Patents by Inventor Rahul Kaduskar

Rahul Kaduskar has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Publication number: 20240389591
    Abstract: The present invention relates to one crystalline form A of methyl 2-[2-[2-bromo-4-fluoro-5-[3-methyl-2,6-dioxo-4-(trifluoromethyl)pyrimidin-1-yl]phenoxy]phenoxy]-2-methoxy-acetate, a process for the production of this crystalline form and formulations for plant protection comprising such form A.
    Type: Application
    Filed: August 19, 2022
    Publication date: November 28, 2024
    Inventors: Rahul Kaduskar, Martin Viertelhaus, Sunil Kolse, Desislava Slavcheva Petkova, Tobias Seiser, Roland Goetz, Harish Shinde, Henning Urch, Ricardo Hugo Pavon Romero
  • Publication number: 20240262816
    Abstract: The present invention relates to a method for preparing an enantiomerically enriched form of 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one of the formula (I) by hydrogenation of 2-[2-(2-chlorothia-201-5-yl)-2-oxo-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one (1) in the presence of a chiral transition metal catalyst.
    Type: Application
    Filed: March 25, 2022
    Publication date: August 8, 2024
    Inventors: Martin John McLaughlin, Christopher Koradin, Rahul Kaduskar, Harish Shinde, Roland Goetz
  • Publication number: 20240116916
    Abstract: The present invention relates to a method for preparing 2-[2-(2-chlorothiazol-5-yl)-2- hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one or a tautomer thereof or enantiomerically enriched forms thereof, to 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one or a tautomer thereof or enantiomerically enriched forms thereof, and to the use thereof as intermediate in the preparation of 2,3-dihydrothiazolo[3,2-a]pyrimidinium compounds, specifically of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo [3,2-a]pyrimidin-4-ium-5-olate and enantiomerically enriched forms thereof.
    Type: Application
    Filed: January 21, 2022
    Publication date: April 11, 2024
    Inventors: Martin John McLaughlin, Christopher Koradin, Rahul Kaduskar, Harish Shinde, Roland Gotez, Guillaume Michel Jacques Garivet
  • Publication number: 20240101516
    Abstract: The presently claimed invention relates to a process for the preparation of mono-, di-, tri-, fluoro arylamide or hetroarylamide.
    Type: Application
    Filed: January 17, 2022
    Publication date: March 28, 2024
    Inventors: Rahul Kaduskar, Kailaskumar Borate, Suyog Adhav, Saravanan Thirunavukkarasu, Harish Shinde, Roland Goetz
  • Publication number: 20240101547
    Abstract: The present invention relates to a method for preparing 2-[2-(2-chlorothiazol-5-yl)-2-oxo-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one or a tautomer thereof, to 2-[2-(2-chlorothiazol-5-yl)-2-oxo-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one or a tautomer thereof and to its use as intermediate in the preparation of 2,3-dihydrotheiazolo [3,2-a]pyrimidinium compounds, and specifically of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo [3,2-a]pyrimidin-4-ium-5-olate and enantiomerically enriched forms thereof.
    Type: Application
    Filed: January 21, 2022
    Publication date: March 28, 2024
    Inventors: Christopher Koradin, Martin John McLaughlin, Roland Goetz, Rahul Kaduskar, Harish Shinde, Guillaume Michel Jacques Garivet
  • Publication number: 20240101575
    Abstract: The present invention relates to a method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate.
    Type: Application
    Filed: January 21, 2022
    Publication date: March 28, 2024
    Inventors: Christopher Koradin, Martin John McLaughlin, Roland Goetz, Rahul Kaduskar, Harish Shinde
  • Publication number: 20240051929
    Abstract: The present invention relates to a process for the preparation 2-chloro-1-(2-chlorothiazol-5-yl)ethanone.
    Type: Application
    Filed: September 28, 2020
    Publication date: February 15, 2024
    Inventors: Harish Shinde, Rahul Kaduskar, Christopher Koradin, Martin John McLaughlin, Roland Goetz, Sunil Khamkar
  • Publication number: 20230416273
    Abstract: The present invention relates to a method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate.
    Type: Application
    Filed: January 21, 2022
    Publication date: December 28, 2023
    Inventors: Christopher Koradin, Martin John McLaughlin, Harish Shinde, Rahul Kaduskar, Ronald Goetz, Guillaaume Michel Jaques Garivet
  • Publication number: 20230322693
    Abstract: The present invention relates to a process for the preparation 2-chloro-1-(2-chlorothiazol-5-yl)ethanone.
    Type: Application
    Filed: September 28, 2021
    Publication date: October 12, 2023
    Inventors: Christopher Koradin, Harish Shinde, Martin John McLaughlin, Rahul Kaduskar, Philipp M. Staehle, Roland Goetz, Sunil Khamkar
  • Publication number: 20230100114
    Abstract: The presently claimed invention relates to a process for the preparation of di-, tri-, or tetra fluoroarylamine by reacting polyfluorinated aryl chlorides with ammonia in the presence of a base, a metal catalyst and a ligand. Di-, tri-, tetrafluoroarylamines are valuable intermediates and find application in several areas, mainly in epoxy polymers, colorants, dyes, polyurethanes, agrochemicals and pharmaceutical active agents.
    Type: Application
    Filed: April 6, 2021
    Publication date: March 30, 2023
    Inventors: Kailaskumar Borate, Saravanan Thirunavukkarasu, Rahul Kaduskar, Harish Shinde, Roland Goetz
  • Patent number: 9340506
    Abstract: Acetamide derivatives, their stereoisomers, tautomers, prodrugs, pharmaceutically acceptable salts, polymorphs, solvates and formulations thereof for the prophylaxis, management, treatment, control of progression, or adjunct treatment of diseases and/or medical conditions where the activation of glucokinase would be beneficial, are disclosed. The disclosure also provides process of preparation of these acetamide derivatives.
    Type: Grant
    Filed: February 17, 2012
    Date of Patent: May 17, 2016
    Assignee: ADVINUS THERAPEUTICS LIMITED
    Inventors: Debnath Bhuniya, Anil Deshpande, Sachin Kandalkar, Balasaheb Kobal, Santosh Kurhade, Vinod Vyavahare, Rahul Kaduskar
  • Publication number: 20120214735
    Abstract: Acetamide derivatives, their stereoisomers, tautomers, prodrugs, pharmaceutically acceptable salts, polymorphs, solvates and formulations thereof for the prophylaxis, management, treatment, control of progression, or adjunct treatment of diseases and/or medical conditions where the activation of glucokinase would be beneficial, are disclosed. The disclosure also provides process of preparation of these acetamide derivatives.
    Type: Application
    Filed: February 17, 2012
    Publication date: August 23, 2012
    Applicant: Advinus Therapeutics Limited
    Inventors: Debnath Bhuniya, Anil Deshpande, Sachin Kandalkar, Balasaheb Kobal, Santosh Kurhade, Vinod Vyavahare, Rahul Kaduskar