Publication number: 20100022769
Abstract: The present invention describes the synthesis of the compounds of formulae (1), (2) and (3) in which m and n, which may be identical or different, may have the values 0, 2, 3, 4, 5 and 6; Z and Y, which may be identical or different, represent a nitrogenated cyclic system bonded by nitrogen or by one of the ring carbons or an NR1R2 system; and X is selected from the group consisting of hydrogen, C1-C12 alkyl, substituted alkyl, C3-C12 aryl, amino, alkylamino, nitro, hydroxy, alkoxy, halogen, carboxy or carboxamido. The use of the compounds of formulae (1), (2) and (3) as anti-HIV agents in the treatment of Acquired Immune Deficiency Syndrome (AIDS) is described.
Type:
Application
Filed:
October 26, 2007
Publication date:
January 28, 2010
Inventors:
Jordi Teixidó Closa, José Ignacio Borrell Bilbao, Santiago Nonell Marrugat, Xavier Batllori Aguilá, Sofia Pettersson Salom, Laia Ros Blancó, Maria Obdulia Rabal Gracia, Violata Pérez Nueno, José Esté Araque, Imma Clotet Codina, Mercedes Armand Ugón, Ralmon Puig De La Bellacasa