Abstract: The invention provides novel heterocyclic compounds having the general formula (I), and pharmaceutically acceptable salts thereof, wherein R1 to R9 and p are as described herein: Further provided are pharmaceutical compositions including the compounds, processes of manufacturing the compounds and methods of using the compounds as medicaments, in particular methods of using the compounds as antibiotics for the treatment or prevention of bacterial infections and resulting diseases.

Abstract: The invention provides novel imidazole pyrazole derivatives having the general formula (I), and pharmaceutically acceptable salts thereof, wherein A and R1-R7 are as described herein: Further provided are pharmaceutical compositions including the compounds, processes of manufacturing the compounds and methods of using the compounds as medicaments, in particular methods of using the compounds as antibiotics for the treatment or prevention of bacterial infections and resulting diseases.

Abstract: A fault arc signal detection method using a convolutional neural network, comprising: enabling a sampling signal subjected to analog-digital conversion to respectively pass through three different band-pass filters; respectively extracting a time-domain feature and a frequency-domain feature from a half wave output of each filter; constructing a two-dimensional feature matrix by means of extracted time-frequency feature vectors from the output of each filter, and stacking the feature matrices corresponding the outputs of the three filters to construct a three-dimensional matrix for each half wave; and processing a multi-channel feature matrix by using a multi-channel two-dimensional convolutional neural network, and determining, according to the output result of the neural network, whether the half wave is an arc.

Abstract: The invention provides novel imidazopyrazine derivatives having the general formula (I), wherein Rx and R3 to R5 are as described herein: or pharmaceutically acceptable salts thereof. Further provided are pharmaceutical compositions including the compounds, processes of manufacturing the compounds and methods of using the compounds as medicaments, in particular methods of using the compounds as antibiotics for the treatment or prevention of bacterial infections and resulting diseases.

Abstract: The invention provides novel heterocyclic compounds having the general formula (I), and pharmaceutically acceptable salts thereof, wherein X, D, R1 to R4, and R6 to R10 are as described herein. Further provided are pharmaceutical compositions including the compounds, processes of manufacturing the compounds and methods of using the compounds as medicaments, in particular methods of using the compounds as antibiotics for the treatment or prevention of bacterial infections and resulting diseases.

Abstract: A water supply simulation method for interlaced system of river and canal system based on groundwater model, includes: S1. constructing simulated water conveyance channel based on first data, and performing attribute definition on water conveyance channels; S2. acquiring initial seepage, evaporation and discharge; S3. performing reverse water demand calculation; S4. performing sequential water supply simulation; S5. acquiring corresponding water head, obtaining current seepage, evaporation, discharge, head-end water demand and water consumption demand of each water conveyance channel based on water head; S6. judging whether current iteration is converged according to water head, if yes, proceeding to S7, otherwise returning to S3 after update; S7. judging whether there is next time period, if yes, returning to S3 after update, otherwise proceeding to S8; and S8. judging whether there is a next stress period, if yes, returning to S3 after update, otherwise outputting the result obtained in S5, and ending.

Abstract: Disclosed is an automobile tire burst simulation experiment device, which is fixed on a rim installed with an automobile tire. The automobile tire burst simulation experiment device comprises a pre-tightening triggering device, a retracting device, a storage battery and a controller, the tire burst simulation experiment device according to the present invention uses two drive motors to drive two sets of roller screw slide rails, so as to drive the breakdown device away from and close to the tire to achieve a simulated tire burst and rapid deflation. The experiment device has the characteristics of quick installation, low cost, strong versatility, and adjustable speed; the device can be applied to the tire burst experiment under different vehicle speeds and road conditions of various automobile models. The structure is simple and the simulation control accuracy is high. After the tire burst, the subsequent experiments of the vehicle are not affected.

Abstract: A sun visor assembly for a vehicle according to an exemplary aspect of the present disclosure includes, among other things, a visor having a transparent portion and a circuit configured to control at least one function of the visor. The visor is pivotable between a first position and a second position.

Abstract: This disclosure generally relates to a headrest assembly, seat, and a method of use. In the disclosure, a head restraint is moveable from an upright position to a folded position by movement of either the push-button or a lever. The disclosed arrangement provides two ways to fold a head restraint, and can further be integrated with another assembly, such as a seat back folding assembly. The disclosed arrangement is further configured to resist vibration, leading to a tighter, more stable design, which provides increased customer satisfaction.

Abstract: A method and an apparatus for retrieving teleplay content is disclosed. The method includes: generating basic summary information corresponding to each teleplay based on basic information of entities of each teleplay; generating episode summary information corresponding to each episode of each teleplay based on episode data of each episode of each teleplay; establishing a teleplay graph database based on the basic summary information corresponding to each teleplay and the episode summary information corresponding to each episode; and feeding a playing portal for a target episode of a target teleplay corresponding to teleplay search information back to a user based on the teleplay graph database.

Abstract: Provided are novel imidazopyrazine derivatives having the general formula (I), wherein A and R1 to R11 are as described herein and pharmaceutically acceptable salts thereof. Further provided are pharmaceutical compositions including the compounds, processes of manufacturing the compounds and methods of using the compounds as medicaments, in particular methods of using the compounds as antibiotics for the treatment or prevention of bacterial infections and resulting diseases.

Abstract: A vector analysis calculation-based arc crosstalk signal identification method. A new sampling circuit manner is proposed in the method, wherein a current signal is sampled on zero and live lines, and the signal is converted into two digital signals with a sampling rate of 200 MHz by means of a dual-channel ADC, and the digital signals are sent to a hardware digital signal processing unit. Five pass bands are selected to perform band-pass filtering on the two signals separately. Time-sharing processing and vector analysis are performed on the filtered signals, and the amplitude ratio and fluctuation characteristics of two resistor terminal voltages, as well as the phase difference between shunt resistor and inductor terminal voltage signals are extracted as crosstalk feature quantities. According to a zero-crossing signal, a system segments the feature quantities extracted by a hardware processing module and sends same to a neural network for classification and determination.

Abstract: Provided are novel imidazopyrazine derivatives having the general formula (I), wherein A and R1 to R11 are as described herein and pharmaceutically acceptable salts thereof. Further provided are pharmaceutical compositions including the compounds, processes of manufacturing the compounds and methods of using the compounds as medicaments, in particular methods of using the compounds as antibiotics for the treatment or prevention of bacterial infections and related diseases.

Abstract: Provided are novel imidazopyrazine derivatives having the general formula (I), wherein A and R1 to R11 are as described herein and pharmaceutically acceptable salts thereof. Further provided are pharmaceutical compositions including the compounds, processes of manufacturing the compounds and methods of using the compounds as medicaments, in particular methods of using the compounds as antibiotics for the treatment or prevention of bacterial infections and resulting diseases.

Abstract: Provided are novel imidazopyrazine derivatives having the general formula (I), wherein R1 to R11 are as described herein and pharmaceutically acceptable salts thereof. Further provided are pharmaceutical compositions including the compounds, processes of manufacturing the compounds and methods of using the compounds as medicaments, in particular methods of using the compounds as antibiotics for the treatment or prevention of bacterial infections and related diseases.

Abstract: An AC/DC leakage detection method, which supports the detection of DC leakage and AC leakage. A DC leakage current and a low-frequency leakage current are measured by means of magnetic modulation technology, an AC signal is measured in the form of pure induction, and two detection modes are performed in a time-sharing manner. A collected leakage signal is converted into a digital signal through an AD converter. By means of the method of the present invention, the processing of a leakage signal is divided into three channels for respectively processing DC leakage, low-frequency AC leakage, and high-frequency AC leakage. The overall effective value of residual current is calculated by integrating results of DC detection and AC detection. The method of the present invention supports the detection of a suddenly increased current; and when there is a suddenly increased current, detection mode switching is performed by detecting the current sudden change of the current.

Abstract: A vacuum degree detection device with buried electrodes in a vacuum interrupter and a method thereof are provided. The vacuum degree wireless detection device includes two parts, wherein a first part is provided inside the vacuum interrupter, including buried electrodes, etc., wherein the buried electrodes are welded on an end cover of the vacuum interrupter; a second part is the external detection device after the arc interrupter is processed, including: detection and calculation components, wireless transmitters, rechargeable energy storage batteries, wireless charging coils, etc. The external detection device and the buried electrode structure is designed separately, and the buried structure such as the buried electrodes can be processed as a whole with the vacuum interrupter. During the detection, the external detection device is installed above the buried electrode structure.

Abstract: Provided are novel heterocyclic compounds having the general formula (I), and pharmaceutically acceptable salts thereof, wherein R1 to R4, m, n, and p are as described herein. Further provided are pharmaceutical compositions including the compounds, processes of manufacturing the compounds and methods of using the compounds as medicaments, in particular methods of using the compounds as antibiotics for the treatment or prevention of bacterial infections and resulting diseases.

Abstract: A fault-arc identification method, device and apparatus, and a storage medium. The method comprises: performing sampling on a target arc at a high frequency, and obtaining a high-frequency sampling signal (S11); preprocessing the high-frequency sampling signal, and obtaining a processed sampling signal (S12); performing feature extraction on the processed sampling signal, and obtaining a target arc feature (S13); and inputting the target arc feature to a neural network model, obtaining a target output result, and determining, according to the target output result, whether the target arc is a fault-arc (S14). Performing sampling on a target arc at a high frequency can obtain more arc features from the target arc. Moreover, since a neural network model has favorable data classification capability, using a neural network model to perform determination with respect to the target arc can improve the accuracy and reliability of a fault-arc detection result.