Patents by Inventor Jean-Marie Derocq

Jean-Marie Derocq has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Slimming cosmetic composition containing a substance inducing the production of IL-6
    Patent number: 8628770
    Abstract: This invention relates to a slimming cosmetic composition containing at least one compound inducing the production of IL-6 by the adipocytes in the form of a mixture with an NPY antagonist and/or an ?2 antagonist and with an excipient for a cosmetic preparation.
    Type: Grant
    Filed: October 28, 2008
    Date of Patent: January 14, 2014
    Assignee: Sanofi
    Inventors: Pierre Casellas, Jean-Marie Derocq, Joelle Guesnet
  • Pyridoindolone derivatives substituted in the 3-position by a phenyl, their preparation and their application in therapeutics
    Patent number: 8012991
    Abstract: The present disclosure relates to pyridoindolone derivatives of general formula (I): to processes for preparing the same and to their use in therapeutics.
    Type: Grant
    Filed: May 12, 2008
    Date of Patent: September 6, 2011
    Assignee: Sanofi-Aventis
    Inventors: Bernard Bourrie, Pierre Casellas, Paola Ciapetti, Jean-Marie Derocq, Samir Jegham, Yvette Muneaux, Camille-Georges Wermuth
  • Pyridoindolone derivatives substituted in the 3-position by a heterocyclic group, their preparation and their application in therapeutics
    Patent number: 7816368
    Abstract: The present disclosure relates to pyridoindolone derivatives of general formula (I): in which R1 to R5 are as defined in the specification, to processes for preparing said derivatives, and to methods of use thereof.
    Type: Grant
    Filed: October 16, 2008
    Date of Patent: October 19, 2010
    Assignee: sanofi-aventis
    Inventors: Bernard Bourrie, Pierre Casellas, Jean-Marie Derocq, Samir Jegham, Yvette Muneaux
  • SLIMMING COSMETIC COMPOSITION CONTAINING A SUBSTANCE INDUCING THE PRODUCTION OF IL-6
    Publication number: 20090123455
    Abstract: This invention relates to a slimming cosmetic composition containing at least one compound inducing the production of IL-6 by the adipocytes in the form of a mixture with an NPY antagonist and/or an ?2 antagonist and with an excipient for a cosmetic preparation.
    Type: Application
    Filed: October 28, 2008
    Publication date: May 14, 2009
    Applicant: SANOFI-AVENTIS
    Inventors: Pierre CASELLAS, Jean-Marie DEROCQ, Joelle GUESNET
  • Pharmaceutical combinations based on pyridoindolone derivatives and anticancer agents
    Patent number: 7524857
    Abstract: The invention relates to the combination of compounds of formula: with one or more anticancer agents.
    Type: Grant
    Filed: April 26, 2002
    Date of Patent: April 28, 2009
    Assignee: Sanofi-Aventis
    Inventors: Bernard Bourrie, Pierre Casellas, Jean-Marie Derocq
  • Pyridoindolone Derivatives Substituted in the 3-position by a Heterocyclic Group, Their Preparation and Their Application in Therapeutics
    Publication number: 20090042924
    Abstract: The present disclosure relates to pyridoindolone derivatives of general formula (I): in which R1 to R5 are as defined in the specification, to processes for preparing said derivatives, and to methods of use thereof.
    Type: Application
    Filed: October 16, 2008
    Publication date: February 12, 2009
    Applicant: SANOFI-AVENTIS
    Inventors: Bernard BOURRIE, Pierre CASELLAS, Jean-Marie DEROCQ, Samir JEGHAM, Yvette MUNEAUX
  • Pyridoindolone derivatives substituted in the 3-position by a heterocyclic group, their preparation and their application in therapeutics
    Patent number: 7456193
    Abstract: The present invention relates to pyridoindolone derivatives substituted in the 3-position by a heterocyclic group of general formula (I): in which: R1 represents a hydrogen atom or a (C1-C4)alkyl group; R2 represents a hydrogen atom or a (C1-C4)alkyl group; R3 represents a thienyl mono- or polysubstituted by a methyl group; or a monocyclic or bicyclic heterocyclic radical chosen from: a pyridyl, an N-oxidopyridinio, a pyrazolyl, an (N-phenyl)pyrazolyl, an (N-halophenyl)pyrazolyl, a furyl, an indolyl, an (N-benzyl)indolyl, an (N-halobenzyl)indolyl, a benzothienyl or a benzofuryl, the said radicals being unsubstituted or substituted one or more times by a halogen atom or a methyl or methoxy group; R4 and R5 are identical or different and each independently represent a hydrogen or halogen atom or a hydroxyl, hydroxymethyl, (C1-C4)alkyl, trifluoromethyl, C1-C4)alkoxy, (C1-C4)alkoxycarbonyl or cyano group. Preparation process and application in therapeutics.
    Type: Grant
    Filed: April 19, 2005
    Date of Patent: November 25, 2008
    Assignee: Sanofi-Aventis
    Inventors: Bernard Bourrie, Pierre Casellas, Jean-Marie Derocq, Samir Jegham, Yvette Muneaux
  • 6-Heteroarylpyridoindolone Derivatives, Their Preparation and Therapeutic Use Thereof
    Publication number: 20080262020
    Abstract: The disclosure relates to compounds of formula (I): wherein R1, R2, R3, R4, are R5 are as defined in the disclosure; their preparation method, compositions containing the same and therapeutic use thereof.
    Type: Application
    Filed: April 9, 2008
    Publication date: October 23, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Yvette MUNEAUX, Samir JEGHAM, Bernard BOURRIE, Pierre CASELLAS, Paola CIAPETTI, Jean-Marie DEROCQ, Camille-Georges WERMUTH
  • Pyridoindolone Derivatives Substituted in the 3-Position by a Phenyl, Their Preparation and Their Application in Therapeutics
    Publication number: 20080214538
    Abstract: The present disclosure relates to pyridoindolone derivatives of general formula (I): to processes for preparing the same and to their use in therapeutics.
    Type: Application
    Filed: May 12, 2008
    Publication date: September 4, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Bernard Bourrie, Pierre Casellas, Paola Ciapetti, Jean-Marie Derocq, Samir Jegham, Yvette Muneaux, Camille-Georges Wermuth
  • Pyridoindolone derivatives substituted in the 3-position by a phenyl, their preparation and their application in therapeutics
    Patent number: 7390818
    Abstract: The present invention relates to pyridoindolone derivatives substituted in the 3-position by a phenyl of general formula (I): to processes for preparing the same and to their use in therapeutics.
    Type: Grant
    Filed: April 19, 2005
    Date of Patent: June 24, 2008
    Assignee: Sanofi-Aventis
    Inventors: Bernard Bourrie, Pierre Casellas, Paola Ciapetti, Jean-Marie Derocq, Samir Jegham, Yvette Muneaux, Camille-Georges Wermuth
  • Use of pyridoindolone derivatives for the preparation of medicinal products
    Patent number: 7160895
    Abstract: The invention relates to a novel use of compounds of formula: for the preparation of medicinal products that are useful as anticancer agents.
    Type: Grant
    Filed: August 15, 2005
    Date of Patent: January 9, 2007
    Assignee: Sanofi-Aventis
    Inventors: Bernard Bourrie, Pierre Casellas, Jean-Marie Derocq
  • Pyridoindolone derivatives substituted in the 3-position by a phenyl, their preparation and their application in therapeutics
    Publication number: 20050288318
    Abstract: The present invention relates to pyridoindolone derivatives substituted in the 3-position by a phenyl of general formula (I): to processes for preparing the same and to their use in therapeutics.
    Type: Application
    Filed: April 19, 2005
    Publication date: December 29, 2005
    Applicant: sanofi-aventis
    Inventors: Bernard Bourrie, Pierre Casellas, Paola Ciapetti, Jean-Marie Derocq, Samir Jegham, Yvette Muneaux, Camille-Georges Wermuth
  • Slimming cosmetic composition containing a substance inducing the production of IL-6
    Publication number: 20050281895
    Abstract: This invention relates to a slimming cosmetic composition containing at least one compound inducing the production of IL-6 by the adipocytes in the form of a mixture with an NPY antagonist and/or an ?2 antagonist and with an excipient for a cosmetic preparation.
    Type: Application
    Filed: July 28, 2005
    Publication date: December 22, 2005
    Applicant: Sanfoi-Synthelabo
    Inventors: Pierre Casellas, Jean-Marie Derocq, Joelle Guesnet
  • Use of pyridoindolone derivatives for the preparation of medicinal products
    Publication number: 20050272760
    Abstract: The invention relates to a novel use of compounds of formula: for the preparation of medicinal products that are useful as anticancer agents.
    Type: Application
    Filed: August 15, 2005
    Publication date: December 8, 2005
    Applicant: Sanofi-Aventis
    Inventors: Bernard Bourrie, Pierre Casellas, Jean-Marie Derocq
  • Use of pyridoindolone derivatives for preparing anticancer medicines
    Patent number: 6967203
    Abstract: The invention relates to a novel use of compounds of formula: for the preparation of medicinal products that are useful as anticancer agents.
    Type: Grant
    Filed: April 26, 2002
    Date of Patent: November 22, 2005
    Assignee: Sanofi-Aventis
    Inventors: Bernard Bourrie, Pierre Casellas, Jean-Marie Derocq
  • Pyridoindolone derivatives substituted in the 3-position by a heterocyclic group, their preparation and their application in therapeutics
    Publication number: 20050222192
    Abstract: The present invention relates to pyridoindolone derivatives substituted in the 3-position by a heterocyclic group of general formula (I): in which: R1 represents a hydrogen atom or a (C1-C4)alkyl group; R2 represents a hydrogen atom or a (C1-C4)alkyl group; R3 represents a thienyl mono- or polysubstituted by a methyl group; or a monocyclic or bicyclic heterocyclic radical chosen from: a pyridyl, an N-oxidopyridinio, a pyrazolyl, an (N-phenyl)pyrazolyl, an (N-halophenyl)pyrazolyl, a furyl, an indolyl, an (N-benzyl)indolyl, an (N-halobenzyl)indolyl, a benzothienyl or a benzofuryl, the said radicals being unsubstituted or substituted one or more times by a halogen atom or a methyl or methoxy group; R4 and R5 are identical or different and each independently represent a hydrogen or halogen atom or a hydroxyl, hydroxymethyl, (C1-C4)alkyl, trifluoromethyl, C1-C4)alkoxy, (C1-C4)alkoxycarbonyl or cyano group. Preparation process and application in therapeutics.
    Type: Application
    Filed: April 19, 2005
    Publication date: October 6, 2005
    Applicant: sanofi-aventis
    Inventors: Bernard Bourrie, Pierre Casellas, Jean-Marie Derocq, Samir Jegham, Yvette Muneaux
  • Use of a substance binding with the peripheral benzodiazepin receptor for treating skin stress
    Patent number: 6767533
    Abstract: A composition containing a peripheral benzodiazepine receptor ligand for topical use in the treatment of cutaneous stress.
    Type: Grant
    Filed: May 14, 2001
    Date of Patent: July 27, 2004
    Assignee: Sanofi-Synthelabo
    Inventors: Pierre Casellas, Jean-Marie Derocq