Patents by Inventor Stéphane Cuisiat

Stéphane Cuisiat has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 8455550
    Abstract: The present invention concerns compounds of general formula (1), where in:—-a- is a single or double bond, Ar is an aromatic group, substituted or unsubstituted, R1 and R2 each independently or together are: a hydrogen atom or C1-C6 alkyl group, branched or unbranched, saturated or unsaturated, substituted or unsubstituted; the groups R1 and R2 may also form a heterocycle, R3 and R3? each independently or together are a hydrogen atom or C1-C6 alkyl group, X is an oxygen atom or a sulphur atom, and the addition salts of the compounds of general formula (1) with pharmaceutically acceptable mineral acids or organic acids.
    Type: Grant
    Filed: April 2, 2010
    Date of Patent: June 4, 2013
    Assignee: Pierre Fabre Medicament
    Inventors: Stéphane Cuisiat, Adrian Newman-Tancredi, Olivier Vitton, Bernard Vacher
  • Publication number: 20120029013
    Abstract: The present invention concerns compounds of general formula (1), where in:—-a- is a single or double bond, Ar is an aromatic group, substituted or unsubstituted, R1 and R2 each independently or together are: a hydrogen atom or C1-C6 alkyl group, branched or unbranched, saturated or unsaturated, substituted or unsubstituted; the groups R1 and R2 may also form a heterocycle, R3 and R3? each independently or together are a hydrogen atom or C1-C6 alkyl group, X is an oxygen atom or a sulphur atom, and the addition salts of the compounds of general formula (1) with pharmaceutically acceptable mineral acids or organic acids.
    Type: Application
    Filed: April 2, 2010
    Publication date: February 2, 2012
    Applicant: PIERRE FABRE MEDICAMENT
    Inventors: Stéphane Cuisiat, Adrian Newman-Tancredi, Olivier Vitton, Bernard Vacher
  • Publication number: 20090082582
    Abstract: The invention relates to a process for the preparation of compounds of general formula (3) wherein: (a) represents a single or double bond; W represents a group CH, CH2, CHCH3, CCH3, C(CH3)2, a group C(CH2)2 (i.e. a carbon atom carrying two methylene groups bonded to one another so as to form a spiro-cyclopropane moiety), with the proviso, however, that when (a) is a double bond then W represents exclusively a group CH or CCH3 and when (a) is a single bond then W represents exclusively a group CH2, CHCH3, C(CH3)2 or C(CH2)2.
    Type: Application
    Filed: March 8, 2007
    Publication date: March 26, 2009
    Applicant: Pierre Fabre Medicament
    Inventors: Bernard Vacher, Stephane Cuisiat, Nicolas Roques
  • Patent number: 7235568
    Abstract: The invention provides compounds of the formula: wherein (a) is a single or double bond; W is CH, CH2, CHCH3, C(CH3)2, C(CH2)2 or C(CH2)3; X is N; and Y is H or F, and salts, hydrates, tautomers, pure enantiomers, and enantiomeric mixtures; and a method of treating schizophrenia comprising administering same.
    Type: Grant
    Filed: July 28, 2006
    Date of Patent: June 26, 2007
    Assignee: Pierre Fabre Medicament
    Inventors: Bernard Vacher, Stéphane Cuisiat, Wouter Koek, Francis Colpaert
  • Patent number: 7163957
    Abstract: The invention provides compounds of the formula: wherein (a) is a single or double bond; W is CH, CH2, CHCH3, CCH3, C(CH3)2, C(CH2)2 or C(CH2)3, provided that when (a) is a double bond, then W is CH or CCH3, and when (a) is a single bond, then W is CH2, CHCH3, C(CH3)2, C(CH2)2 or C(CH2)3; X is CH or N; and Y is H or F, and salts, hydrates, tautomers, pure enantiomers, and enantiomeric mixtures; and a method of treating schizophrenia comprising administering same.
    Type: Grant
    Filed: October 16, 2003
    Date of Patent: January 16, 2007
    Assignee: Pierre Fabre Medicament
    Inventors: Bernard Vacher, Stéphane Cuisiat, Wouter Koek, Francis Colpaert
  • Publication number: 20060264471
    Abstract: The invention provides compounds of the formula wherein (a) is a single or double bond; W is CH, CH2, CHCH3, C(CH3)2, C(CH2)2 or C(CH2)3; X is N; and Y is H or F, and salts, hydrates, tautomers, pure enantiomers, and enantiomeric mixtures; and a method of treating schizophrenia comprising administering same.
    Type: Application
    Filed: July 28, 2006
    Publication date: November 23, 2006
    Applicant: PIERRE FABRE MEDICAMENT
    Inventors: Bernard Vacher, Stephane Cuisiat, Wouter Koek, Francis Colpaert
  • Publication number: 20060014827
    Abstract: The invention provides compounds of the formula: wherein (a) is a single or double bond; W is CH, CH2, CHCH3, CCH3, C(CH3)2, C(CH2)2 or C(CH2)3, provided that when (a) is a double bond, then W is CH or CCH3, and when (a) is a single bond, then W is CH2, CHCH3, C(CH3)2, C(CH2)2 or C(CH2)3; X is CH or N; and Y is H or F, and salts, hydrates, tautomers, pure enantiomers, and enantiomeric mixtures; and a method of treating schizophrenia comprising administering same.
    Type: Application
    Filed: October 16, 2003
    Publication date: January 19, 2006
    Applicant: PIERRE FABRE MEDICAMENT
    Inventors: Bernard Vacher, Stephane Cuisiat, Wouter Koek, Francis Colpaert
  • Patent number: 6417222
    Abstract: The present invention relates to novel [(2-substituted-5-[3-thienyl])-benzyl]-[2-([2-isopropoxy-5-fluoro]-phenoxy)-ethyl]-amine derivatives having formula (1) and the use thereof as medicaments, especially anti-psychotic medicaments.
    Type: Grant
    Filed: September 28, 2001
    Date of Patent: July 9, 2002
    Assignee: Pierre Fabre Medicament
    Inventors: Bernard Vacher, Stéphane Cuisiat, Wouter Koek
  • Patent number: 6350913
    Abstract: The present invention relates to novel 3-alkoxybenzylamine derivatives of general formula (1): which are useful as medicinal products and in particular as antipsychotic agents.
    Type: Grant
    Filed: May 29, 2001
    Date of Patent: February 26, 2002
    Assignee: Pierre Fabre Medicament
    Inventors: Bernard Vacher, Stéphane Cuisiat, Wouter Koek