Patents by Inventor Josef D. Riggenberg

Josef D. Riggenberg has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Process for the preparation of 1,2-dihydroquinolines
    Patent number: 6180794
    Abstract: A method for preparing 1,2-dihydroquinolines that is more flexible than the Skraup reaction is provided. The method comprises treating an ortho-alkenyl aniline with a ketone in the presence of a Lewis acid. Novel intermediates and products of this method useful as steroid receptor modulators, as well as pharmaceutical compositions and methods of use thereof are also claimed.
    Type: Grant
    Filed: October 15, 1999
    Date of Patent: January 30, 2001
    Assignee: Ligand Pharmacueticals Incorparated
    Inventors: James P. Edwards, Todd K. Jones, Josef D. Riggenberg, Erick M. Carreira
  • Process for the preparation of 1,2-dihydroquinolines
    Patent number: 6172241
    Abstract: A method for preparing 1,2-dihydroquinolines that is more flexible than the Skraup reaction is provided. The method comprises treating an ortho-alkenyl aniline with a ketone in the presence of a Lewis acid. Novel intermediates and products of this method useful as steroid receptor modulators, as well as pharmaceutical compositions and methods of use thereof are also claimed.
    Type: Grant
    Filed: October 15, 1999
    Date of Patent: January 9, 2001
    Assignee: Ligand Pharmaceuticals Incorporated
    Inventors: James P. Edwards, Todd K. Jones, Josef D. Riggenberg, Erick M. Carreira
  • Process for the preparation of 1,2-dihydroquinolines
    Patent number: 6001846
    Abstract: A method for preparing 1,2-dihydroquinolines that is more flexible than the Skraup reaction is provided. The method comprises treating an ortho-alkenyl aniline with a ketone in the presence of a Lewis acid. Novel intermediates and products of this method useful as steroid receptor modulators, as well as pharmaceutical compositions and methods of use thereof are also claimed.
    Type: Grant
    Filed: February 17, 1998
    Date of Patent: December 14, 1999
    Assignee: Ligand Pharmaceuticals Incorporated
    Inventors: James P. Edwards, Todd K. Jones, Josef D. Riggenberg, Erick M. Carreira