Patents by Inventor Jean-Yves Trosset

Jean-Yves Trosset has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Pyridopyrimidinones derivatives as telomerase inhibitors
    Patent number: 7019002
    Abstract: The invention provides pyrido[2,3-d]pyrimidin-7(8H)-one telomerase inhibitors of the formula where R1, R2 are as defined herein. The invention also provides methods for preparing the compounds of formula I, methods of using the compounds to treat diseases such as cancer, and pharmaceutical compositions comprising the compounds.
    Type: Grant
    Filed: December 4, 2002
    Date of Patent: March 28, 2006
    Assignee: Pharmacia & Upjohn, S.p.A.
    Inventors: Mauro Angiolini, Dario Ballinari, Domenico Fusar Bassini, Luisella Bonomini, Markus Gude, Maria Menichincheri, Jurgen Moll, Jean-Yves Trosset
  • Interaction inhibitors of tcf-4 with beta-catenin
    Publication number: 20040204477
    Abstract: A compound of formula (I) is provided which is able to interact with &bgr;-catenin/TCF-4 binding site, having a structure essentially equivalent to a pharmacophore (IA), as herein described.
    Type: Application
    Filed: May 24, 2004
    Publication date: October 14, 2004
    Inventors: Juergen Moll, Stefan Knapp, Claudio Dalvit, Jean-Yves Trosset, Michael Sundstrom, Sergio Mantegani
  • Pyridopyrimidinones derivatives as telomerase inhibitors
    Publication number: 20040009993
    Abstract: The invention provides novel pyrido[2,3-d]pyrimidin-7(8H)-ones derivatives active as telomerase inhibitors, the use of the derivatives as therapeutic agents, such as antitumoral agents, processes for preparation of the derivatives, and to pharmaceutical compositions comprising the derivatives.
    Type: Application
    Filed: December 4, 2002
    Publication date: January 15, 2004
    Applicant: Pharmacia Italia S.p.A.
    Inventors: Mauro Angiolini, Dario Ballinari, Domenico Fusar Bassini, Luisella Bonomini, Markus Gude, Maria Menichincheri, Jurgen Moll, Jean-Yves Trosset