyl; andX, Y and Z are independently oxygen or sulfur;the agronomically acceptable metal salts and metal salt complexes thereof; and to methods of using them to control nematodes.
    Type: Grant
    Filed: March 1, 1976
    Date of Patent: March 31, 1981
    Assignee: Rohm and Haas Company
    Inventors: Harold E. Aller, Edward E. Kilbourn, Ernest D. Weiler, William D. Weir
  • Patent number: 4241079
    Abstract: 2-Imino substituted isothioureidobenzene products useful as anthelmintics and fungicides are disclosed. The products may be prepared by several different methods including treating a 2-iminothioureidobenzene with a base and either an organic halide, a diester of sulfuric acid or a diester of sulfurous acid or treating a 2-aminoisothioureidobenzene with an appropriately substituted aldehyde.
    Type: Grant
    Filed: May 4, 1978
    Date of Patent: December 23, 1980
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, W. David Weir
  • Patent number: 4234575
    Abstract: This invention relates to novel anthelmintic compounds containing an arylene or divalent heterocyclic ring whose free valences are satisfied by(1) a disubstituted phosphoryl ureido or thioureido group and(2) an amino group or a substituted amido or thioamido group,to compositions containing them, and to methods of using them for the treatment of intestinal parasites in mammals and birds.
    Type: Grant
    Filed: January 31, 1979
    Date of Patent: November 18, 1980
    Assignee: Rohm and Haas Company
    Inventors: W. David Weir, Edward E. Kilbourn
  • Patent number: 4233289
    Abstract: Novel 3-pyridylmethyl N-(4-substituted-phenyl)thiocarbamates are disclosed. These compounds are useful as single-dose rodenticides, which have high baitacceptance.
    Type: Grant
    Filed: January 31, 1979
    Date of Patent: November 11, 1980
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, Ernest D. Weiler, William D. Weir
  • Patent number: 4183921
    Abstract: This invention relates to novel anthelmintic compounds containing an arylene or divalent heterocyclic ring whose free valences are satisfied by(1) a disubstituted phosphoryl ureido or thioureido group and(2) an amino group or a substituted amido or thioamido group,to compositions containing them, and to methods of using them for the treatment of intestinal parasites in mammals and birds.
    Type: Grant
    Filed: October 17, 1977
    Date of Patent: January 15, 1980
    Assignee: Rohm and Haas Company
    Inventors: W. David Weir, Edward E. Kilbourn
  • Patent number: 4156780
    Abstract: Novel 3-pyridylmethyl N-(4-substituted-phenyl)thiocarbamates are disclosed. These compounds are useful as single-dose rodenticides, which have high bait acceptance.
    Type: Grant
    Filed: June 30, 1975
    Date of Patent: May 29, 1979
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, Ernest D. Weiler, William D. Weir
  • Patent number: 4139614
    Abstract: This invention relates to novel anthelmintic compositions containing as the essential active ingredient, a compound of the formula: ##STR1## wherein R.sup.1 is cylcoalkyl, or optionally substituted aralkyl, aryl, pyridyl, or pyrazinyl;R.sup.2 is hydrogen, alkyl, cycloalkyl, alkoxyalkyl, alkylthioalkyl, cyanoalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.1 and R.sup.2 taken together with the nitrogen atom to which they are attached form an optionally substituted morpholino or piperidino group;R.sup.3 is hydrogen, alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.4 is alkoxy, haloalkoxy, dialkylamino, alkylthio, phenoxy or phenylthio; andR.sup.5 is alkyl, alkoxy, haloalkoxy, dialkylamino, alkylthio, phenyl, phenoxy or phenylthio; andX is oxygen or sulfur;And pharmaceutically acceptable metal salts and metal salt complexes thereof, and to methods of employing them in the treatment of intestinal parasites in animals, e.g. mammals, fish, and birds.
    Type: Grant
    Filed: March 1, 1976
    Date of Patent: February 13, 1979
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, Ernest Weiler, William D. Weir
  • Patent number: 4087521
    Abstract: This invention relates to novel phosphoramidates of the formula: ##STR1## wherein R.sup.1 is (C.sub.6 -C.sub.10) aryl optionally substituted with alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, dialkylamino, haloalkyl, hydroxyalkyl, cyano, nitro, hydroxy, or halogen;R.sup.2 is hydrogen, alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.3 is (C.sub.1 -C.sub.6) alkyl;R.sup.4 is (C.sub.3 -C.sub.4) alkyl; andX, y and Z are independently oxygen or sulfur;And the agronomically acceptable metal salts and metal salt complexes thereof; to compositions containing them; and to methods of using them to control certain harmful pests, e.g. arthropods and nematodes.
    Type: Grant
    Filed: March 1, 1976
    Date of Patent: May 2, 1978
    Assignee: Rohm and Haas Company
    Inventors: Harold E. Aller, Edward E. Kilbourn, Ernest D. Weiler, William D. Weir
  • Patent number: 4076809
    Abstract: This invention relates to novel anthelmintic compounds containing an arylene or divalent heterocyclic ring whose free valences are satisfied by1. a disubstituted phosphoryl ureido or thioureido group and2. an amino group or a substituted amido or thioamido group,To compositions containing them, and to methods of using them for the treatment of intestinal parasites in mammals and birds.
    Type: Grant
    Filed: October 28, 1975
    Date of Patent: February 28, 1978
    Assignee: Rohm and Haas Company
    Inventors: W. David Weir, Edward E. Kilbourn
  • Patent number: 4075345
    Abstract: Rodenticidal compositions containing as the active ingredient novel 1-(3-pyridylmethyl)-3-(4'-substituted-phenyl or -naphthyl)ureas and their acid addition salts. The 4'-substituent may be nitro, cyano, trifluoromethyl, butyryl, thiocyano, alkylthio, phenylsulfonyl or diethylsulfonamide.
    Type: Grant
    Filed: April 11, 1974
    Date of Patent: February 21, 1978
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, David L. Peardon, J. Edgar Ware
  • Patent number: 4060636
    Abstract: Acetyl- and carbalkoxythioureidobenzophenones having a substituted amine adjacent to the thioureido radical are disclosed as having anthelmintic and antifungal activity.
    Type: Grant
    Filed: June 10, 1976
    Date of Patent: November 29, 1977
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, W. David Weir
  • Patent number: 4033972
    Abstract: 3-Pyridylmethyl-(N-substituted-phenyl-N-hydrocarbyl)carbamates. They are useful as rodenticides.
    Type: Grant
    Filed: September 9, 1975
    Date of Patent: July 5, 1977
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, Ernest D. Weiler
  • Patent number: 3994905
    Abstract: Novel 1-(3-pyridylmethyl)-3-(4'-substituted-phenyl or -naphthyl)-ureas and their acid addition salts. The 4'-substituent may be -NO.sub.2, -CN, -CF.sub.3, -C(O)R.sub.1, -SCN, SR.sub.2, -SO.sub.2 C.sub.6 H.sub.5 or -SO.sub.2 NR.sub.3 R.sub.4. These compounds are biologically active, and many are active rodenticides.
    Type: Grant
    Filed: October 16, 1975
    Date of Patent: November 30, 1976
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, David L. Peardon, J. Edgar Ware
  • Patent number: 3966947
    Abstract: 3-Pyridylmethyl N-(4'-substitutedmercaptophenyl) carbamates and their acid salts and metal salt complexes useful as a rodenticide.
    Type: Grant
    Filed: October 3, 1975
    Date of Patent: June 29, 1976
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, Ernest D. Weiler
  • Patent number: 3931202
    Abstract: Certain 3-pyridylmethyl N-(4'-substituted-phenyl)carbamates are useful as rodenticides, e.g., in baits or tracking powders. The 4'-substituent may be --NO.sub.2, --CN, --CF.sub.3, --SO.sub.2 NH.sub.2, --SR, --SOR or --SO.sub.2 R where R is lower alkyl. Their salts can also be made and applied as rodenticides.
    Type: Grant
    Filed: June 12, 1974
    Date of Patent: January 6, 1976
    Assignee: Rohm and Haas Company
    Inventors: J. Edgar Ware, Jr., Edward E. Kilbourn, David L. Peardon
  • Patent number: 3931203
    Abstract: Novel 1-(3-pyridylmethyl)-3-(4'-substituted-phenyl or -naphthyl)-ureas and their acid addition salts. The 4'-substituent may be --NO.sub.2, --CN, --CF.sub.3, --C(O)R.sub.1, --SCN, SR.sub.2, --SO.sub.2 C.sub.6 H.sub.5 or --SO.sub.2 NR.sub.3 R.sub.4. These compounds are biologically active, and many are active rodenticides.
    Type: Grant
    Filed: April 11, 1974
    Date of Patent: January 6, 1976
    Assignee: Rohm and Haas Company
    Inventors: Edward E. Kilbourn, David L. Peardon, J. Edgar Ware
  • Patent number: RE30240
    Abstract: This invention relates to novel phosphoramidates of the formula: ##STR1## wherein R.sup.1 is (C.sub.6 -C.sub.10) aryl optionally substituted with alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, dialkylamino, haloalkyl, hydroxyalkyl, cyano, nitro, hydroxy, or halogen;R.sup.2 is hydrogen.[., alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl.].R.sup.3 is (C.sub.1 -C.sub.6) alkyl;R.sup.4 is (C.sub.3 -C.sub.4) alkyl; .Iadd.X is sulfur; .Iaddend.and.[.X,.]. Y and Z are independently oxygen or sulfur;and the agronomically acceptable metal salts and metal salt complexes thereof; to compositions containing them; and to methods of using them to control certain harmful pests, e.g. arthropods and nematodes.
    Type: Grant
    Filed: January 8, 1979
    Date of Patent: March 25, 1980
    Assignee: Rohm and Haas Company
    Inventors: Harold E. Aller, Edward E. Kilbourn, Ernest D. Weiler, William D. Weir