Patents by Inventor Franco Pellacini

Franco Pellacini has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Diastereoselective process for the preparation of intermediates useful for the synthesis of peptide derivatives
    Patent number: 5157143
    Abstract: A diastereoselective process for the preparation of compounds of formula ##STR1## (wherein R and R.sub.1 have the meanings reported in the specification and the asterisks show the asymmetric carbon atoms) starting from the corresponding N-protected 2-amino-3-aryl-propan-1-ol is described.The compounds of formula I are intermediates useful for the synthesis of pharmacologically active peptides.
    Type: Grant
    Filed: May 11, 1989
    Date of Patent: October 20, 1992
    Assignee: Zambon Group S.p.A.
    Inventors: Franco Pellacini, Dario Chiarino, Angelo Carenzi
  • Peptides with pharmaceutical activity
    Patent number: 5145872
    Abstract: Compounds of the formula ##STR1## wherein R, R.sub.1, R.sub.2, R.sub.3, R.sub.4, R.sub.5 and n have the meanings reported in the specification, processes for their preparation and pharmaceutical compositions containing them as active ingredient are described.The compounds of formula I are inhibitor of enzymatic systems and they are useful in pharmaceutical field.
    Type: Grant
    Filed: March 15, 1989
    Date of Patent: September 8, 1992
    Assignee: Zambon Group, S.p.A.
    Inventors: Dario Chiarino, Angelo Carenzi, Davide Della Bella, Franco Pellacini
  • Peptides with pharmaceutical activity
    Patent number: 5028626
    Abstract: Compounds of formula ##STR1## wherein R.sub.1, R.sub.2, R.sub.3, R.sub.4, and n have the meanings reported in the specification, processes for their preparation and pharmaceutical compositions containing them as active ingredient are described. The compounds of formula I are inhibitors of enzymatic systems and they are useful in pharmaceutical field.
    Type: Grant
    Filed: March 15, 1989
    Date of Patent: July 2, 1991
    Assignee: Zambon Group S.p.A.
    Inventors: Dario Chiarino, Angelo Carenzi, Davide Della Bella, Franco Pellacini
  • Derivatives of thiazolidine-4-carboxylic acid having pharmacological activity
    Patent number: 4952596
    Abstract: Compounds of the formula ##STR1## wherien R, R.sub.1, R.sub.2 and Y have the meanings mentioned in the description, processes for their preparation and their use in the pharmaceutical field are described.The compounds of formula I are endowed with antipyretic, anti-inflammatory, mucolitic and analgesic activity together with good gastric tolerability.In addition, the compounds of formula I are active in the treatment of ischemic or reperfusion syndromes.
    Type: Grant
    Filed: December 21, 1988
    Date of Patent: August 28, 1990
    Assignee: Zambon S.p.A.
    Inventors: Davide Della Bella, Angelo Carenzi, Dario Chiarino, Franco Pellacini
  • Pharmaceutically useful derivatives of thiazolidine-4-carboxylic acid
    Patent number: 4840936
    Abstract: Compounds of formula ##STR1## in which R, R.sub.1 and Y have the meanings shown in the description, their preparation by condensing an aldehyde or a ketone with cysteine or a derivative thereof and their use in the pharmaceutical field.The compounds of formula I possess antipyretic, anti-inflammatory, mucolytic and analgesic activity together with a low capacity to cause gastric injuries.The compounds of formula I, furthermore, are particularly useful in the treatment of ischemia and reperfusion syndromes.
    Type: Grant
    Filed: July 13, 1987
    Date of Patent: June 20, 1989
    Assignee: Zambon S.p.A.
    Inventors: Davide Della Bella, Angelo Carenzi, Dario Chiarino, Franco Pellacini