Patents by Inventor Pierre Girault

Pierre Girault has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4808210
    Abstract: A 5-pyrazolone of the formula ##STR1## wherein R is selected from the group consisting of mono- and polycyclic aromatic of 6 to 14 carbon atoms, heterocyclic optionally substituted with phenyl, ##STR2## and benzyl, all optionally substituted with at least one member of the group consisting of fluorine, chlorine, bromine, --CF.sub.3, optionally unsaturated alkyl of 1 to 8 carbon atoms and the radical OZ in which Z is an optionally unsaturated alkyl of 1 to 8 carbon atoms or an acyl of a carboxylic acid of 1 to 6 carbon atoms, A is selected from the group consisting of halogen, --CF.sub.3 and --CN, B and C are individually selected from the group consisting of hydrogen, halogen, --OH, --OR' and R' is optionally unsaturated alkyl of 1 to 8 carbon atoms, acyl of 1 to 6 carbon atoms, alkyl sulfonyl of 1 to 8 carbon atoms, aryl sulfonyl of 6 to 18 carbon atoms and benzyl optionally substituted with a member of the group consisting of fluorine, chlorine, bromine, --CF.sub.
    Type: Grant
    Filed: September 11, 1987
    Date of Patent: February 28, 1989
    Assignee: Roussel Uclaf
    Inventors: Jean Tessier, Pierre Girault
  • Patent number: 4801717
    Abstract: Novel hydroxylamino derivatives of the formulaAr--ONH.sub.2 Iwherein Ar is selected from the group consisting of mono- and polycyclic aromatics and hetero-aromatics, both optionally substituted with at least one member of the group consisting of --OH, halogen, --NO.sub.2, --CN, ##STR1## --R.sub.7, --OR.sub.8, ##STR2## --SO.sub.2 R.sub.12, --SO.sub.3 R.sub.13, --COOR.sub.14, aryl of 6 to 14 carbon atoms, --OR.sub.16, --CH.sub.2 --CN and --CH.sub.2 SO.sub.2 --R.sub.15, R.sub.1, R.sub.2, R.sub.3, R.sub.4, R.sub.5 and R.sub.6 are individually selected from the group consisting of hydrogen and alkyl of 1 to 8 carbon atoms, R.sub.7 and R.sub.8 are optionally unsaturated alkyl of 1 to 8 carbon atoms optionally substituted with at least one member of the group consisting of halogen and cyano, R.sub.9, R.sub.10, R.sub.11, R.sub.12 and R.sub.
    Type: Grant
    Filed: June 24, 1986
    Date of Patent: January 31, 1989
    Assignee: Roussel Uclaf
    Inventors: Jean Tessier, Pierre Girault, Jean-Jacques Herve, Charles-Jacques Van Assche
  • Patent number: 4777180
    Abstract: Novel esters in all stereoisomeric forms and mixtures of said isomers of the formula ##STR1## wherein one of X and Y is ##STR2## and the other is selected from the group consisting of --CH.sub.2 --, --CH.sub.2 --CH.sub.2 -- and --CH.sub.2 --CH.sub.2 --CH.sub.2 --, n is an integer from 2 to 3 and R.sub.1 is selected from the group consisting of alkyl of 1 to 3 carbon atoms and alkenyl and alkynyl of 2 to 3 carbon atoms having pesticidal activity.
    Type: Grant
    Filed: October 7, 1987
    Date of Patent: October 11, 1988
    Assignee: Roussel Uclaf
    Inventors: Jean Tessier, Pierre Girault
  • Patent number: 4618364
    Abstract: Novel uracils of the formula ##STR1## wherein R.sub.1 is selected from the group consisting of alkyl of 1 to 8 carbon atoms, alkoxy of 1 to 8 carbon atoms, halogen and --C(Hal).sub.3, Hal is halogen and R.sub.2 is hydrogen or R.sub.1 and R.sub.2 taken together with the benzene ring to which they are attached form a system of two coupled rings optionally containing at least one heteroatom having selective herbicidal activity.
    Type: Grant
    Filed: July 6, 1984
    Date of Patent: October 21, 1986
    Assignee: Roussel Uclaf
    Inventors: Jean Tessier, Pierre Girault
  • Patent number: 4565822
    Abstract: Novel cyclopropanecarboxylates in all possible isomeric forms or mixtures thereof of the formula ##STR1## with a 1R,cis or 1R,trans structure and wherein X is a halogen, R is selected from the group consisting of (A) optionally unsaturated alkyl of 2 to 12 carbon atoms, (B) optionally unsaturated cycloalkyl of 3 to 12 carbon atoms, (c) ##STR2## Z is selected from the group consisting of --C.tbd.CH, --CH.sub.3 and --CN and Ar is selected from the group consisting of --C.sub.6 H.sub.5, --C.sub.6 F.sub.5, ##STR3## B is hydrogen or fluorine and X is fluorine, chlorine or bromine ##STR4## Y.sub.2 is selected from the group consisting of hydrogen, fluorine, chlorine bromine, --C.tbd.N and --C.tbd.CH, Y.sub.3, Y.sub.4, and Y.sub.
    Type: Grant
    Filed: August 2, 1984
    Date of Patent: January 21, 1986
    Assignee: Roussel Uclaf
    Inventors: Jean Tessier, Andre Teche, Pierre Girault
  • Patent number: 4501894
    Abstract: Novel heterocyclic compounds of the formula ##STR1## wherein X is selected from the group consisting of chlorine, bromine, iodine and --OH, W is selected from the group consisting of hydrogen and --CN, Z is selected from the group consisting of --CH.sub.2 -- and --O-- attached to the carbon atom included between a nitrogen and the sulfur atom of Y and Y is selected from the group consisting of thiazolyl or thiadiazolyl connected to ##STR2## at one of its available positions except for (2-benzyl-4 and 5-thiazolyl) methanol and .alpha.-cyano-(2-benzyl-5-thiazolyl)-methanol and the compounds wherein X is halogen when W is --CN whose esters have insecticidal activity.
    Type: Grant
    Filed: February 25, 1982
    Date of Patent: February 26, 1985
    Assignee: Roussel Uclaf
    Inventors: Francois Nezot, Pierre Girault, Jean Tessier, Jacques Martel
  • Patent number: 4450169
    Abstract: Novel esters of the formula ##STR1## wherein R is selected from the group consisting of ##STR2## W is selected from the group consisting of hydrogen and --CN, Z is selected from the group consisting of --CH.sub.2 -- and --O--, and is attached to a carbon atom included between a nitrogen and the sulfur atom of Y and Y is selected from the group consisting of thiazolyl or thiadiazolyl connected to ##STR3## at one of its available positions.
    Type: Grant
    Filed: February 25, 1982
    Date of Patent: May 22, 1984
    Assignee: Roussel Uclaf
    Inventors: Francois Nezot, Pierre Girault, Jean Tessier, Jacques Martel
  • Patent number: 4401673
    Abstract: Novel 3-(buta-1',3'-dienyl)-cyclopropane-1-carboxylic acid compounds of the formula ##STR1## wherein X.sub.1 and X.sub.2 are individually a halogen and A is selected from the group consisting of (A) benzyl optionally substituted (B) ##STR2## wherein R.sub.1 is selected from the group consisting of hydrogen and --CH.sub.3 and R.sub.2 is selected from the group consisting of aryl and --CH.sub.2 --C.tbd.CH, (C) ##STR3## wherein R.sub.3 is an aliphatic of 2 to 6 carbon atoms containing at least one carbon-carbon unsaturation, (D) ##STR4## wherein R'.sub.1 and R'.sub.2 are individually selected from the group consisting of hydrogen, halogen, alkyl of 1 to 6 carbon atoms, aryl of 6 to 10 carbon atoms, alkoxycarbonyl of 2 to 5 carbon atoms and cyano and R.sub.3 has the above definition, (E) ##STR5## wherein R.sub.4 is selected from the group consisting of hydrogen, --CN, --CH.sub.3, --CONH.sub.2, --CSNH.sub.2 and --C.tbd.CH, R.sub.5 is selected from the group consisting of chlorine and --CH.sub.
    Type: Grant
    Filed: January 26, 1981
    Date of Patent: August 30, 1983
    Assignee: Roussel Uclaf
    Inventors: Jacques Martel, Jean Tessier, Pierre Girault
  • Patent number: 4364928
    Abstract: Ion exchange resins of the acid type at least partially salified with 7-bromo-6-chloro-febrifugin having very good coccidiostatic activity, a very good anti-leucocytozoonosis activity and a low toxicity and their preparation.
    Type: Grant
    Filed: October 7, 1980
    Date of Patent: December 21, 1982
    Assignee: Roussel-Uclaf
    Inventors: Jacques Martel, Jean Tessier, Pierre Girault, Jean A. Grandadam
  • Patent number: 4170465
    Abstract: Novel crotonamides of the formula ##STR1## wherein R is selected from the group consisting of adamantyl, bornyl, 5',6'-dihydroendo-5'-dicyclopentadienyl and saturated and unsaturated cycloalkyl of 3 to 8 carbon atoms optionally substituted with a member of the group consisting of alkyl of 1 to 6 carbon atoms, hydroxy, chlorine and alkoxycarbonyl of 1 to 6 alkyl carbon atoms and R.sub.1 is alkyl of 1 to 3 carbon atoms having pre- and post-emergence herbicidal properties.
    Type: Grant
    Filed: April 16, 1975
    Date of Patent: October 9, 1979
    Assignee: Roussel UCLAF
    Inventors: Jacques Perronnet, Pierre Girault
  • Patent number: 4137068
    Abstract: Novel ureas of the formula ##STR1## wherein A and B are chlorine or A is chlorine or hydrogen and B is --CF.sub.3, R and R.sub.1 are individually alkyl of 1 to 3 carbon atoms and R.sub.2 is alkyl of 1 to 6 carbon atoms optionally substituted with a halogen having herbicidal properties, particularly useful in cultivated grass crops and their preparation and use.
    Type: Grant
    Filed: March 18, 1976
    Date of Patent: January 30, 1979
    Assignee: Roussel Uclaf
    Inventors: Jacques Perronnet, Jean-Pierre Demoute, Pierre Girault, Andre Teche
  • Patent number: 4097578
    Abstract: Imidazolidines of the formula ##STR1## wherein X is selected from the group consisting of oxygen and amine which inhibit the effects of androgens on peripheric receptors without interfering with normal hypophysial functions.
    Type: Grant
    Filed: October 21, 1976
    Date of Patent: June 27, 1978
    Assignee: Roussel Uclaf
    Inventors: Jacques Perronnet, Pierre Girault, Claude Bonne
  • Patent number: 4039316
    Abstract: Novel crotonanilides of the formula ##STR1## wherein R' is selected from the group consisting of ##STR2## R and R.sub.1 are alkyl of 1 to 6 carbon atoms and R.sub.2 is selected from the group consisting of hydrogen, methyl and methoxy having pre- and post-emergence herbicidal activity.
    Type: Grant
    Filed: September 24, 1975
    Date of Patent: August 2, 1977
    Assignee: Roussel Uclaf
    Inventors: Jacques Perronnet, Pierre Girault
  • Patent number: 4036633
    Abstract: Novel crotonanilides of the formula ##STR1## wherein R is selected from the group consisting of ##STR2## X is selected from the group consisting of alkyl of 1 to 8 carbon atoms and cycloalkyl of 3 to 7 carbon atoms, Z is alkyl of 1 to 6 carbon atoms, X.sub.1 is alkoxyalkyl of 2 to 12 carbon atoms, X.sub.2 is alkyl of 1 to 3 carbon atoms, X.sub.3 is selected from the group consisting of alkyl or alkoxy of 1 to 3 carbon atoms and R.sub.1 and R.sub.2 are individually alkyl of 1 to 3 carbon atoms having pre- and post-emergence herbicidal activity.
    Type: Grant
    Filed: September 16, 1975
    Date of Patent: July 19, 1977
    Assignee: Roussel-UCLAF
    Inventors: Jacques Perronnet, Pierre Girault
  • Patent number: 4014679
    Abstract: Novel crotonanilides of the formula ##STR1## wherein Z is selected from the group consisting of --O-- and --S--, R is selected from the group consisting of alkyl of 1 to 6 carbon atoms and optionally substituted phenyl, X and Y are individually selected from the group consisting of hydrogen, halogen, lower alkyl of 1 to 6 carbon atoms optionally substituted with at least one halogen, alkoxy of 1 to 3 carbon atoms, alkylthio and alkylsulfinyl of 1 to 6 carbon atoms, acyl of an organic carboxylic acid of 1 to 6 carbon atoms, --NO.sub.2 and --CF.sub.3, R.sub.1 is selected from the group consisting of hydrogen, chlorine, bromine, alkoxycarbonyl with 1 to 6 alkyl carbon atoms, nitro and alkylthio, alkylsulfinyl and alkylsulfonyl of 1 to 3 alkyl carbon atoms and R.sub.2 is alkyl of 1 to 6 carbon atoms, said compounds existing in the form of their E or Z isomers or mixtures thereof and having herbicidal properties.
    Type: Grant
    Filed: May 30, 1975
    Date of Patent: March 29, 1977
    Assignee: Roussel-UCLAF
    Inventors: Jacques Perronnet, Pierre Girault
  • Patent number: 4000298
    Abstract: Novel benzimidazole derivatives of the formula ##STR1## wherein R is alkyl of 1 to 2 carbon atoms and R.sub.1 is selected from the group consisting of tetrahydrofurfuryl, a saturated or unsaturated oxygen heterocycle of 4 to 5 carbon atoms and ##STR2## wherein Z is unsaturated hydrocarbon radical of 2 to 4 carbon atoms having at least 2 halogen atoms which possess fungicidal activity.
    Type: Grant
    Filed: October 30, 1975
    Date of Patent: December 28, 1976
    Assignee: Roussel-UCLAF
    Inventors: Jacques Perronnet, Pierre Girault
  • Patent number: 3983129
    Abstract: Novel 3-phosphoryloxy-isothiazoles of the formula ##SPC1##Wherein R is selected from the group consisting of alkyl of 1 to 3 carbon atoms, alkoxy of 1 to 3 carbon atoms and ##EQU1## R' and R" being individually SELECTED FROM THE GROUP CONSISTING OF HYDROGEN AND ALKYL OF 1 TO 3 CARBON ATOMS, R.sub.1 is alkyl of 1 to 3 carbon atoms, R.sub.2 is selected from the group consisting of hydrogen, alkyl of 1 to 5 carbon atoms, aryl of 6 to 10 carbon atoms, aralkyl of 7 to 12 carbon atoms, cyano, carbalkoxy of 2 to 4 carbon atoms and NHR'", and R'" is selected from the group consisting of hydrogen and aryl of 6 to 10 carbon atoms, R.sub.
    Type: Grant
    Filed: January 13, 1975
    Date of Patent: September 28, 1976
    Assignee: Roussel-UCLAF
    Inventors: Jacques Perronnet, Laurent Taliani, Pierre Girault, Andre Poittevin
  • Patent number: 3958005
    Abstract: Novel tetrahydrofuran derivatives of the formula ##EQU1## wherein R is a branched or linear alkyl of 1 to 10 carbon atoms and R.sub.1 is alkyl of 1 to 5 carbon atoms and X is selected from the group consisting of chlorine, bromine, --OH and alkylcarbonyloxy of 2 to 5 carbon atoms useful as insecticides and their preparation.
    Type: Grant
    Filed: February 3, 1975
    Date of Patent: May 18, 1976
    Assignee: Roussel Uclaf
    Inventors: Daniel Hainaut, Jean-Pierre Demoute, Pierre Girault
  • Patent number: 3932447
    Abstract: Novel benzimidazole derivatives of the formula ##SPC1##Wherein R is alkyl of 1 to 2 carbon atoms and R.sub.1 is selected from the group consisting of tetrahydrofurfuryl, a saturated or unsaturated oxygen heterocycle of 4 to 5 carbon atoms and ##EQU1## wherein Z is unsaturated hydrocarbon radical of 2 to 4 carbon atoms having at least 2 halogen atoms which possess fungicidal activity.
    Type: Grant
    Filed: September 18, 1973
    Date of Patent: January 13, 1976
    Assignee: Roussel-UCLAF
    Inventors: Jacques Perronnet, Pierre Girault