Patents by Inventor Edward E. Kilbourn
Edward E. Kilbourn has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).
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Patent number: 4310537Abstract: Acetyl- and carbalkoxythioureidobenzophenones having a substituted amine adjacent to the thioureido radical are disclosed as having anthelmintic and antifungal activity.Type: GrantFiled: October 7, 1977Date of Patent: January 12, 1982Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, W. David Weir
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Patent number: 4297342Abstract: Novel 3-pyridylmethyl N-(4-substituted-phenyl)thiocarbamates are disclosed. These compounds are useful as single-dose rodenticides, which have high bait acceptance.Type: GrantFiled: January 17, 1980Date of Patent: October 27, 1981Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, Ernest D. Weiler, William D. Weir
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Patent number: 4276290Abstract: This invention relates to novel anthelmintic compounds containing an arylene or divalent heterocyclic ring whose free valences are satisfied by(1) a disubstituted phosphoryl ureido or thioureido group and(2) an amino group or a substituted amido or thioamido group,to compositions containing them, and to methods of using them for the treatment of intestinal parasites in mammals and birds.Type: GrantFiled: September 6, 1979Date of Patent: June 30, 1981Assignee: Rohm and Haas CompanyInventors: W. David Weir, Edward E. Kilbourn
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Patent number: 4259330Abstract: This invention relates to novel phosphoramidates of the formula: ##STR1## wherein R.sup.1 is hydrogen, alkyl, cycloalkyl, or optionally substituted aralkyl, aryl, pyridyl, pyridylmethyl, pyridylethyl or pyrazinyl;R.sup.2 is hydrogen provided R.sup.1 is other than optionally substituted aryl; alkyl; cycloalkyl; alkoxyalkyl; alkylthioalkyl; cyanoalkyl; alkenyl; optionally substituted aralylky; or optionally substituted aryl, provided R.sup.1 is other than hydrogen;R.sup.1 and R.sup.2 taken together with the nitrogen to which they are attached form an optionally substituted morpholino or piperidino group;R.sup.3 is hydrogen, alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.4 is (C.sub.1 -C.sub.6) alkyl;R.sup.5 is (C.sub.3 -C.sub.4) alkyl; andX, Y and Z are independently oxygen or sulfur;the agronomically acceptable metal salts and metal salt complexes thereof; and to methods of using them to control nematodes.Type: GrantFiled: March 1, 1976Date of Patent: March 31, 1981Assignee: Rohm and Haas CompanyInventors: Harold E. Aller, Edward E. Kilbourn, Ernest D. Weiler, William D. Weir
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Patent number: 4241079Abstract: 2-Imino substituted isothioureidobenzene products useful as anthelmintics and fungicides are disclosed. The products may be prepared by several different methods including treating a 2-iminothioureidobenzene with a base and either an organic halide, a diester of sulfuric acid or a diester of sulfurous acid or treating a 2-aminoisothioureidobenzene with an appropriately substituted aldehyde.Type: GrantFiled: May 4, 1978Date of Patent: December 23, 1980Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, W. David Weir
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Patent number: 4234575Abstract: This invention relates to novel anthelmintic compounds containing an arylene or divalent heterocyclic ring whose free valences are satisfied by(1) a disubstituted phosphoryl ureido or thioureido group and(2) an amino group or a substituted amido or thioamido group,to compositions containing them, and to methods of using them for the treatment of intestinal parasites in mammals and birds.Type: GrantFiled: January 31, 1979Date of Patent: November 18, 1980Assignee: Rohm and Haas CompanyInventors: W. David Weir, Edward E. Kilbourn
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Patent number: 4233289Abstract: Novel 3-pyridylmethyl N-(4-substituted-phenyl)thiocarbamates are disclosed. These compounds are useful as single-dose rodenticides, which have high baitacceptance.Type: GrantFiled: January 31, 1979Date of Patent: November 11, 1980Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, Ernest D. Weiler, William D. Weir
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Patent number: 4183921Abstract: This invention relates to novel anthelmintic compounds containing an arylene or divalent heterocyclic ring whose free valences are satisfied by(1) a disubstituted phosphoryl ureido or thioureido group and(2) an amino group or a substituted amido or thioamido group,to compositions containing them, and to methods of using them for the treatment of intestinal parasites in mammals and birds.Type: GrantFiled: October 17, 1977Date of Patent: January 15, 1980Assignee: Rohm and Haas CompanyInventors: W. David Weir, Edward E. Kilbourn
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Patent number: 4156780Abstract: Novel 3-pyridylmethyl N-(4-substituted-phenyl)thiocarbamates are disclosed. These compounds are useful as single-dose rodenticides, which have high bait acceptance.Type: GrantFiled: June 30, 1975Date of Patent: May 29, 1979Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, Ernest D. Weiler, William D. Weir
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Patent number: 4139614Abstract: This invention relates to novel anthelmintic compositions containing as the essential active ingredient, a compound of the formula: ##STR1## wherein R.sup.1 is cylcoalkyl, or optionally substituted aralkyl, aryl, pyridyl, or pyrazinyl;R.sup.2 is hydrogen, alkyl, cycloalkyl, alkoxyalkyl, alkylthioalkyl, cyanoalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.1 and R.sup.2 taken together with the nitrogen atom to which they are attached form an optionally substituted morpholino or piperidino group;R.sup.3 is hydrogen, alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.4 is alkoxy, haloalkoxy, dialkylamino, alkylthio, phenoxy or phenylthio; andR.sup.5 is alkyl, alkoxy, haloalkoxy, dialkylamino, alkylthio, phenyl, phenoxy or phenylthio; andX is oxygen or sulfur;And pharmaceutically acceptable metal salts and metal salt complexes thereof, and to methods of employing them in the treatment of intestinal parasites in animals, e.g. mammals, fish, and birds.Type: GrantFiled: March 1, 1976Date of Patent: February 13, 1979Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, Ernest Weiler, William D. Weir
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Patent number: 4087521Abstract: This invention relates to novel phosphoramidates of the formula: ##STR1## wherein R.sup.1 is (C.sub.6 -C.sub.10) aryl optionally substituted with alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, dialkylamino, haloalkyl, hydroxyalkyl, cyano, nitro, hydroxy, or halogen;R.sup.2 is hydrogen, alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.3 is (C.sub.1 -C.sub.6) alkyl;R.sup.4 is (C.sub.3 -C.sub.4) alkyl; andX, y and Z are independently oxygen or sulfur;And the agronomically acceptable metal salts and metal salt complexes thereof; to compositions containing them; and to methods of using them to control certain harmful pests, e.g. arthropods and nematodes.Type: GrantFiled: March 1, 1976Date of Patent: May 2, 1978Assignee: Rohm and Haas CompanyInventors: Harold E. Aller, Edward E. Kilbourn, Ernest D. Weiler, William D. Weir
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Patent number: 4076809Abstract: This invention relates to novel anthelmintic compounds containing an arylene or divalent heterocyclic ring whose free valences are satisfied by1. a disubstituted phosphoryl ureido or thioureido group and2. an amino group or a substituted amido or thioamido group,To compositions containing them, and to methods of using them for the treatment of intestinal parasites in mammals and birds.Type: GrantFiled: October 28, 1975Date of Patent: February 28, 1978Assignee: Rohm and Haas CompanyInventors: W. David Weir, Edward E. Kilbourn
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Patent number: 4075345Abstract: Rodenticidal compositions containing as the active ingredient novel 1-(3-pyridylmethyl)-3-(4'-substituted-phenyl or -naphthyl)ureas and their acid addition salts. The 4'-substituent may be nitro, cyano, trifluoromethyl, butyryl, thiocyano, alkylthio, phenylsulfonyl or diethylsulfonamide.Type: GrantFiled: April 11, 1974Date of Patent: February 21, 1978Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, David L. Peardon, J. Edgar Ware
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Patent number: 4060636Abstract: Acetyl- and carbalkoxythioureidobenzophenones having a substituted amine adjacent to the thioureido radical are disclosed as having anthelmintic and antifungal activity.Type: GrantFiled: June 10, 1976Date of Patent: November 29, 1977Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, W. David Weir
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Patent number: 4033972Abstract: 3-Pyridylmethyl-(N-substituted-phenyl-N-hydrocarbyl)carbamates. They are useful as rodenticides.Type: GrantFiled: September 9, 1975Date of Patent: July 5, 1977Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, Ernest D. Weiler
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Patent number: 3994905Abstract: Novel 1-(3-pyridylmethyl)-3-(4'-substituted-phenyl or -naphthyl)-ureas and their acid addition salts. The 4'-substituent may be -NO.sub.2, -CN, -CF.sub.3, -C(O)R.sub.1, -SCN, SR.sub.2, -SO.sub.2 C.sub.6 H.sub.5 or -SO.sub.2 NR.sub.3 R.sub.4. These compounds are biologically active, and many are active rodenticides.Type: GrantFiled: October 16, 1975Date of Patent: November 30, 1976Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, David L. Peardon, J. Edgar Ware
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Patent number: 3966947Abstract: 3-Pyridylmethyl N-(4'-substitutedmercaptophenyl) carbamates and their acid salts and metal salt complexes useful as a rodenticide.Type: GrantFiled: October 3, 1975Date of Patent: June 29, 1976Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, Ernest D. Weiler
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Patent number: 3931202Abstract: Certain 3-pyridylmethyl N-(4'-substituted-phenyl)carbamates are useful as rodenticides, e.g., in baits or tracking powders. The 4'-substituent may be --NO.sub.2, --CN, --CF.sub.3, --SO.sub.2 NH.sub.2, --SR, --SOR or --SO.sub.2 R where R is lower alkyl. Their salts can also be made and applied as rodenticides.Type: GrantFiled: June 12, 1974Date of Patent: January 6, 1976Assignee: Rohm and Haas CompanyInventors: J. Edgar Ware, Jr., Edward E. Kilbourn, David L. Peardon
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Patent number: 3931203Abstract: Novel 1-(3-pyridylmethyl)-3-(4'-substituted-phenyl or -naphthyl)-ureas and their acid addition salts. The 4'-substituent may be --NO.sub.2, --CN, --CF.sub.3, --C(O)R.sub.1, --SCN, SR.sub.2, --SO.sub.2 C.sub.6 H.sub.5 or --SO.sub.2 NR.sub.3 R.sub.4. These compounds are biologically active, and many are active rodenticides.Type: GrantFiled: April 11, 1974Date of Patent: January 6, 1976Assignee: Rohm and Haas CompanyInventors: Edward E. Kilbourn, David L. Peardon, J. Edgar Ware
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Patent number: RE30240Abstract: This invention relates to novel phosphoramidates of the formula: ##STR1## wherein R.sup.1 is (C.sub.6 -C.sub.10) aryl optionally substituted with alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, dialkylamino, haloalkyl, hydroxyalkyl, cyano, nitro, hydroxy, or halogen;R.sup.2 is hydrogen.[., alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl.].R.sup.3 is (C.sub.1 -C.sub.6) alkyl;R.sup.4 is (C.sub.3 -C.sub.4) alkyl; .Iadd.X is sulfur; .Iaddend.and.[.X,.]. Y and Z are independently oxygen or sulfur;and the agronomically acceptable metal salts and metal salt complexes thereof; to compositions containing them; and to methods of using them to control certain harmful pests, e.g. arthropods and nematodes.Type: GrantFiled: January 8, 1979Date of Patent: March 25, 1980Assignee: Rohm and Haas CompanyInventors: Harold E. Aller, Edward E. Kilbourn, Ernest D. Weiler, William D. Weir