Abstract: The present invention discloses a process for the preparation of pregnadiene derivatives having formula I, their stereoisomer and intermediate thereof.

Abstract: The present invention discloses a process for the preparation of pregnadiene derivatives having formula I, their stereoisomer and intermediate thereof.

Abstract: The present invention discloses a process for the preparation of 16, 17-acetals of pregnane derivatives having formula I wherein each substituent is independently selected from; R1 is H or CH3; R2 is C1-C6 linear or branched alkyl, alkynyl group or cycloalkyl group; aryl or heteroaryl group; or R1 and R2 combine to form saturated, unsaturated C3-C6 cyclic or heterocyclic ring; R3 and R4 are same or different and each independently represents H or halogen; R5 is —OH or —OCOR wherein R represents H or C1-C6 linear, branched or cyclic alkyl group that may be substituted.

Abstract: The present invention discloses a process for the preparation of 16, 17-acetals of pregnane derivatives having formula I wherein each substituent is independently selected from; R1 is H or CH3; R2 is C1-C6 linear or branched alkyl, alkynyl group or cycloalkyl group; aryl or heteroaryl group; or R1 and R2 combine to form saturated, unsaturated C3-C6 cyclic or heterocyclic ring; R3 and R4 are same or different and each independently represents H or halogen; R5 is —OH or —OCOR wherein R represents H or C1-C6 linear, branched or cyclic alkyl group that may be substituted.

Abstract: The present invention relates to novel triazine compounds of formula (1). The present invention also discloses compounds of formula I along with other pharmaceutical acceptable excipients and use of the compounds to modulate the PI3K/mTOR pathway.

Abstract: A process for synthesis of enatiomerically pure or enatiomerically enriched or racemic mixture of (+ and/or ?) epicatechin and its intermediates, comprising the steps of: (i) obtaining penta-protected quercetin; (ii) reducing the penta-protected quercetin obtained from step (i); (iii) optionally deprotecting the compound of step (ii); (iv) reducing the compound obtained from step (ii) or step (iii) in the presence of a chiral/achiral reducing agent to obtain a chiral intermediate; (v) deprotecting and/or hydrogenation of the chiral intermediate obtained from step (iv) to obtain (?)-epicatechin; (vi) optionally simultaneously deprotecting and by drogenation of the compound obtained from step (ii) to obtain racemic epicatechin.

Abstract: A process for synthesis of enatiomerically pure or enatiomerically enriched or racemic mixture of (+and/or?) epicatechin echm and its intermediates, comprising the steps of: (i) obtaining penta-protected quercetin; (ii) reducing the penta-protected quercetin obtained from step (i); (iii) optionally deprotecting the compound of step (ii); (iv) reducing the compound obtained from step (ii) or step (iii) in the presence of a chiral/achiral reducing agent to obtain a chiral intermediate; (v) deprotecting and/or hydrogenation of the chiral intermediate obtained from step (iv) to obtain (?)-epicatechin; (vi) optionally simultaneously deprotecting and by drogenation of the compound obtained from step (ii) to obtain racemic epicatechin.

Abstract: The present invention relates to novel triazine compounds of formula (1). The present invention also discloses compounds of formula I along with other pharmaceutical acceptable excipients and use of the compounds to modulate the PI3K/mTOR pathway.

Abstract: In order to establish routing to/from a base station within a hybrid-cellular network, each network element is assigned a “class” based on a received signal strength of the base station. Each network element is allowed to choose a network element of lower class for relaying information to the base station.

Abstract: The invention provides an adaptive turbo decision feedback equalizer for executing an adaptive turbo decision feedback equalization method in response to a reception a packet including samples transmitted to the adaptive turbo decision feedback equalizer via a channel. The adaptive turbo decision feedback equalizer generates a first set of soft estimates of bits based upon a computation of a first feed-forward filter and a first feedback filter as a function of an estimation of the channel. The adaptive turbo decision feedback equalizer subsequently generates additional sets of soft estimates of the bits and a set of hard estimates of the bits based upon a computation of additional feed-forward filters and additional feedback filters as a function of a plurality of additional soft symbol estimates.

Abstract: In order to establish routing to/from a base station within a hybrid-cellular network, each network element is assigned a “class” based on a received signal strength of the base station. Each network element is allowed to choose a network element of lower class for relaying information to the base station.

Abstract: A communication system employs a HARQ-type retransmission scheme. Bits (701) received on a first transmission are stored and combined with the bits received on later transmissions thereby increasing the likelihood of a correct decoding on later transmissions. Similarly the bits received on the second or later transmissions are stored for combining with subsequent received bits. Specific information needed at the receiver is identified and requested from the transmitter. More particularly, information that is retransmitted in a second or later transmission in the HARQ scheme is determined from a reliability of individual constituent bits in the mother codeword or from an overall reliability of the received codeword. Based on these reliability metrics, the most unreliable set of the constituent bits are requested or, in the alternative, a specific number of constituent bits is requested.

Abstract: A communication system employs a HARQ-type retransmission scheme. Bits (701) received on a first transmission are stored and combined with the bits received on later transmissions thereby increasing the likelihood of a correct decoding on later transmissions. Similarly the bits received on the second or later transmissions are stored for combining with subsequent received bits. Specific information needed at the receiver is identified and requested from the transmitter. More particularly, information that is retransmitted in a second or later transmission in the HARQ scheme is determined from a reliability of individual constituent bits in the mother codeword or from an overall reliability of the received codeword. Based on these reliability metrics, the most unreliable set of the constituent bits are requested or, in the alternative, a specific number of constituent bits is requested.

Abstract: The invention provides an adaptive turbo decision feedback equalizer for executing an adaptive turbo decision feedback equalization method in response to a reception a packet including samples transmitted to the adaptive turbo decision feedback equalizer via a channel. The adaptive turbo decision feedback equalizer generates a first set of soft estimates of bits based upon a computation of a first feed-forward filter and a first feedback filter as a function of an estimation of the channel. The adaptive turbo decision feedback equalizer subsequently generates additional sets of soft estimates of the bits and a set of hard estimates of the bits based upon a computation of additional feed-forward filters and additional feedback filters as a function of a plurality of additional soft symbol estimates.

Abstract: The invention provides a novel compound 4-(p-methoxy-phenyl)-2-aminobutane exhibiting growth inhibition and antifeedant activity and represented by the structural formula. C11H17ON=4-(p-methoxy phenyl)-2-amino butane and an insecticidal composition comprising an effective amount of the novel compound and appropriate adjuvant.

Abstract: The invention provides a novel compound 4-(p-methoxy-phenyl)-2-aminobutane exhibiting growth inhibition and antifeedant activity and represented by the structural formula.

Abstract: The present invention relates to a process for the production of (−)3,4-divanillyl tetrahydrofiran of formula (2) which comprises (a) isolating) (−) secoisolariciresinol of formula (1) from the heartwood and roots of Taxus wallichiana by an improved process which consists of partitioning of the alcoholic extract of the heartwood and roots of T. wallichiana between water and chlorinated solvent, (b) extracting the chlorinated solvent extract with alkali and (c) isolating (−) secoisolariciresinol from the alkali extract upon neutralization with mineral acid and extracting with organic solvent and (d) crystallizing it from suitable organic solvent, (e) dissolving the isolated (−) secoisolariciresinol in suitable organic solvent and (f) reacting with triphenyl phosphine halide at 0-80° C. for 1-10 hours and (g) isolating (−) 3,4-divanillyl tetrahydrofuran by column chromatography.

Abstract: This invention relates to a process for the production of a compound (+) catechin penta acetate of formula I from Taxus wallichiana tissue cultures which comprises : (a) inoculation of explants on different media compositions supplemented with combinations of auxins (1-5 mg/l) and cytokinins (0.1-1.0 mg/l); (b) incubation of the cultures under continuous light or dark conditions for 4-6 weeks for callus cultures followed by subculturing at 4-6 weeks intervals; (c) harvesting of the calli at different growth phases ranging from 12-36 months; (d) extraction of fresh pulverized calli with polar solvents at room temperature; (e) evaporating the solvent to give a residue; and partitioning of the residue between water and chlorinated solvents and evaporating the solvent to a semisolid mass; (f) subjecting the resultant mass to column chromatography over suitable adsorbent and (g) eluting with organic solvent/mixtures of organic solvents to get (+) catechin penta acetate.

Abstract: The invention provides a process for the preparation of 4-(p-methoxyphenyl)-2-aminobutane represented by structural formula (1) as shown herein below: [C11H17ON=4-(p-methoxy phenyl)-2-amino butane] said process comprising the steps of, (a) isolating a phenolic compound 4-hydroxyphenyl)-butan-2-ol from the leaves of Taxus wallichiana by known methods, (b) treating the phenolic compound in aqueous mineral acid to obtain a phenolic halide derivative, (c) converting the phenolic halide derivative into its methyl ether by treating it with a methating agent, (d) reacting the methyl ether halide with azide to obtain an azido derivative, and (e) hydrogenating the azido compound to obtain 4-(p-methoxyphenyl)-2-aminobutane.