Patents by Inventor Alain A. Champseix

Alain A. Champseix has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4505916
    Abstract: Compounds, useful as medicaments, of the formula: ##STR1## in which R is hydrogen, alkyl, alkenyl or arylalkyl, R.sub.1 is hydrogen, alkyl or alkenyl, R.sub.2 is hydrogen, alkyl, arylalkyl, phenyl, pyridyl, thienyl or substituted phenyl, X is hydrogen, halogen, alkyl, alkoxy, alkylthio, trifluoromethyl, nitro, amino or amino substituted by one or two alkyl groups, and A represents a CO or CH.sub.2 group.
    Type: Grant
    Filed: September 29, 1982
    Date of Patent: March 19, 1985
    Assignee: Pharmindustrie
    Inventors: Alain A. Champseix, Gerard R. Le Fur, Christian L. A. Renault
  • Patent number: 4493838
    Abstract: Compounds useful as medicaments, particularly useful as a hypnotic, an anticonvulsant and for the treatment of anxiety states and psychoneurotic states of the formula: ##STR1## in which X is hydrogen, halogen, alkyl containing 1 to 4 carbon atoms, alkoxy containing 1 to 4 carbon atoms or alkylthio containing 1 to 4 carbon atoms, one of the substituents R.sub.1 and R.sub.2 is hydrogen, alkyl containing 1 to 4 carbon atoms, phenyl or phenyl substituted by halogen, alkyl containing 1 to 4 carbon atoms, alkoxy containing 1 to 4 carbon atoms, alkylthio containing 1 to 4 carbon atoms, trifluoromethyl, nitro, unsubstituted amino or amino substituted by one or two alkyl containing 1 to 2 carbon atoms, and the other of the substituents R.sub.1 and R.sub.2 is a group of the formula: ##STR2## in which n is 1, 2 or 3 and R is hydrogen or alkyl containing 1 to 4 carbon atoms.
    Type: Grant
    Filed: September 29, 1982
    Date of Patent: January 15, 1985
    Assignee: Pharmindustrie
    Inventors: Alain A. Champseix, Gerard R. Le Fur
  • Patent number: 4433150
    Abstract: Compounds, useful as medicaments, of the formula: ##STR1## in which R is hydrogen, alkyl, alkenyl or arylalkyl, R.sub.1 is hydrogen, alkyl or alkenyl, R.sub.2 is hydrogen, alkyl, arylalkyl, phenyl, pyridyl, thienyl or substituted phenyl, X is hydrogen, halogen, alkyl, alkoxy, alkylthio, trifluoromethyl, nitro, amino or amino substituted by one or two alkyl groups, and A represents a CO or CH.sub.2 group.
    Type: Grant
    Filed: December 2, 1980
    Date of Patent: February 21, 1984
    Assignee: Pharmindustrie
    Inventors: Alain A. Champseix, Gerard R. Le Fur, Christian L. A. Renault
  • Patent number: 4405789
    Abstract: Compounds useful as medicaments, of the formula: ##STR1## in which X is hydrogen, halogen, alkyl containing 1 to 4 carbon atoms, alkoxy containing 1 to 4 carbon atoms or alkylthio containing 1 to 4 carbon atoms, one of the substituents R.sub.1 and R.sub.2 is hydrogen, alkyl containing 1 to 4 carbon atoms, phenyl or phenyl substituted by halogen, alkyl containing 1 to 4 carbon atoms, alkoxy containing 1 to 4 carbon atoms, alkylthio containing 1 to 4 carbon atoms, trifluoromethyl, nitro, unsubstituted amino or amino substituted by one or two alkyl containing 1 to 2 carbon atoms, and the other of the substituents R.sub.1 and R.sub.2 is a group of the formula: ##STR2## in which n is 1, 2 or 3 and R is hydrogen or alkyl containing 1 to 4 carbon atoms.
    Type: Grant
    Filed: February 24, 1981
    Date of Patent: September 20, 1983
    Assignee: Pharmindustrie
    Inventors: Alain A. Champseix, Gerard R. Le Fur
  • Patent number: 4299835
    Abstract: Pharmaceutical preparations containing as active ingredient a compound having the formula: ##STR1## wherein R represents hydrogen, alkyl having 1 to 4 carbon atoms or alkenyl having 2 to 4 carbon atoms; andX represents hydrogen, alkyl, alkoxy or alkylthio, the alkyl groups of each containing 1 to 4 carbon atoms, halogen (chlorine, fluorine, bromine or iodine), trifluoromethyl, nitro, hydroxy, amino or amino substituted by one or two alkyl groups or by acyl or alkylsulphonyl, the alkyl groups of each containing 1 to 4 carbon atoms, which are particularly advantageous for the treatment of pathological states caused by a disturbance in the functioning of the serotoninergical systems in mammals. These preparations may also be used as anxiolytics.
    Type: Grant
    Filed: November 24, 1980
    Date of Patent: November 10, 1981
    Assignee: Pharmindustrie
    Inventors: Alain A. Champseix, Claude G. A. Gueremy, Gerard R. Le Fur
  • Patent number: 4294841
    Abstract: A drug useful as antiarhythmic, antidepressant and anxiolytic containing as an active agent a compound of the formula ##STR1## wherein X and Y are the same or different and represent hydrogen or halogen atoms, or 1-4C alkyl groups, 1-4C alkoxy groups, 1-4C alkylthio groups, CF.sub.3, OH, NH.sub.2, 1-4C monoalkylamino or amino groups substituted by a 1-4C alkylsulfonyl group, a 1-5C alkylcarbonyl group or an aroyl group and A is a CO, CHOH or CH.sub.2 group, or a salt of said compound with a pharmaceutically acceptable acid, is disclosed together with methods for the preparation thereof and its use in human therapy.
    Type: Grant
    Filed: November 27, 1979
    Date of Patent: October 13, 1981
    Assignee: Pharmindustrie
    Inventors: Alain A. Champseix, Gerard R. Le Fur
  • Patent number: 4237139
    Abstract: Pharmaceutical preparations containing as active ingredient a compound having the formula: ##STR1## wherein R represents hydrogen, alkyl having 1 to 4 carbon atoms or alkenyl having 2 to 4 carbon atoms; andX represents hydrogen, alkyl, alkoxy or alkylthio, the alkyl groups of each containing 1 to 4 carbon atoms, halogen (chlorine, fluorine, bromine or iodine), trifluoromethyl, nitro, hydroxy, amino or amino substituted by one or two alkyl groups or by acyl or alkylsulphonyl, the alkyl groups of each containing 1 to 4 carbon atoms, which are particularly advantageous for the treatment of pathological states caused by a disturbance in the functioning of the serotoninergical systems in mammals. These preparations may also be used as anxiolytics.
    Type: Grant
    Filed: December 12, 1978
    Date of Patent: December 2, 1980
    Assignee: Pharmindustrie
    Inventors: Alain A. Champseix, Claude G. A. Gueremy, Gerard R. Le Fur