Polycyclo Ring System Having The Six-membered Hetero Ring As One Of The Cyclos Patents (Class 514/222.8)
1,2,4 - benzothiadiazine - 1,1 - dioxides (including hydrogenated) (Class 514/223.2)
  • Synergistic compositions comprising an oxathiazine and a benzothiophene-2-carboxamide-S,S-dioxide
    Patent number: 6242440
    Abstract: This invention relates to synergistic compositions of oxathiazines and benzothiophene-2-carboxamide-S,S-dioxides for use as fungicidal preservatives in the protection of materials, such as protection of wood, wood products, biodegradable materials and coatings.
    Type: Grant
    Filed: April 10, 2000
    Date of Patent: June 5, 2001
    Assignee: Janssen Pharmaceutica N.V.
    Inventors: Ludo Antoinnette De Witte, Alex Raymond Albert Valcke, Mark Arthur Josepha Van der Flaas, Willy Modest Louisa Willems
  • Fused 1,2,4-thiadiazine derivatives, their preparation and use
    Patent number: 6225310
    Abstract: 1,2,4-Thiadiazine and 1,4-thiazine derivates represented by formula (I): wherein A, B, D, R1, R2, R3 and R4 are defined in the description, compositions thereof and methods for preparing the compounds are described. The compounds are useful in the treatment of diseases of the central nervous system, the cardiovascular system, the pulmonary system, the gastrointestinal system and the endocrinological system.
    Type: Grant
    Filed: March 30, 2000
    Date of Patent: May 1, 2001
    Assignee: Novo Nordisk A/S
    Inventors: Flemming Elmelund Nielsen, John Bondo Hansen, Holger Claus Hansen, Tina Møller Tagmose, John Patrick Mogensen
  • Insecticidal dihydrooxadiazine compounds
    Patent number: 6197766
    Abstract: Insecticidal dihydrooxadiazine compounds having the formula: wherein X is O, N or S; R is a substituted or unsubstituted phenyl or C4-C5 heterocyclic group; R2, R3, R4, and R5 are one of the following: a) R2, R3, and R4 are, independently, hydrogen, alkyl, alkoxy, or furanyl; and R5 is nitro, cyano, alkyl, dialkylamino, alkylthio, alkoxy, haloalkoxy, phenoxy, phenylthio, or alkoxycarbonyl, wherein R3 and R5 together can form a ring; or b) R3, R4, and R5 are hydrogen; and R2 is alkylthio, alkylsulfinyl, alkylsulfonyl, nitroalkoxy, hydroxy, dialkoxyphosphinyl, cyano, acyloxy, alkoxy, haloalkoxy, cycloalkyl, or alkenyl; or R2 is a substituted or unsubstituted phenyl, phenylthio, phenylsulfinyl, phenylsulfonyl, pyrazolyl, furanyl, thienyl, phenylalkoxy, or benzoyloxy; and R6 is hydrogen, alkyl, alkylthio, alkoxyalkyl, acyl, benzyl, or alkoxycarbonyl.
    Type: Grant
    Filed: January 11, 1999
    Date of Patent: March 6, 2001
    Assignees: Uniroyal Chemical Company, Inc. and Uniroyal Chemical Co., Uniroyal Chemical Cie.
    Inventors: Sheldon Bernard Park, Anupama Mishra, Mark Achiel Dekeyser, Paul Thomas McDonald
  • Pyrano, piperidino, and thiopyrano compounds and methods of use
    Patent number: 6191140
    Abstract: The present invention provides novel compounds of formula I which may be useful in hyperpolarizing cell membranes, opening potassium channels, relaxing smooth muscle cells, and inhibiting bladder contractions.
    Type: Grant
    Filed: October 20, 1999
    Date of Patent: February 20, 2001
    Assignee: Abbott Laboratories
    Inventors: William A. Carroll, Konstantinos A. Agrios, Robert J. Altenbach, Irene Drizin, Michael E. Kort