Patents by Inventor Jean J. Gallay

Jean J. Gallay has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4762830
    Abstract: The invention relates to novel 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives of the general formula I ##STR1## wherein X is oxygen or sulfur;R.sub.1 is C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy, C.sub.3 -C.sub.6 cycloalkyl or allyl;R.sub.2 is C.sub.1 -C.sub.6 alkyl or allyl;R.sub.3 is an unsubstituted or substituted five-membered azole ring which is bound through carbon and is selected from the group consisting of benzimadazole, benzoxazole, benzothiazole, imidazole, oxazole, thiazole, oxadiazole, thiadiazole and triazole; andR.sub.4 and R.sub.5 are each independently of the other hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkoxy or C.sub.1 -C.sub.6 haloalkoxy;and to the tautomers and salts thereof, as anthelmintic compounds. Together with suitable carriers and further assistants, these compounds may be used in particular for controlling helminths which are parasites of animals.
    Type: Grant
    Filed: February 13, 1986
    Date of Patent: August 9, 1988
    Assignee: Ciba-Geigy Corporation
    Inventors: Elmar Sturm, Jean J. Gallay, Haukur Kristinsson, Georg Pissiotas
  • Patent number: 4753940
    Abstract: The invention relates to novel phenylcarbamoylbarbituric acid derivatives of the general formula ##STR1## wherein R.sub.1 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.3 alkoxy, allyl or C.sub.3 -C.sub.6 cycloalkyl,R.sub.2 is C.sub.1 -C.sub.4 alkyl or allyl,R.sub.3 is an unsubstituted or substituted heteroaromatic 6-membered ring which contains 2 or 3 nitrogen atoms, or is an unsubstituted or substituted heteroaromatic 6-membered ring which is fused to a benzene ring and which contains 1 to 3 nitrogen atoms,R.sub.4 and R.sub.5 are each independently of the other hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy or C.sub.1 -C.sub.3 haloalkyl andX is an oxygen or sulfur atom,and to the tautomers and salts thereof.These compounds may be used for controlling helminths which are parasites of animals.
    Type: Grant
    Filed: February 7, 1986
    Date of Patent: June 28, 1988
    Assignee: Ciba-Geigy Corporation
    Inventors: Elmar Sturm, Jean J. Gallay, Georg Pissiotas
  • Patent number: 4748178
    Abstract: Novel phenylcarbamoylbarbituric acid derivatives of the general formula I ##STR1## and tautomeric forms and salts thereof in which R.sub.1 and R.sub.2 independently of one another are C.sub.1 -C.sub.5 -alkyl, C.sub.1 -C.sub.3 -alkoxy, C.sub.3 -C.sub.6 -cycloalkyl, allyl or phenyl; R.sub.3 is substituted or unsubstituted pyridyl as herein defined; and X is oxygen or sulfur; they possess anthelmintic activity. The active substances can be employed in conjunction with suitable carriers and further adjuncts for controlling zooparasitic helminths.
    Type: Grant
    Filed: February 13, 1986
    Date of Patent: May 31, 1988
    Assignee: Ciba-Geigy Corporation
    Inventors: Urs Burckhardt, Jean J. Gallay, Manfred Kuhne
  • Patent number: 4670441
    Abstract: The invention relates to novel 5-phenylcarbamoylthiobarbituric acid derivatives of the general formula ##STR1## wherein R.sub.1 and R.sub.2 are each independently C.sub.1 -C.sub.5 alkyl or methoxy,R.sub.3 is unsubstituted phenyl, unsubstituted pyridyl, or phenyl which is substituted by 1 to 3 identical or different members selected from the group consisting of C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.4 cyanoalkyl, halogen, nitro and C.sub.1 -C.sub.5 haloalkyl containing 1 to 5 halogen atoms, or is pyridyl which is substituted by 1 to 3 identical or different members selected from the group consisting of C.sub.1 -C.sub.5 alkyl, halogen, nitro and C.sub.1 -C.sub.5 haloalkyl containing 1 to 5 halogen atoms andR.sub.4 and R.sub.5 are each independently hydrogen, halogen, C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.2 haloalkyl containing 1 to 3 halogen atoms, or are C.sub.1 -C.sub.3 -alkoxy or nitro,and to the tautomers and salts thereof, as anthelmintics.
    Type: Grant
    Filed: July 5, 1985
    Date of Patent: June 2, 1987
    Assignee: Ciba-Geigy Corporation
    Inventors: Manfred Kuhne, Jean J. Gallay
  • Patent number: 4602912
    Abstract: The invention relates to a composition for protecting keratinous material, in particular woollen textiles, from attack by pests that feed on keratin, in particular moth and beetle larvae, which composition contains, as active ingredient combination, a specifically substituted 5-(pyridyloxyphenylcarbamoyl)barbituric acid or a salt thereof and a synthetic pyrethroid, as well as to a process comprising the use of this active ingredient combination for providing said material with a protective finish against attack by pests that feed on keratin.
    Type: Grant
    Filed: June 24, 1985
    Date of Patent: July 29, 1986
    Assignee: Ciba-Geiby Corporation
    Inventors: Bernardo de Sousa, Urs Burckhardt, Jean J. Gallay, Manfred Kuhne, Ernst Beriger, Dieter Reinehr
  • Patent number: 4511567
    Abstract: The invention relates to a process for the manufacture of novel benzazole derivatives of the formula I ##STR1## in which R.sub.1 represents an optionally 4-substituted piperazino group or a group of the formula R.sub.2 --alk--X.sub.2 --,R.sub.2 represents optionally esterified carboxy or represents hydroxymethyl,alk represents lower alkylene or lower alkylidene,X.sub.1 and X.sub.2, independently of one another, each represents oxygen or sulphur,Ph represents 1,2-phenylene optionally substituted as well as by the group R.sub.1 --C(.dbd.X.sub.1)--NH--,X.sub.3 represents oxygen, sulphur or optionally substituted imino, andR.sub.3 represents optionally fluorine-substituted lower alkyl or cycloalkyl,and their salts.The compounds of the formula I, which have proved to be excellent micro- and macrofilaricides and schistosomacides, are manufactured according to methods known per se.
    Type: Grant
    Filed: September 16, 1982
    Date of Patent: April 16, 1985
    Assignee: Ciba-Geigy Corporation
    Inventors: Jean J. Gallay, Ernst Schweizer
  • Patent number: 4428957
    Abstract: The isothiocyanobenzothiazole derivative of the formula ##STR1## and also salts thereof nontoxic to warm-blooded animals have, besides generally good anthelmintic properties, especially a particularly pronounced action against filariasis, schistosomiasis and gastrointestinal helminths in warm-blooded organisms and equally against liver flukes in sheep. The active substance, together with suitable carriers and additives, is administered perorally or via the abomasum, in the form of solutions, emulsions, suspensions, powders, tablets, boluses and capsules.
    Type: Grant
    Filed: May 4, 1981
    Date of Patent: January 31, 1984
    Assignee: Ciba-Geigy Corporation
    Inventors: Joseph C. Boray, Jean J. Gallay, Gedeon Sarasin
  • Patent number: 4205077
    Abstract: Benzimidazole derivatives of the formula ##STR1## in which R and R.sub.1 independently of one another are each hydrogen, an alkanoyl group having 1 to 4 carbon atoms, an alkoxycarbonyl group having 1 to 4 carbon atoms, an alkylsulphonyl group having 1 to 4 carbon atoms, a benzoyl group, a phenylsulphonyl group or a p-methylphenylsulphonyl group; R.sub.2 and R.sub.4 independently of one another are each hydrogen, halogen or a methyl group, R.sub.3 is hydrogen, halogen, a methyl group or a methoxy group; X is oxygen or sulphur; Y is halogen, an alkyl group having 1 to 4 carbon atoms, an alkoxy group having 1 to 4 carbon atoms, a methylthio group, a methylsulphinyl group, a methylsulphonyl group, a trifluoromethyl group, a nitro group, a hydroxyl group, a cyano group or an acetyl group; and m is 0, 1, 2 or 3; and if one of the two radicals R or R.sub.1 is hydrogen, the position of the other of these radicals on the N atoms cannot be clearly established, including, when at least one of the two radicals R or R.
    Type: Grant
    Filed: April 10, 1978
    Date of Patent: May 27, 1980
    Assignee: Ciba-Geigy Corporation
    Inventors: Ernst Aufderhaar, Jean J. Gallay, Manfred Kuhne, Alfred Meyer, Oswald Rechsteiner, Max Schellenbaum, Jean-Paul Fumeaux