Three Or More Ring Hetero Atoms In The Six-membered Hetero Ring Patents (Class 514/229.2)
  • Publication number: 20120094988
    Abstract: Treatment with N-(2-phenylethyl)succinamic acid or its salts protects against inhibition of growth by a neonicotinoid compound applied as a seed treatment or applied directly on or near the root zone of the seedling.
    Type: Application
    Filed: December 20, 2011
    Publication date: April 19, 2012
    Inventors: Franklin Paul Silverman, Dale O. Wilson, JR., Jennifer C. Kochan, Nicole Higgs, Peter D. Petracek, Prem Warrior, Karen S. Arthur
  • Publication number: 20120083491
    Abstract: The invention relates to novel insecticidal active compound combinations comprising, firstly, compounds which act as insecticides on nicotinergic acetylcholine receptors as agonists and antagonists, and at least one active compound from the group of the anthranilamides, which combinations are suitable for protecting plants against attack by pests.
    Type: Application
    Filed: December 12, 2011
    Publication date: April 5, 2012
    Applicant: BAYER CROPSCIENCE AG
    Inventors: Christian FUNKE, Reiner Fischer, Rüdiger Fischer, Heike Hungenberg, Wolfram Andersch, Wolfgang Thielert, Anton Kraus
  • Publication number: 20120083463
    Abstract: The present invention relates to active compound combinations consisting, firstly, of a known halogen-substituted derivative (component A) and, secondly, of further known pesticidally active compounds (component B), which active compound combinations are suitable for controlling animal and microbial pests.
    Type: Application
    Filed: July 8, 2011
    Publication date: April 5, 2012
    Applicant: Bayer CropScience AG
    Inventors: Michael MAUE, Friedrich August MÜHLTHAU, Isabelle ADELT, Markus HEIL, Peter JESCHKE, Tobias KAPFERER, Alexander SUDAU, Heike HUNGENBERG
  • Publication number: 20120077765
    Abstract: This invention recites naphthyl isoxazoline oxime derivatives of Formula (1) geometric isomers, stereoisomers thereof, pharmaceutically or veterinarily acceptable salts thereof, compositions thereof, and their use as a parasiticide in animals. The variables, R1a, R1b, R1c, R2, R3, and are as described herein.
    Type: Application
    Filed: September 15, 2011
    Publication date: March 29, 2012
    Applicant: PFIZER INC.
    Inventors: Michael Curtis, Edmund L. Ellsworth
  • Publication number: 20120058891
    Abstract: Novel dioxazine- and oxdiazine-substituted arylamides of the formula (I) in which A1, A2, R1, R2, R3, R4 and R5 are as defined in the description, a plurality of processes for preparing these compounds and their use for controlling pests, and also novel intermediates and processes for their preparation.
    Type: Application
    Filed: November 9, 2011
    Publication date: March 8, 2012
    Applicant: Bayer CropScience AG
    Inventors: Bernd-Wieland Krüger, Achim Hense, Bernd Alig, Rüdiger Fischer, Christian Funke, Ernst Rudolf Gesing, Olga Malsam, Mark Wilhelm Drewes, Christian Arnold, Peter Lümmen, Erich Sanwald
  • Publication number: 20120035165
    Abstract: The present invention relates to the use of a fungicidal composition comprising at least one carboxamide and at least one further compound selected from strobilurins or from triazoles, for controlling certain rust fungi, such as soy bean rust and coffee rust, in crop protection.
    Type: Application
    Filed: August 21, 2009
    Publication date: February 9, 2012
    Applicant: Bayer CropScience AG
    Inventors: Karl-Wilhelm Münks, Heiko Rieck, Ulrike Wachendorff-Neumann, Ingo Wetcholowsky, Jose Augusto Geraldes
  • Publication number: 20120034216
    Abstract: The present invention relates to spiroketal compounds that are useful in methods of treating or preventing protozoal infections, parasitic infections, bacterial infections, cell proliferative disorders and anti inflammatory disorders. The spiroketal compounds are also useful as immunosuppressive agents, and also in methods of controlling pests.
    Type: Application
    Filed: August 11, 2011
    Publication date: February 9, 2012
    Applicant: ECOBIOTICS LTD
    Inventors: Paul Warren Reddell, Victoria Anne Gordon
  • Publication number: 20120028971
    Abstract: The present application relates to novel alkylcarboxylic acids having an oxo-substituted azaheterocyclic partial structure, to processes for their preparation, to their use for the treatment and/or prevention of diseases, and to their use for producing medicaments for the treatment and/or prevention of diseases, especially for the treatment and/or prevention of cardiovascular disorders.
    Type: Application
    Filed: February 24, 2010
    Publication date: February 2, 2012
    Applicant: BAYER PHARMA AKTIENGESELLSCHAFT
    Inventors: Thomas Lampe, Michael Hahn, Johannes-Peter Stasch, Karl-Heinz Schlemmer, Frank Wunder, Stefan Heitmeier, Nils Griebenow, Sherif El Sheikh, Volkhart Min-Jian Li, Eva-Maria Becker, Friederike Stoll, Andreas Knorr
  • Publication number: 20120022054
    Abstract: The present invention concerns novel substituted aryl derivatives, their process of preparation and their use for inhibiting virus replication and for treating viral diseases or disorders such as HIV and/or HCV infection.
    Type: Application
    Filed: December 10, 2009
    Publication date: January 26, 2012
    Applicant: LABORATOIRE BIODIM
    Inventors: Richard Benarous, Sabine Barbey-Treve, Jean-Marc Paris, Sebastien Berrut, Clarisse Berlioz-Torrent, Stephane Emiliani
  • Publication number: 20120022021
    Abstract: The present invention relates to mixtures comprising a) a compound of the formula I in which X, m, Q and a are as defined in the description and b) one or more ethylene modulators (II) selected from the group consisting of: inhibitors of ethylene biosynthesis which inhibit the conversion of S-adenosyl-L-methionine into 1-aminocyclopropane-1-carboxylic acid (ACC), inhibitors of ethylene biosynthesis which block the conversion of ACC into ethylene, or inhibitors of ethylene action, and also to compositions comprising them and to their use for controlling harmful fungi.
    Type: Application
    Filed: September 28, 2011
    Publication date: January 26, 2012
    Applicant: BASF SE
    Inventors: Wilhelm RADEMACHER, John S. HARDEN, Dan E. WESTBERG, Joseph E. ZAWIERUCHA, Thomas J. HOLT, Hendrik YPEMA, Ted R. BARDINELLI, Albert C. EVERSON, Edson BEGLIOMINI
  • Publication number: 20120022055
    Abstract: The present invention provides a pest controlling composition comprising, as active ingredients, an amide compound of the formula (I) and a neonicotinoid compound; and so on.
    Type: Application
    Filed: February 24, 2010
    Publication date: January 26, 2012
    Inventors: Norihisa Sakamoto, Shinya Nishimura
  • Publication number: 20120022053
    Abstract: Compounds of the formula in which A is an unsubstituted or mono- to tetrasubstituted, aromatic or non-aromatic, monocyclic or bicyclic heterocyclic radical, where one to two of the substituents of A can be selected from the group consisting of halo-C1-C3alkyl, cyclopropyl, halocyclopropyl, C2-C3alkenyl, C2-C3alkynyl, halo-C2-C3alkenyl, halo-C2-C3alkynyl, halo-C1-C3alkoxy, C1-C3alkylthio, halo-C1-C3alkylthio, allyloxy, propargyloxy, allylthio, propargylthio, haloallyloxy, haloallylthio, cyano and nitro, and one to four of the substituents of A can be selected from the group consisting of C1-C3alkyl, C1-C3alkoxy and halogen; R is hydrogen, C1-C6alkyl, phenyl-C1-C4alkyl, C3-C6cycloalkyl, C2-C6alkenyl or C2-C6alkynyl; and X is N—NO2 or N—CN, and, if appropriate, tautomers thereof, in each case in free form or in salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se.
    Type: Application
    Filed: January 25, 2010
    Publication date: January 26, 2012
    Applicant: SYNGENTA CROP PROTECTION, INC.
    Inventors: Peter Maienfisch, Laurenz Gsell
  • Publication number: 20120010073
    Abstract: The present invention relates to novel active compound combinations which include of the insecticidally active compounds of the formula (I) in combination with fungicidally active compounds (II) and are highly suitable for controlling unwanted animal pests, such as insects, and unwanted phytopathogenic fungi.
    Type: Application
    Filed: July 7, 2011
    Publication date: January 12, 2012
    Applicant: BAYER CROPSCIENCE AG
    Inventors: Christian FUNKE, Heike HUNGENBERG, Rüdiger FISCHER
  • Publication number: 20120004103
    Abstract: Insecticidal compositions suitable for use in preparation of insecticidal liquid fertilizers comprising a pyrethroid, a hydrated aluminum-magnesium silicate, and at least one dispersant selected from the group consisting of a sucrose ester, a lignosulfonate, an alkylpolyglycoside, a naphthalenesulfonic acid formaldehyde condensate and a phosphate ester are disclosed.
    Type: Application
    Filed: September 9, 2011
    Publication date: January 5, 2012
    Applicant: FMC CORPORATION
    Inventor: Timothy Martin
  • Publication number: 20120004104
    Abstract: Selective insect neonicotinoids is a class of pesticide active ingredients that share some characteristics in their chemical structures and bind to the nAChR acetylcholine receptors. Formulation of such compounds in oil suspension or oil dispersion is challenging due to their electrostatic interactions of the heteroatoms in oily media, that lead to irreversible flocculation or diminished homogeneicity and bleeding of such oil dispersions. Imidacloprid, Thiamethoxam, Thiachloprid, Nitenpyram, Acetamiprid, Clothianidin and Dinetofuran and derivatives thereof with nAChR binding ability are successfully formulated in oil suspension with the use of certain copolymeric anionic fatty-acid based dispersants, sorbitan derivatives, ionic surfactants, other non-ionic surfactants and inorganic polyvalent cationic salt dispersed in the oil.
    Type: Application
    Filed: March 4, 2010
    Publication date: January 5, 2012
    Applicant: GAT Microencapsulation AG
    Inventors: Victor Casaña Giner, Miguel Gimeno Sierra, Barbara Gimeno Sierra
  • Publication number: 20110319401
    Abstract: This invention discloses that the five crystal forms of XLF-III-43 can be used as crude drugs. The invention also relates to the preparation methods of the five crystal forms of XLF-III-43 as crude drugs, to the applications of the sterling of the five crystal forms of XLF-III-43 and mixed crystals in different proportions as medicinally active components to develop various kinds of medicines and compound medicines. In addition, this invention also relates to applying the crystal samples of XLF-III-43 as crude drugs to treat kidney dysfunction, cardiocerebral vessel diseases, hypertension, type II diabetic mellitus, complications of hypertension and diabetic mellitus, tumor, precancerosis, edema, and achieves therapeutic effects by enhancing blood drug levels resulted from effects of crystal forms in the processes of treating all kinds of diseases.
    Type: Application
    Filed: November 28, 2009
    Publication date: December 29, 2011
    Applicant: INSTITUTE OF MATARIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES
    Inventors: Yang Lv, Xiaoguang Chen, Ping Xie, Li Zhang, Cheng Wang
  • Publication number: 20110319262
    Abstract: A combination, suitable for agricultural use comprising (I): a compound of formula (X) and (II): one or more agents selected, independently of each other, from any one of (A) to (G): (A) a certain fungicide; (B) a certain insecticide and/or nematicide; (C) a certain protein produced by the plant pathogenic bacterium, Erwinia amylovora; (D) a certain biological strain, (E) a certain Isoflavone; (F) a plant growth regulator; and (G) a plant activator, wherein compound of formula (X) is:
    Type: Application
    Filed: September 16, 2009
    Publication date: December 29, 2011
    Applicant: SYNGENTA CROP PROTECTION, LLC
    Inventors: Michael Schade, Christoph Grimm, Martin Faerber, Dieter Hofer, Kaspar Müller, Scott Campbell
  • Publication number: 20110311503
    Abstract: The novel active ingredient combinations which consist of the compounds of the formula (I) in combination with further active insecticidal ingredients (II) are very suitable for control of animal pests such as insects and/or unwanted acarids.
    Type: Application
    Filed: June 16, 2011
    Publication date: December 22, 2011
    Applicant: BAYER CROPSCIENCE AG
    Inventors: Christian FUNKE, Heike HUNGENBERG, Rüdiger FISCHER
  • Publication number: 20110306502
    Abstract: A water dispersible granular composition comprising: at least one solid agrochemically active substance; at least one sorptive filler; at least one first agrochemically acceptable excipient; at least one liquid or low melting agrochemically active substance; and, at least one second agrochemically acceptable excipient. The invention further relates to a process of preparing the water dispersible granular composition.
    Type: Application
    Filed: January 26, 2009
    Publication date: December 15, 2011
    Inventors: Deepak Pranjivandas Shah, Puthenveetil Kunjukrishna Menon Ramdas, Balachandran Thankappan Vadakkekuttu
  • Publication number: 20110306593
    Abstract: In its many embodiments, the present invention provides a novel class of heterocyclic compounds of the formula: as modulators of gamma secretase, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more disease associated with the central nervous system using such compounds or pharmaceutical compostions.
    Type: Application
    Filed: November 11, 2009
    Publication date: December 15, 2011
    Inventors: Zhaoning Zhu, William J. Greenlee, Hongmei Li, Monica L. Vicarel, Jun Qin, Pawan Kumar Dhondi, Xianhai Huang, Anandan Palani, Xiaoxiang Liu, Zhong-Yue Sun, Hubert B. Josien, Ruo Xu, David James Cole, Duane A. Burnett, Chad E. Bennett, Troy McCracken, Malcolm MacCoss
  • Patent number: 8076328
    Abstract: Process for the protection of fish and invertebrates and all their stages of development against or for the treatment of mycoses caused by fungi of the genera Saprolegnia, Aphanomyces, Achlyaflagellata and other species important in aquacultures by use of 2-[[[[1-[3-(1-fluoro-2-phenylethyl)oxy]phenyl]ethylidene]amino]oxy]methyl]alpha-(methoxyimino)-N-methyl-alphaE-benzeneacetamide, amisulbrom, cyazofamid, enestrobin, famoxadone, fenamidone, fluoxastrobin, orysastrobin, picoxystrobin and pyribencarb. This use leads to an inhibition or destruction of pathogenic fungi. The composition, comprising at least one fungicide selected from the abovementioned group for use in fish farming and keeping is suitable for the prophylaxis and therapy of diseases of fish in aquaculture, in breeding ponds, breeding tanks, aquariums, natural stretches of game fish waters, ponds, and marine fish farms. Addition to the water and feed and direct application are the associated use forms.
    Type: Grant
    Filed: April 8, 2008
    Date of Patent: December 13, 2011
    Assignee: Bayer CropScience AG
    Inventors: Isolde Häuser-Hahn, Klaus Stenzel, Ulrike Wachendorff-Neumann
  • Publication number: 20110301029
    Abstract: The present invention relates to plant-protecting active ingredient mixtures comprising, as active components, a neonicotinoid and one or two fungicides selected from pyraclostrobin and boscalid, in synergistically effective amounts and to a method of improving the health of plants by to the plants or the locus thereof by applying said mixtures.
    Type: Application
    Filed: August 15, 2011
    Publication date: December 8, 2011
    Applicant: BASF SE
    Inventors: Dirk VOESTE, Martin P. MASCIANICA, Hendrik YPEMA, Henry Van Tuyl COTTER
  • Patent number: 8071590
    Abstract: A subject of the invention is the compounds of formula (I): wherein R1, R2, R3, R?3, R4, R?4, R5, R6 and R7 are as described in the application, in the form of enantiomers or mixtures, as well as their salts with acids and bases, their preparation and their application as anti-bacterials, in both human and veterinary medicine.
    Type: Grant
    Filed: June 23, 2009
    Date of Patent: December 6, 2011
    Assignee: Vetoquinol SA
    Inventors: Sandrine Ropp, Christophe Morice, Bruno Giethlen, Paola Ciapetti, Florence Chery-Mozziconacci, Camille G. Wermuth, Francoise Leblanc, Marc Schneider
  • Publication number: 20110293533
    Abstract: Disclosed are mixtures and compositions for controlling invertebrate pests relating to combinations comprising (a) 3-bromo-N-[4-chloro-2-methyl-6-[(methylamino)carbonyl]phenyl]-1-(3-chloro-2-pyridinyl)-1H-pyrazole-5-carboxamide, and its N-oxides, and suitable salts thereof and a component (b) wherein the component (b) is at least one compound or agent selected from neonicotinoids, cholinesterase inhibitors, sodium channel modulators, chitin synthesis inhibitors, ecdysone agonists, lipid biosynthesis inhibitors, macrocyclic lactones, GABA-regulated chloride channel blockers, juvenile hormone mimics, ryanodine receptor ligands, octopamine receptor ligands, mitochondrial electron transport inhibitors, nereistoxin analogs, pyridalyl, flonicamid, pymetrozine, dieldrin, metaflumizone, biological agents, and suitable salts of the foregoing.
    Type: Application
    Filed: August 11, 2011
    Publication date: December 1, 2011
    Applicant: E.I. DU PONT NEMOURS AND COMPANY
    Inventors: Isaac Billy Annan, John Lindsey Flexner, Hector Eduardo Portillo, George Philip Lahm, Thomas Paul Selby, Thomas Martin Stevenson
  • Publication number: 20110294756
    Abstract: In its many embodiments, the present invention provides a novel class of heterocyclic compounds of Group A or Group, as defined herein, as modulators of gamma secretase, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more diseases associated with the central nervous system using such compounds or pharmaceutical compositions.
    Type: Application
    Filed: November 12, 2009
    Publication date: December 1, 2011
    Inventors: Zhaoning Zhu, William J., Xianhai Huang, Jun Qin, XIaoxiang Liu, Hongmei Li, Wei Zhou, Anandan Palani, Xiaohong Zhu, Monica L. Vicarel, Mihirbaran Mandal, Zhong-Yue Sun, Chad E. Bennett, Troy Michael McCracken, Gioconda V. Gallo
  • Publication number: 20110275583
    Abstract: Novel active compound combinations comprising compounds of the formula (I) and compounds of the formula (II) have very good insecticidal and acaricidal properties.
    Type: Application
    Filed: April 28, 2011
    Publication date: November 10, 2011
    Applicant: Bayer CropScience AG
    Inventors: Thomas BRETSCHNEIDER, Heike HUNGENBERG, Martin Füsslein
  • Publication number: 20110275520
    Abstract: Polymeric materials are provided that are produced from a blend of hydrophilic and hydrophobic biodegradable polymers. The polymeric materials can form fibers, nonwoven fabrics, films, coatings, pellets, capsules, etc. A compound can be incorporated in the polymeric materials. The delivery of the compound can be controlled by diffusion of the compound from the polymeric material and during biodegradation of the polymeric material. The release rate is controlled by varying the composition of the polymeric material to control diffusion rates of the compound and/or biodegradation rate of the polymeric material. This technology provides methods for delivering and controlling release rates of pesticides and related compounds in agricultural and non-agricultural settings. When adhered to plants or plant parts, the polymeric materials can provide protection from insect and disease pests. In pellet or capsule form, pesticides can be delivered into seed furrows along with crop seeds, providing similar protection.
    Type: Application
    Filed: September 30, 2009
    Publication date: November 10, 2011
    Inventors: Margaret W. Frey, Chunhui Xiang, Michael P. Hoffmann, Alan G. Taylor, Jeffrey Gardner
  • Publication number: 20110263586
    Abstract: A pest controlling composition comprising tolclofos-methyl and a neonicotinoid compound represented by the formula (1) as active ingredients.
    Type: Application
    Filed: November 20, 2009
    Publication date: October 27, 2011
    Applicant: SUMITOMO CHEMICAL COMPANY, LIMITED
    Inventors: Masato Soma, Atsushi Iwata
  • Publication number: 20110263421
    Abstract: The present invention provides a composition for controlling pests comprising, as active ingredients, ethaboxam and a neonicotinoid compound represented by formula (1).
    Type: Application
    Filed: November 20, 2009
    Publication date: October 27, 2011
    Inventors: Makoto Kurahashi, Yuichi Matsuzaki
  • Publication number: 20110263585
    Abstract: The present invention relates to polypeptides, preferably from Drosophila melanogaster (DmShaI) as target for insecticides.
    Type: Application
    Filed: November 5, 2009
    Publication date: October 27, 2011
    Applicant: BASF SE
    Inventors: Paul Bernasconi, John Dorsch, Lynn Stam, Scott Zitko, Nancy B. Rankl, Mike Griswold, Franz-Josef Braun, Gang Lu, Robert D. Kirkton, Barbara Wedel, Joachim Dickhaut, Angela Hofhine, Jennifer Zink, Fae Malone, Daniel Houtz, Steffen Gross, Ramani Kandasamy, Damian London, Thomas M. Gurganus
  • Publication number: 20110263520
    Abstract: Disclosed is a composition for use in controlling harmful organisms, comprising as active ingredients at least one of 16-keto aspergillimide, its enantiomers, their mixture, or their acid addition salts and at least one of other harmful organism control agents. The present invention provides a composition for use in controlling harmful organisms that has excellent insecticidal activity or penetrative transferable insecticidal activity against a wide range of harmful organisms, particularly agricultural and horticultural insect pests.
    Type: Application
    Filed: December 21, 2009
    Publication date: October 27, 2011
    Inventors: Ryo Horikoshi, Masahiro Nomura, Satoshi Nakamura, Mizuki Hayashimoto, Mariko Tsuchida, Kazuhiko Oyama, Masaaki Mitomi
  • Publication number: 20110257166
    Abstract: The present invention provides an aqueous suspoemulsion comprising (a) an oil phase comprising (i) at least one triazole active compound as emulsified component, solid at room temperature, (ii) at least one alkyl carboxylic acid amide as a solvent and a crystal growth inhibitor, and (iii) a polymeric stabilizer, and (b) a continuous water phase comprising (i) at least one strobilurin active compound as suspended solid component, solid at room temperature, (ii) at least one dispersant selected from the group consisting of methacrylic acid-methyl methacrylate-polyethyleneglycol graft copolymer, tristyrylphenolethoxylates and/or propylene oxide/ethylene oxide block copolymer with 10% to 50% EO, preferably with 20% to 50% EO and most preferably with 30% to 40% EO, (iii) water, and (iiii) additives, if appropriate. a process for preparing the suspoemulsion and its use for applying the active compounds comprised therein to plants and/or their habitat are also provided.
    Type: Application
    Filed: January 11, 2010
    Publication date: October 20, 2011
    Applicant: ROTAM AGROCHEM INTERNATIONAL CO., LTD.
    Inventors: Antonio Carlos Damaceno, Jose Gilberto Hermann
  • Publication number: 20110251062
    Abstract: The invention relates to active compound combinations, in particular within a fungicide composition, which comprises (A) a compound of formula (I) and at least one further respiratory chain complex in inhibitor (B). Moreover, the invention relates to a method for curatively or preventively controlling the phytopathogenic fungi of plants or crops, to the use of a combination according to the invention for the treatment of seed, to a method for protecting a seed and not at least to the treated seed.
    Type: Application
    Filed: December 5, 2009
    Publication date: October 13, 2011
    Applicant: Bayer Corp Science AG
    Inventors: Burkhard Schütz, Peter Dahmen, Ulrike Wachendorff-Neumann, Peter Herold
  • Publication number: 20110230475
    Abstract: Plant propagation material expressing aphid resistance and application of an insecticide to the plant propagation material.
    Type: Application
    Filed: September 24, 2009
    Publication date: September 22, 2011
    Applicant: SYNGENTA CROP PROTECTION, LLC
    Inventors: Clifford Watrin, Virgil Sparks
  • Patent number: 8022067
    Abstract: Disclosed are mixtures and compositions for controlling invertebrate pests relating to combinations comprising (a) 3-bromo-N-[4-chloro-2-methyl-6-[(methylamino)carbonyl]phenyl]-1-(3-chloro-2-pyridinyl)-1H-pyrazole-5-carboxamide, and its N-oxides, and suitable salts thereof and a component (b) wherein the component (b) is at least one compound or agent selected from neonicotinoids, cholinesterase inhibitors, sodium channel modulators, chitin synthesis inhibitors, ecdysone agonists, lipid biosynthesis inhibitors, macrocyclic lactones, GABA-regulated chloride channel blockers, juvenile hormone mimics, ryanodine receptor ligands, octopamine receptor ligands, mitochondrial electron transport inhibitors, nereistoxin analogs, pyridalyl, flonicamid, pymetrozine, dieldrin, metaflumizone, biological agents, and suitable salts of the foregoing.
    Type: Grant
    Filed: June 30, 2005
    Date of Patent: September 20, 2011
    Assignee: E. I. du Pont de Nemours and Company
    Inventors: Isaac Billy Annan, John Lindsey Flexner, Hector Eduardo Portillo, George Philip Lahm, Thomas Paul Selby, Thomas Martin Stevenson
  • Publication number: 20110224075
    Abstract: The present invention relates to pesticidal mixtures comprising as active compounds 1) at least one aminothiazoline compound I of formula I: wherein R1 is selected from hydrogen, COCH3, COCH2CH3 or COCH2C(CH3)3; R2 and R3 together with the carbon atoms of the phenyl ring to which they are attached form a ring which, depending on the tautomeric formula I a) or b) is depicted as: a benzene ring, a saturated 5-, 6-, or 7-membered carbocycle, a partially unsaturated 5-, 6-, or 7-membered carbocycle, a 5-, 6-, or 7-membered saturated heterocycle, a partially unsaturated 5-, 6-, or 7-membered heterocycle, which heterocycles contain 1, 2, or 3 heteroatoms selected from O, S and N as ring members, and a 5- or 6-membered heteroaromatic ring which contains 1, 2, or 3 heteroatoms selected from O, S and N as ring members, and wherein the ring is unsubstituted or may carry any combination of 1, 2, 3, or 4 radicals selected from the group consisting of halogen, CH3, CH2CH3, CF3, CH3O, cyano and (?O) (oxo); R4 is se
    Type: Application
    Filed: March 24, 2009
    Publication date: September 15, 2011
    Applicant: BASF SE
    Inventors: Markus Kordes, Ronan Le Vezouet, Jurgen Langewald, Ralph Paulini, Deborah L. Culbertson, Douglas D. Anspaugh, Luiz Antonio Jose, Hassan Oloumi-Sadeghi
  • Publication number: 20110224200
    Abstract: Provided is a novel prophylactic or therapeutic agent for a chorioretinal degenerative disease. The compound of formula (1) or its salt has inhibitory effects on photoreceptor cell death or visual cell death in a mouse model of light damage. Therefore, the compound or its salt is useful as a prophylactic or therapeutic agent for a chorioretinal degenerative disease such as age-related macular degeneration, retinitis pigmentosa. In the formula (1), A is a group (p1), (p2) or (p3); R1 is H, alkyl, aralkyl or OH or its ester; R2 is H or alkyl; R3 is halogen, H, alkyl or OH or its ester; R4 is halogen, H, OH, alkoxy, amino, alkylamino or cycloalkylamino, R3 and R4 may be joined to each other through N to form an unsaturated [1,2,4]oxadiazine ring; R5 is H, alkyl or cycloalkyl; m is 0 or 1; and n is 0 or 1.
    Type: Application
    Filed: November 18, 2009
    Publication date: September 15, 2011
    Inventors: Shin-ichiro Hirai, Atsushi Yoshida
  • Publication number: 20110218100
    Abstract: The present invention relates to novel active compound combinations comprising a known carboxamide, a known azole and additionally a second known azole or alternatively a known strobilurin, which combinations are highly suitable for controlling unwanted phytopathogenic fungi.
    Type: Application
    Filed: May 4, 2011
    Publication date: September 8, 2011
    Applicant: Bayer CropScience AG
    Inventors: Peter Dahmen, Ulrike Wachendorff-Neumann, Isolde Häuser-Hahn, Hans-Ludwig Elbe, Ralf Dunkel, Anne Suty-Heinze
  • Publication number: 20110218194
    Abstract: Disclosed are compounds of the formula I or a stereoisomer, tautomer, or pharmaceutically acceptable salt or solvate thereof, wherein W is a bond, —C(?S)—, —S(O)—, —S(O)2—, —C(?O)—, —O—, —C(R6)(R7)—, —N(R5)— or —C(?N(R5))—; X is —O—, —N(R5)— or —C(R6)(R7)—; provided that when X is —O—, U is not —O—, —S(O)—, —S(O)2—, —C(?O)— or —C(?NR5)—; U is a bond, —S(O)—, —S(O)2—, —C(O)—, —O—, —P(O)(OR15)—, —C(?NR5)—, —(C(R6)(R7))b— or —N(R5)—; wherein b is 1 or 2; provided that when W is —S(O)—, —S(O)2—, —O—, or —N(R5)—, U is not —S(O)—, —S(O)2—, —O—, or —N(R5)—; provided that when X is —N(R5)— and W is —S(O)—, —S(O)2—, —O—, or —N(R5)—, then U is not a bond; and R1, R2, R3, R4, R5, R6, and R7 are as defined in the specification; and pharmaceutical compositions comprising the compounds of formula I.
    Type: Application
    Filed: May 16, 2011
    Publication date: September 8, 2011
    Applicant: Schering Corporation & Pharmacopeia Drug Discovery Inc.
    Inventors: Zhaoning Zhu, Brian A. Mckittrick, Zhong-Yue Sun, Yuanzan C. Ye, Johannes H. Voight, Corey Strickland, Elizabeth M. Smith, Andrew Stamford, William J. Greenlee, Robert Mazzola, John Caldwell, Jared N. Cumming, Lingyan Wang, Yusheng Wu, Ulrich Iserloh, Tao Guo, Thuy X. H. Le, Kurt W. Saionz, Suresh D. Babu, Rachel C. Hunter, Michelle L. Morris, Huizhong Gu, Gang Qian, Dawit Tadesse
  • Publication number: 20110218188
    Abstract: The present invention relates to phenyl-pyrimidinyl-amino derivatives of formula (I) wherein Q1 and p, Ra to Rc, L1, Y, L2 and Q2 represent various substituents, their process of preparation, preparation intermediate compounds, their use as fungicide active agents, particularly in the form of fungicide compositions, and methods for the control of phytopathogenic fungi, notably of plants, using these compounds or compositions.
    Type: Application
    Filed: November 12, 2009
    Publication date: September 8, 2011
    Inventors: Christian Beier, Jurgen Benting, Isabelle Christian, Pierre-Yves Coqueron, Peter Dahmen, Ralf Dunkel, Jorg Greul, Marie-Claire Grosjean-Cournoyer, Hiroyuki Hadano, Philippe Rinolfi, Arnd Voerste, Jean-Pierre Vors, Ulrike Wachendorff-Neumann
  • Publication number: 20110212949
    Abstract: The present application relates to the use of heterocyclic compounds, some of which are known, for controlling animal pests, including arthropods and in particular insects, furthermore to novel heterocyclic compounds and to processes for their preparation.
    Type: Application
    Filed: July 4, 2009
    Publication date: September 1, 2011
    Inventors: Thomas Bretschneider, Eva-Maria Franken, Ulrich Görgens, Martin Füßlein, Achim Hense, Joachim Kluth, Hans-Georg Schwarz, Adeline Köhler, Olga Malsam, Arnd Voerste, Angela Becker
  • Publication number: 20110200684
    Abstract: Synergistic pesticidal mixtures are provided.
    Type: Application
    Filed: April 28, 2011
    Publication date: August 18, 2011
    Applicant: DOW AGROSCIENCES LLC
    Inventors: Jim X. Huang, Jonathan M. Babcock, Thomas Meade, Marc Farrow
  • Publication number: 20110195961
    Abstract: The invention relates to antibacterial compounds of formula I wherein is a bond or is absent, V is CH, CR6 or N; R0 is H or, if is a bond, may also be alkoxy; R1 is notably H or halogen; U is CH or N when is a bond, or, if is absent, U is CH2, NH or NR9; R2 is H, alkylcarbonyl or —CH2—R3; R3 is H, alkyl or hydroxyalkyl; R4 is H or, if n is not 0 and R5 is H, may also be OH; R5 is H, alkyl, hydroxyalkyl, aminoalkyl, alkoxyalkyl, carboxy or alkoxycarbonyl; R6 is hydroxyalkyl, carboxy, alkoxycarbonyl or —(CH2)q—NR7R8, q being 1, 2 or 3 and each of R7 and R8 independently being H or alkyl or R7 and R8 forming with the N atom bearing them a ring; R9 is alkyl or hydroxyalkyl; A is —(CH2)p—, —CH2CH2CH(OH)— or —COCH2CH(OH)—; G is substituted phenyl or G1 or G2 wherein Q is O or S and X is CH or N; and Y1, Y2 and Y3 may each be CH or N; and n is 0 when A is —CH2CH2CH(OH)— or —COCH2CH(OH)—, and n is 0, 1 or 2 when A is —(CH2)p—, p being 1, 2, 3 or 4, with the proviso that the sum of n and p is then 2, 3 or
    Type: Application
    Filed: October 6, 2009
    Publication date: August 11, 2011
    Applicant: Actelion Pharmaceuticals Ltd.
    Inventors: Christian Hubschwerlen, Daniel Ritz, Georg Rueedi, Jean-Philippe Surivet, Cornelia Zumbrunn-Acklin
  • Publication number: 20110190121
    Abstract: The invention relates to active compound combinations, in particular a fungicidal and/or insecticidal composition, comprising Isotianil (3,4-dichloro-N-(2-cyanophenyl)-5-isothiazolecarboxamide) and at least one further insecticide of the anthranilamide group and optionally one further insecticide of the neonicotinoids. Moreover, the invention relates to a method for curatively or preventively controlling the phytopathogenic fungi and/or microorganisms and/or pests of plants or crops, to the use of a combination according to the invention for the treatment of seed, to a method for protecting a seed and not at least to the treated seed.
    Type: Application
    Filed: November 28, 2008
    Publication date: August 4, 2011
    Applicant: Bayer CropScience AG
    Inventors: Lutz Assmann, Ulrike Wachendorff-Neumann, Peter Dahmen, Heike Hungenberg, Wolfgang Thielert
  • Publication number: 20110189294
    Abstract: A formulated composition suitable for controlling or preventing pathogenic damage in a plant comprising (A) at least one solid active ingredient having a water solubility of at most 100 ?g/litre at 25° C. at neutral pH, in an amount of at least 1 weight %, based on the total weight of the formulated composition, (B) at least one non-ionic surface active compound having a hydrophile-lipophile balance (HLB) of between 10 and 18, one or more customary formulation auxiliaries, and water; wherein active ingredient (A) is suspended or dispersed in the water, the weight ratio of surface active compound (B) to active ingredient (A) is in the range of from 1.5 to 15.0, provided the minimum amount of surface active compound (B) is at least 6 weight %, based on the total weight of the formulated composition. Also a method of improving pesticide residue levels in agriculture.
    Type: Application
    Filed: May 25, 2009
    Publication date: August 4, 2011
    Applicant: SYNGENTA CROP PROTECTION, INC.
    Inventors: Jason Keiper, Joshua Koon, Sarah Beth Cush, Michael James Hopkinson, Johnny D. Reynolds, Jorge Cisneros, Jennifer Peterson, Roy Boykin
  • Publication number: 20110183970
    Abstract: A synergistic insecticide composition comprising: a) an ethoxylated surfactant of the formula: R—O—(CH2—CH2O)x—H wherein R is a linear alkyl group of from approximately 0 to 15 carbon atoms and X has an average value from about 1 to 3; and b) an insecticide selected from the group consisting of nicotinoids, chlorfenapyr, pyrethrum and piperonyl butoxide. Such compositions are effective against a wide range of insects.
    Type: Application
    Filed: April 1, 2011
    Publication date: July 28, 2011
    Applicant: BASF CORPORATION
    Inventor: Steven R. Sims
  • Publication number: 20110183012
    Abstract: Pesticidal mixtures comprising, as active components, 1) an anthranilamid compound of the formula I wherein Q is H, Cl, Cr, I, CN or methyl; B1 is halogen, alkyl, haloalkyl, or haloalkoxy; B2 is halogen, haloalkyl, alkoxy, haloalkoxy, alkenyloxy, alkynyloxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, alkyl-S(?O)x—O— or haloalkyl S(O)x—O—, wherein x is 1 or 2 and the alkoxy radical may be substituted, or C(Ri)?N—ORj, C(Ri)?N(RjRk), wherein Ri, Rj and Rk are alkyl; R is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, alkylene-cycloalkyl, wherein these groups are optionally substituted; R1 is F, Cl, Br, methyl or trifluoromethyl; or the enantiomers or salts or N-oxides thereof, n is 1, 2 or 3; and 2) one or more compounds II selected from group A consisting of organo(thio)-phosphates, carbamates, pyrethroids, growth regulators, nicotinic receptor agonists/antagonists compounds, GABA antagonist compounds, macrocyclic lactone insecticides, METI I acaricides,
    Type: Application
    Filed: January 12, 2007
    Publication date: July 28, 2011
    Applicant: BASF Aktiengesellschaft
    Inventors: Markus Gewehr, Michael Puhl, Joachim Dickhaut, Henricus Maria Martinus Bastiaans, Douglas D. Anspaugh, David G. Kuhn, Hassan Oloumi-Sadeghi, Nigel Armes
  • Patent number: 7973083
    Abstract: A pesticidally active combination comprising an HPPD-inhibiting herbicide in the form of an agrochemically acceptable salt and an insecticide is disclosed, provided that the HPPD inhibiting herbicide is not a compound of formula (A) wherein Ra is C1-2 alkyl or chloro; Rb is hydrogen or C1-4 alkyl; and Rc is C1-4 alkyl is disclosed.
    Type: Grant
    Filed: November 3, 2004
    Date of Patent: July 5, 2011
    Assignee: Syngenta Crop Protection LLC
    Inventors: Christopher Glen Clemens, Willy Thaddaeus Rueegg, Michael Joseph Urwiler
  • Publication number: 20110159065
    Abstract: The present invention provides an agricultural chemical composition containing an agricultural chemical active ingredient A, a sorbitan fatty acid ester and a wax, and a production process thereof. In addition, the present invention provides an agricultural chemical sheet or a fruit bag in which the agricultural chemical composition is retained, and a production process thereof.
    Type: Application
    Filed: August 24, 2009
    Publication date: June 30, 2011
    Applicant: Nippon Soda Co., Ltd.
    Inventors: Kaoru Nishimura, Takao Iwasa
  • Publication number: 20110159110
    Abstract: The present invention provides a plant disease control agent containing at least one of tetrazoyloxime derivatives and salts thereof, and at least one selected from the group consisting of fosetyl, propamocarb, basic copper chloride, chlorothalonil, manzeb, cymoxanil, folpet, iminoctadine, cyazofamid, metalaxyl, fludioxonil, tebuconazole, prothioconazole, thiamethoxam, azoxystrobin and salts thereof.
    Type: Application
    Filed: March 24, 2009
    Publication date: June 30, 2011
    Applicant: Nippon Soda Co., Ltd.
    Inventors: Ichirou Urihara, Atsunori Isshiki, Hiroyasu Hosokawa, Tomoyuki Saiga