Additional Ring Containing Patents (Class 544/211)
  • Patent number: 4534789
    Abstract: N-(Heterocycliccarbamoyl)arylsulfonamides, such as N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-hydroxybenzenesulfonamide , methanesulfonate are useful for plant growth retardation, brush control and weed control in crops.
    Type: Grant
    Filed: October 21, 1983
    Date of Patent: August 13, 1985
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: James J. Reap
  • Patent number: 4523947
    Abstract: There are described triazine derivatives of the formula I ##STR1## wherein R.sub.1, R.sub.2 and R.sub.3 independently of one another are each C.sub.1 -C.sub.5 -alkyl which is unsubstituted or monosubstituted by C.sub.3 -C.sub.6 -cycloalkyl, or mono- or polysubstituted by halogen, or is C.sub.3 -C.sub.6 - cycloalkyl which is unsubstituted or mono- or polysubstituted by halogen, or one of the substituents R.sub.1, R.sub.2 and R.sub.3 is also halogen or --NR.sub.4 R.sub.5, in which R.sub.4 is hydrogen or C.sub.1 -C.sub.5 -alkyl and R.sub.5 is hydrogen, C.sub.1 -C.sub.5 -alkyl, monochloroacetyl or dichloroacetyl. The triazine derivatives are used for the protection of maize and sorghum plants against the harmful effects of herbicidal chloroacetanilides and chloroacetamides.
    Type: Grant
    Filed: May 29, 1984
    Date of Patent: June 18, 1985
    Assignee: Ciba-Geigy Corporation
    Inventors: Henry Szczepanski, Dagmar Berrer
  • Patent number: 4521597
    Abstract: A novel process for producing sulfonylureas of the formula I having a herbicidal action and an action regulating plant growth ##STR1## wherein A is an unsubstituted or substituted phenyl, naphthyl, furan, thiophene or pyridine group, E is a nitrogen atom or the methine group, R.sub.a is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.1 -C.sub.5 -haloalkyl, C.sub.1 -C.sub.5 -alkoxy, C.sub.1 -C.sub.5 -haloalkoxy, C.sub.1 -C.sub.5 -alkylthio or C.sub.2 -C.sub.10 -alkoxyalkoxy, and R.sub.b is the same as R.sub.
    Type: Grant
    Filed: October 14, 1983
    Date of Patent: June 4, 1985
    Assignee: Ciba Geigy Corporation
    Inventors: Haukur Kristinsson, Werner Topfl
  • Patent number: 4518776
    Abstract: There is described a process for producing sulfonylureas of the formula ##STR1## wherein G is an unsubstituted or substituted furanyl, thienyl, pyrrolyl, pyridinyl or phenyl radical,X is alkyl, haloalkyl, alkoxy, alkylthio, halogen, haloalkoxy, alkylamino or dialkylamino,Y is alkyl, alkoxy or haloalkoxy,Z is a nitrogen atom or the methyne group --CH.dbd..This novel process comprises reacting a sulfonamide of the formulaG--SO.sub.2 --NH.sub.2,in the presence of a base, with a chloroformic acid ester of the formulaCl--CO--Q--T,or a sulfonyl chloride of the formulaG--SO.sub.2 Cl,in the presence of a base, with a urethane of the formulaH.sub.2 N--CO--Q--T;and converting the formed carbamate of the formulaG--SO.sub.2 --NH--CO--Q--Tby reaction with an amine of the formula ##STR2## into the sulfonylurea of the above formula. There is also described novel sulfonylcarbamates of the above formula as intermediates.
    Type: Grant
    Filed: July 8, 1983
    Date of Patent: May 21, 1985
    Assignee: Ciba Geigy Corporation
    Inventors: Willy Meyer, Werner Fory, Werner Topfl
  • Patent number: 4515626
    Abstract: N-(Cyclopropyl-triazinyl- and -pyrimidinyl)-N'-arylsulfonyl ureas of the formula ##STR1## wherein Ar is a phenyl group ##STR2## or a naphthyl group ##STR3## and Q is a group X-A or R.sub.3,A is a C.sub.3 -C.sub.6 -alkynyl group, a C.sub.1 -C.sub.6 -alkyl group which is unsubstituted or substituted by halogen, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -alkylsulfinyl, C.sub.1 -C.sub.4 -alkylsulfonyl, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -haloalkylthio, C.sub.1 -C.sub.4 -haloalkylsulfinyl or C.sub.1 -C.sub.4 -haloalkylsulfonyl, or a C.sub.2 -C.sub.6 -alkenyl group which is unsubstituted or substituted by the groups given in the foregoing for C.sub.1 -C.sub.6 -alkyl, or A is a phenyl or benzyl group,E is the methine group or nitrogen,X is oxygen, sulfur, or a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur,R.sub.1 is hydrogen, C.sub.1 -C.sub.4 -alkyl or C.sub.1 -C.sub.4 -alkoxy,R.sub.2 is halogen, C.sub.1 -C.sub.3 -alkyl, C.sub.1 -C.sub.3 -haloalkyl, C.sub.1 -C.sub.
    Type: Grant
    Filed: September 26, 1983
    Date of Patent: May 7, 1985
    Assignee: Ciba Geigy Corporation
    Inventor: Henry Szczepanski
  • Patent number: 4515620
    Abstract: Triaza compounds of the general formula I ##STR1## and their basic addition salts have good selective herbicidal and plant growth regulating properties when applied pre- and postemergence. In the formula, each of A.sub.1 and A.sub.2 is a homocyclic or heterocyclic aromatic radical such as phenyl, naphthyl, indanyl, imidazolyl, pyridinyl, pyrimidinyl, pyrazolyl or triazolyl, each of which is unsubstituted or mono- to trisubstituted, while only one of A.sub.1 and A.sub.2 may be a phenyl, naphthyl or indanyl radical, and each of R.sub.1 and R.sub.3 is hydrogen or C.sub.1 -C.sub.4 alkyl and R.sub.2 is hydrogen or a cation.
    Type: Grant
    Filed: January 3, 1983
    Date of Patent: May 7, 1985
    Assignee: Ciba Geigy Corporation
    Inventor: Beat Bohner
  • Patent number: 4515624
    Abstract: Certain sulfonylurea compounds with oxysulfonyl-, thiosulfonyl- or aminosulfonyl-containing groups are useful as pre- and/or post-emergence herbicides.
    Type: Grant
    Filed: March 23, 1983
    Date of Patent: May 7, 1985
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: James J. Reap
  • Patent number: 4514212
    Abstract: N-Phenylsulfonyl-N'-triazinylureas of the general formula ##STR1## and the salts thereof with amines, alkali metal or alkaline earth metal bases or with quaternary ammonium bases, have good pre- and postemergence selective herbicidal and growth regulating properties. In the above formulaQ is fluorine, fluoromethyl, chloromethyl, trichloromethyl, 1,2-dichloroethyl, 1,2-dibromoethyl, 1,2-dichloropropyl, 1,2-dibromopropyl, 1,2-dibromoisobutyl, 1,2-dichloro-1-methyl-ethyl or 1,2-dibromo-1-methyl-ethyl,X is oxygen, sulfur, a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur,R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.5 alkyl, C.sub.2 -C.sub.5 alkenyl, C.sub.1 -C.sub.4 haloalkyl, or a radical --Y--R.sub.5, --COOR.sub.6, --NO.sub.2 or --CO--NR.sub.7 --R.sub.8,R.sub.3 and R.sub.4, each independently of the other, are hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 haloalkyl, halogen or alkoxyalkyl of at most 4 carbon atoms,R.sub.5 and R.sub.
    Type: Grant
    Filed: January 17, 1983
    Date of Patent: April 30, 1985
    Assignee: Ciba Geigy Corporation
    Inventors: Willy Meyer, Werner Fory
  • Patent number: 4514213
    Abstract: Novel benzenesulfonylurea compounds containing phenyl or phenoxy substituents such as 2-[[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]aminosulfonyl]-4-phenylbenz oic acid, methyl ester, and 2-[[(4-methoxy-6-methyl-1,3,5-triazin-2-yl)aminocarbonyl]aminosulfonyl]-4- phenylbenzoic acid, methyl ester, herbicidal compositions containing these compounds, and their method of use as general or selective pre-emergent or post-emergent herbicides.
    Type: Grant
    Filed: March 19, 1984
    Date of Patent: April 30, 1985
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: William T. Zimmerman
  • Patent number: 4510325
    Abstract: N-Phenylsulfonyl-N'-pyrimidinyl- and -triazinylureas of the general formula ##STR1## and the salts thereof with amines, alkali metal or alkaline earth metal bases or with quaternary ammonium bases, have good pre- and postemergence selective herbicidal and growth regulating properties. In the above formulaA is a C.sub.1 -C.sub.6 alkyl radical which is substituted by C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 alkylsulfinyl, C.sub.1 -C.sub.4 -alkylsulfonyl, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 haloalkylthio, C.sub.1 -C.sub.4 haloalkylsulfinyl or C.sub.1 -C.sub.4 haloalkylsulfonyl, or a C.sub.2 -C.sub.6 -alkenyl radical which is unsubstituted or substituted by the above substituents, or is a C.sub.2 -C.sub.6 haloalkenyl radical,E is the methine group or nitrogen,X is oxygen, sulfur, a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur,m is 1 or 2,R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.5 alkyl, C.sub.2 -C.sub.5 alkenyl or a radical --Y--R.sub.5,R.sub.
    Type: Grant
    Filed: September 13, 1982
    Date of Patent: April 9, 1985
    Assignee: Ciba-Geigy Corporation
    Inventors: Willy Meyer, Werner Fury
  • Patent number: 4508898
    Abstract: Compounds to general formula ##STR1## in which R and R' are hydrogen or benzyl and X represents a purine on pyrimidine base group selected from isoguanine, guanine, cytosine, 5-fluorouracil, S-methyl uracil (thymine) and chloroguanine, exhibit anti-viral properties.
    Type: Grant
    Filed: June 8, 1982
    Date of Patent: April 2, 1985
    Inventor: Kelvin K. Ogilvie
  • Patent number: 4501607
    Abstract: N-(heterocyclicaminocarbonyl)arylsulfonamides and thienylsulfonamides in which the heterocyclic radical is disubstituted; e.g., N-[[4-(2-methoxyethoxy)-6-methylpyrimidin-2-yl]aminocarbonyl]-2-nitrobenze nesulfonamide and N-[[(4-(2,2,2-trifluoroethoxy)-6-methylpyrimidin-2-yl]aminocarbonyl]-2-nit robenzenesulfonamide; are useful for the regulation of plant growth and as pre-emergence and post-emergence herbicides.
    Type: Grant
    Filed: January 30, 1980
    Date of Patent: February 26, 1985
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: George Levitt
  • Patent number: 4501744
    Abstract: Nucleoside analogues having a ring-open structure, of general formula: ##STR1## where R and R' may be hydrogen, silyl groups, substituted alkyl groups, benzyl groups and the like, and X is an optionally substituted pyrimidine or triazine base, exhibit anti-viral activities e.g. against herpes simplex virus and cytomegalo-virus at non-toxic levels.
    Type: Grant
    Filed: July 28, 1983
    Date of Patent: February 26, 1985
    Assignee: ens BIO LOGICALS Inc.
    Inventor: Kelvin K. Ogilvie
  • Patent number: 4500344
    Abstract: Ortho-(alkoxy)benzenesulfonamides, such as N-[(4-methoxy-6-methyl-1,3,5-triazin-2-yl)aminocarbonyl]-2-(2-hydroxyethox y)benzenesulfonamide, are useful as pre- and post-emergent herbicides.
    Type: Grant
    Filed: March 21, 1983
    Date of Patent: February 19, 1985
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: Robert W. Freerksen
  • Patent number: 4500342
    Abstract: Herbicidally active substituted phenylsulfonyl urea derivatives of the formula ##STR1## in which X is phenyl or phenoxy,R is ##STR2## and R.sup.1 and R.sup.2 each independently is methyl or methoxy.They are made from phenylisocyanates of the formula--SO.sub.2 --N.dbd.C.dbd.Owhich are produced by reacting a phenylsulfonamide of the formula ##STR3## with phosgene or with trichloromethyl chloroformate in the presence of an aliphatic isocyanate.
    Type: Grant
    Filed: January 20, 1982
    Date of Patent: February 19, 1985
    Assignee: Nihon Tokushu Noyaku Seizo K.K.
    Inventors: Masahiro Aya, Junichi Saito, Kazuomi Yasui, Kozo Shiokawa, Norihisa Morishima, Toshio Goto
  • Patent number: 4497951
    Abstract: Acetylene terminated s-triazine oligomers are disclosed which polymerize into stable high temperature resins. The oligomers of this invention are readily prepared from off-the-shelf starting materials, they are soluble in conventional low boiling solvents and exhibit low melting points which facilitate ease of processing.
    Type: Grant
    Filed: April 21, 1983
    Date of Patent: February 5, 1985
    Assignee: Hughes Aircraft Company
    Inventor: Thomas W. Giants
  • Patent number: 4496564
    Abstract: The invention relates to amide derivatives which are histamine H-2 antagonists and which inhibit gastric acid secretion. According to the invention there is provided a guanidine derivative of the formula I: ##STR1## in which R.sup.1 is a hydrogen or 1-10C alkyl, 3-8C cycloalkyl, 4-14C cycloalkylalkyl, 3-6C alkenyl, 3-6C alkynyl, 1-6C alkanoyl, 6-10C aryl, 7-11C aralkyl or 7-11C aroyl, the aryl, aralkyl and aroyl radical being optionally substituted; ring X is a heterocyclic ring as defined in the specification; A is phenylene or 5-7C cycloalkylene, or a 1-8C alkylene into which is optionally inserted one or two groups; D is O or S; and R.sup.2 and R.sup.3 are hydrogen or a variety of radicals described in the specification: and the pharmaceutically-acceptable acid-addition salts thereof. Manufacturing processes and pharmaceutical compositions are also described.
    Type: Grant
    Filed: March 1, 1982
    Date of Patent: January 29, 1985
    Assignees: ICI Americas Inc., Imperial Chemical Industries PLC
    Inventors: Tobias O. Yellin, David J. Gilman
  • Patent number: 4492599
    Abstract: This invention relates to novel urea and isourea compounds, agricultural compositions containing them and to their method of use as pre- and post- emergence herbicides and to plant growth regulants.
    Type: Grant
    Filed: September 27, 1982
    Date of Patent: January 8, 1985
    Assignee: E. I. Du Pont de Nemours and Company
    Inventors: George Levitt, Wallace C. Petersen
  • Patent number: 4492598
    Abstract: Compounds of the formula ##STR1## wherein R.sub.1 is (among others) (halo)cycloalkyl or (halo)cycloalkenyl, R.sub.2 and R.sub.3 are preferably hydrogen, X is preferably oxygen and R.sub.4 is substituted pyrimidyl or s-triazinyl, are valuable herbicides and growth regulators.
    Type: Grant
    Filed: August 6, 1982
    Date of Patent: January 8, 1985
    Assignee: Hoechst Aktiengesellschaft
    Inventors: Lothar Willms, Thomas Huttelmaier, Hilmar Mildenberger, Klaus Bauer, Helmut Burstell, Hermann Bieringer
  • Patent number: 4486589
    Abstract: N-(heterocyclicaminocarbonyl)-ortho-haloalkylbenzenesulfonamides, such as 2-(dichloromethyl)-N-[(4-methoxy-6-methylprimidin-2-yl) aminocarbonyl]-benzenesulfonamide, are useful as preemergent or postemergent herbicides or as plant growth regulants.
    Type: Grant
    Filed: October 21, 1982
    Date of Patent: December 4, 1984
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: William B. Farnham
  • Patent number: 4479948
    Abstract: Hypotensively active triazino-(2,1-a)isoquinoline compounds having the ring system ##STR1## and methods of making and using such compounds.
    Type: Grant
    Filed: July 8, 1982
    Date of Patent: October 30, 1984
    Assignee: Hoechst Aktiengesellschaft
    Inventors: Bansi Lal, Adolf D'Sa, Alihussein N. Dohadwalla, Noel J. de Souza, Horst Dornauer
  • Patent number: 4479821
    Abstract: N-Phenylsulfonyl-N'-triazinylureas of the general formula ##STR1## and the salts thereof with amines, alkali metal or alkaline earth metal bases or with quaternary ammonium bases, have good pre- and postemergence selective herbicidal and growth regulating properties. In the above formulaA is a C.sub.1 -C.sub.6 alkyl radical which is substituted by C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 alkylsulfinyl or C.sub.1 -C.sub.4 alkylsulfonyl,X is oxygen, sulfur, a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur,m is 1 or 2,R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.5 alkyl, C.sub.2 -C.sub.5 alkenyl, C.sub.1 -C.sub.4 haloalkyl, or a radical --Y--R.sub.5, --COOR.sub.6, --NO.sub.2 or --CO--NR.sub.7 --R.sub.8,R.sub.3 and R.sub.4, each independently of the other, are hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 haloalkyl, halogen or alkoxyalkyl or at most 4 carbon atoms,R.sub.5 and R.sub.6, each independently of the other, are C.
    Type: Grant
    Filed: January 17, 1983
    Date of Patent: October 30, 1984
    Assignee: Ciba-Geigy Corporation
    Inventors: Willy Meyer, Werner F/o/ ry
  • Patent number: 4477635
    Abstract: Polymeric and copolymeric aminotriarylmethane dyes having polyester, polyethyleneimine, or polyurethane backbones, and a process for their preparation, are disclosed. The novel dyes are highly colored and resistant to leaching by solvents.
    Type: Grant
    Filed: January 4, 1982
    Date of Patent: October 16, 1984
    Assignee: Minnesota Mining and Manufacturing Company
    Inventor: Smarajit Mitra
  • Patent number: 4474600
    Abstract: Substituted phenylsulfonylurea-derivatives of the general formula ##STR1## wherein X represents an oxygen atom or a direct bond, Y and Z each represents a halogen atom, a lower alkyl group, a lower alkoxy group or a nitro group, R represents a group: ##STR2## wherein R.sup.1 and R.sup.2 each represents a lower alkyl group or a lower alkoxy group, m and n each represents 0, 1 or 2 with the proviso that m and n do not represent 0 at the same time, are novel and find use as herbicides. Corresponding substituted benzenesulfonyl isocyanates are novel intermediate compounds for use in preparing compounds of formula (I).
    Type: Grant
    Filed: September 7, 1982
    Date of Patent: October 2, 1984
    Assignee: Nihon Tokushu Noyaku Seizo K.K.
    Inventors: Masahiro Aya, Junichi Saito, Kazuomi Yasui, Kozo Shiokawa, Norihisa Morishima, Toshio Goto
  • Patent number: 4473394
    Abstract: This invention relates to pyrrole sulfonamides which are useful as herbicides. Typical of the pyrrole sulfonamides of the instant application in N-[(4-methoxy-6-methyl-1,3,5-triazin-2-yl)aminocarbonyl]-2,5-dimethyl-1H-p yrrole-3-sulfonamide.
    Type: Grant
    Filed: September 27, 1982
    Date of Patent: September 25, 1984
    Assignee: E. I. DuPont De Nemours & Company
    Inventors: John C. Budzinski, George Levitt
  • Patent number: 4472168
    Abstract: Lithium salts of fiber reactive dyestuffs are stabilized in aqueous solution with N,N dialkylamine benzene sulfonic acid salt/acid buffers.
    Type: Grant
    Filed: July 5, 1983
    Date of Patent: September 18, 1984
    Assignee: ICI Americas Inc.
    Inventor: Donald R. Gauthier
  • Patent number: 4467088
    Abstract: s-Triazine compounds of the formula: ##STR1## in which R.sub.1 and R.sub.2 independently of one another are C.sub.1-4 alkyl, R.sub.3 and R.sub.4 independently of one another are one of the following radicals; C.sub.1-10 alkoxy which is unsubstituted or substituted by alkoxy; N-C.sub.1-10 alkylamino which is unsubstituted or substituted by phenyl; phenylamino which is unsubstituted or substituted by halogen, C.sub.1-4 alkyl or C.sub.1-4 alkoxy; naphthylamino which is unsubstituted or substituted by halogen, C.sub.1-4 alkyl or C.sub.1-4 alkoxy; halogen; N-phenyl-N-alkylamino; dialkylamino; alkylmercapto; cyclohexyloxy; N-alkyl-N-cyclohexylamino and cyclohexylamino; M is hydrogen or one equivalent of a cation and n is 1 or 2. These compounds may be used in the preparation of dyes.
    Type: Grant
    Filed: September 28, 1982
    Date of Patent: August 21, 1984
    Assignee: Ciba-Geigy Corporation
    Inventor: Hansrudolf Schwander
  • Patent number: 4465506
    Abstract: N-[Heterocyclicaminocarbonyl]-1H-indene and tetrahydronaphthalene sulfonamides, such as 2,3-dihydro-N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1H-indene-4-sul fonamide, are useful for the regulation of plant growth and as preemergent and postemergent herbicides.
    Type: Grant
    Filed: November 10, 1982
    Date of Patent: August 14, 1984
    Assignee: E. I. DuPont de Nemours and Company
    Inventor: John T. Welch
  • Patent number: 4461640
    Abstract: Alkenylsulfonylureas have been found to be effective as herbicides and plant growth regulants.
    Type: Grant
    Filed: June 2, 1982
    Date of Patent: July 24, 1984
    Assignee: E. I. Du Pont de Nemours and Company
    Inventors: George Levitt, William T. Zimmerman
  • Patent number: 4460585
    Type: Grant
    Filed: January 17, 1983
    Date of Patent: July 17, 1984
    Assignee: William H. Rorer, Inc.
    Inventors: Henry F. Campbell, Thomas H. Scholz, George H. Douglas
  • Patent number: 4460404
    Abstract: Condensed ring aromatic ureas and isoureas are useful as plant growth regulants and as pre- and/or post-emergence herbicides.
    Type: Grant
    Filed: September 22, 1982
    Date of Patent: July 17, 1984
    Assignee: E. I. DuPont de Nemours and Company
    Inventor: George Levitt
  • Patent number: 4455424
    Abstract: The present invention relates to naphthoquinone derivatives of formula I, ##STR1## in which R.sub.1 signifies a halogen atom, a nitro group or an unsubstituted or substituted alkoxy or amino group,R.sub.2 signifies the atoms necessary to form an unsaturated ring system, which ring system has 1 or 2 nuclei and is unsubstituted or substituted,R.sub.3 signifies an unsubstituted or substituted s-triazinyl or pyrimidyl radical, andn is 0, 1 or 2,which compounds are free from sulphonic acid groups are useful as pigments or disperse dyes.
    Type: Grant
    Filed: February 24, 1977
    Date of Patent: June 19, 1984
    Assignee: Sandoz Ltd.
    Inventor: Bansi L. Kaul
  • Patent number: 4453971
    Abstract: N-(heterocyclicaminocarbonyl)arylsulfonamides, such as 3-isocyanato-N-[(4-methoxy-6-methyl-1,3,5-triazin-2-yl)aminocarbonyl]benze nesulfonamide or methyl [3-[[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]aminosulfonyl]phenyl] carbamate, are useful for the regulation of plant growth and as herbicides.
    Type: Grant
    Filed: September 22, 1982
    Date of Patent: June 12, 1984
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: George Levitt
  • Patent number: 4452628
    Abstract: This invention pertains to benzenesulfonamides and their use as agricultural chemicals.
    Type: Grant
    Filed: May 30, 1980
    Date of Patent: June 5, 1984
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: John B. Adams, Jr.
  • Patent number: 4452980
    Abstract: Novel s-triazine compounds are prepared as derivatives of the corresponding amidinourea and amidinothiourea compounds by reacting with an activated form of an acid amide to give substituted s-triazinones and thiones respectively, of the formula ##STR1## The s-triazinones and thiones are useful derivatives in analyzing for the corresponding amidinourea or amidino thiourea precursors and also have useful pharmacological properties which make them suitable for a variety of medicinal purposes including use as antidiarrheal agents.
    Type: Grant
    Filed: July 1, 1982
    Date of Patent: June 5, 1984
    Assignee: William H. Rorer, Inc.
    Inventors: George H. Douglas, William L. Studt, Chong M. Won, Stuart A. Dodson, Jerome J. Zalipsky
  • Patent number: 4444583
    Abstract: N-Phenylsulfonyl-N'-triazinylureas of the general formula ##STR1## and the salts thereof with amines, alkali metal or alkaline earth metal bases or with quaternary ammonium bases, have good pre- and postemergence selective herbicidal and growth regulating properties. In the above formulaA is difluoromethyl or 1,1,2,2-tetrafluoroethyl,X is oxygen, sulfur, a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur andR.sub.3 and R.sub.4, each independently of the other, are hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 haloalkyl, halogen or alkoxyalkyl or at most 4 carbon atoms.
    Type: Grant
    Filed: January 17, 1983
    Date of Patent: April 24, 1984
    Assignee: Ciba-Geigy Corporation
    Inventors: Willy Meyer, Werner Fory
  • Patent number: 4443243
    Abstract: N-Phenylsulfonyl-N'-pyrimidinyl- and -triazinylureas of the general formula ##STR1## and the salts of these compounds with amines, with alkali or alkaline-earth metal bases or with quaternary ammonium bases, have good pre- and post-emergence selective, herbicidal and growth-regulating properties.The symbols in this formula are as follows:A is a C.sub.3 -C.sub.6 -alkynyl group,E is the methine group or nitrogen,X is oxygen, sulfur or a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur,m is the number one or two,R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl or C.sub.2 -C.sub.5 -alkenyl or a group --Y--R.sub.5,R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.1 -C.sub.4 -haloalkyl, or a group --Y--R.sub.5, --COOR.sub.6, --NO.sub.2 or --CO--NR.sub.7 --R.sub.8,R.sub.3 and R.sub.4 independently of one another are each hydrogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.
    Type: Grant
    Filed: July 9, 1982
    Date of Patent: April 17, 1984
    Assignee: Ciba-Geigy Corporation
    Inventors: Werner Fory, Karl Gass, Willy Meyer, Rolf Schurter
  • Patent number: 4443245
    Abstract: N-Phenylsulfonyl-N'-triazinyl-ureas of the formula ##STR1## and the salts thereof with amines, alkali metal or alkaline earth metal bases or with quaternary ammonium bases, have good pre- and postemergence selective herbicidal and growth regulating properties. In the above formulaA is a C.sub.2 -C.sub.6 -alkenyloxy, a C.sub.2 -C.sub.6 -haloalkenyloxy a C.sub.2 -C.sub.6 -haloalkenylthio, a C.sub.2 -C.sub.6 -haloalkenylsulfinyl or a C.sub.2 -C.sub.6 -haloalkenylsulfonyl radicalZ is oxygen or sulfur,m is 1 or 2,R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl, C.sub.1 -C.sub.4 -haloalkyl, or a radical --Y--R.sub.5, --COOR.sub.6, --NO.sub.2 or --CO--NR.sub.7 --R.sub.8,R.sub.3 and R.sub.4, each independently of the other, are hydrogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkyl, halogen or alkoxyalkyl of at most 4 carbon atoms,R.sub.5 and R.sub.6, each independently of the other, are C.sub.1 -C.sub.5 -alkyl, C.sub.
    Type: Grant
    Filed: January 17, 1983
    Date of Patent: April 17, 1984
    Assignee: Ciba-Geigy Corporation
    Inventors: Willy Meyer, Werner Fory
  • Patent number: 4435205
    Abstract: N-(Heterocycliccarbamoyl)arylsulfonamides, such as N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-hydroxybenzenesulfonamide , methanesulfonate are useful for plant growth retardation, brush control and weed control in crops.
    Type: Grant
    Filed: April 15, 1982
    Date of Patent: March 6, 1984
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: James J. Reap
  • Patent number: 4425153
    Abstract: This invention relates to ortho(acyloxy)benzenesulfonamides and their use as herbicides.
    Type: Grant
    Filed: January 18, 1982
    Date of Patent: January 10, 1984
    Assignee: E. I. Du Pont de Nemours & Co.
    Inventor: John B. Adams, Jr.
  • Patent number: 4420325
    Abstract: This invention relates to benzylsulfonylureas which are active pre- and post-emergence herbicides.
    Type: Grant
    Filed: April 22, 1982
    Date of Patent: December 13, 1983
    Assignee: E. I. Du Pont de Nemours & Company
    Inventor: Richard F. Sauers
  • Patent number: 4417917
    Abstract: Certain benzene-1,2-disulfonic acid derivatives are useful as agricultural chemicals, and in particular as herbicides.
    Type: Grant
    Filed: October 20, 1981
    Date of Patent: November 29, 1983
    Assignee: E. I. Du Pont de Nemours and Company
    Inventors: George Levitt, Richard F. Sauers
  • Patent number: 4412856
    Abstract: The novel compounds of the formula I are useful selective herbicides for postemergence application in crops of cereals, maize and rice.In formula I, ##STR1## A is an unsubstituted or substituted amino group, Q is a C.sub.2 -C.sub.6 alkylene bridge, Y is an oxygen or sulfur atom or an unsubstituted or substituted nitrogen atom, and Z is an unsubstituted or substituted phenyl, naphthyl or heterocyclic radical, which phenyl radical, containing the bridge member Y, can additionally carry one to four further substituents.
    Type: Grant
    Filed: May 22, 1981
    Date of Patent: November 1, 1983
    Assignee: Ciba-Geigy Corporation
    Inventors: Hans-Georg Brunner, Rolf Schurter, Henry Szczepanski
  • Patent number: 4406897
    Type: Grant
    Filed: July 6, 1981
    Date of Patent: September 27, 1983
    Assignee: William H. Rorer, Inc.
    Inventors: Henry F. Campbell, Thomas H. Scholz, George H. Douglas
  • Patent number: 4394506
    Abstract: N-(heterocyclicaminocarbonyl)arylsulfonamides in which the aryl radical is substituted in the 2-position by a carboxy radical, ester, thioester, or amide thereof; e.g. N-[(4,6-dimethylpyrimidin-2-yl)aminocarbonyl]-2-methoxycarbonylbenzenesulf onamide or N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-2-methoxycarbonylbenze nesulfonamide; are useful for the regulation of plant growth and as pre-emergence and post-emergence herbicides.
    Type: Grant
    Filed: November 30, 1979
    Date of Patent: July 19, 1983
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: George Levitt
  • Patent number: 4394153
    Abstract: The compounds are of the class of aryl esters of N-[(heterocyclic)aminocarbonyl]sulfamic acid, such as N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]sulfamic acid, (2-methylsulfonyloxy)-phenyl ester, useful for weed control in crops, brush control and plant growth retardation.
    Type: Grant
    Filed: May 18, 1981
    Date of Patent: July 19, 1983
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: James J. Reap
  • Patent number: 4391976
    Abstract: A process for producing an N-(heterocyclo-aminocarbonyl)-arylsulfamate of the general formula I ##STR1## wherein R.sub.1 is hydrogen, methoxy or C.sub.1 -C.sub.3 -alkyl,R.sub.2 is hydrogen, fluorine, chlorine, bromine, nitro, CF.sub.3, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.4 -alkoxycarbonyl,R.sub.3 is hydrogen, fluorine, chlorine, bromine, methyl or C.sub.1 -C.sub.4 -alkoxy,R.sub.4 is hydrogen, fluorine, chlorine, bromine, nitro, cyano, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.4 -alkoxycarbonyl,R.sub.5 is hydrogen, fluorine, chlorine, bromine, nitro or CF.sub.3,R.sub.6 is hydrogen, fluorine, chlorine, bromine, C.sub.1 -C.sub.4 -alkyl or C.sub.1 -C.sub.4 -alkoxy,X is C.sub.1 -C.sub.2 -alkyl, C.sub.1 -C.sub.3 -alkoxy, C.sub.1 -C.sub.2 -alkylthio, methoxymethyl, methoxyethyl, CF.sub.3 or chlorine,Y is C.sub.1 -C.sub.2 -alkyl, C.sub.1 -C.sub.3 -alkoxy, C.sub.1 -C.sub.
    Type: Grant
    Filed: October 19, 1981
    Date of Patent: July 5, 1983
    Assignee: Ciba-Geigy Corporation
    Inventor: Beat Bohner
  • Patent number: 4387225
    Abstract: Heterocyclic alkyl s-triazine compounds are prepared from the corresponding amidinourea and amidinothiourea compounds by reacting with an activated form of an acid amide to give respectively substituted s-triazinones and thiones of the formula ##STR1## which have pharmacological properties that render them suitable for use for a variety of medicinal purposes, including use as antidiarrheal agents, and which are also useful derivatives in analyzing for the corresponding amidinourea or amidinothiourea precursors.
    Type: Grant
    Filed: May 12, 1981
    Date of Patent: June 7, 1983
    Assignee: William H. Rorer, Inc.
    Inventors: George H. Douglas, William L. Studt, Chong M. Won, Stuart A. Dodson, Jerome J. Zalipsky
  • Patent number: 4383113
    Abstract: N-(heterocyclicaminocarbonyl)arylsulfonamides in which the aryl radical is substituted in the 2-position by a carboxy radical, ester, thioester, or amide thereof; e.g. N-[(4,6-dimethylpyrimidin-2-yl)aminocarbonyl]-2-methoxycarbonylbenzenesulf onamide or N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-2-methoxycarbonylbenze nesulfonamide; are useful for the regulation of plant growth and as pre-emergence and post-emergence herbicides.
    Type: Grant
    Filed: June 1, 1981
    Date of Patent: May 10, 1983
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: George Levitt
  • Patent number: 4382956
    Abstract: N-Sulphenylated biurets of the formula ##STR1## in which R.sup.1 represents a trihalogenomethyl radical,R.sup.2 represents an optionally substituted aliphatic, cycloaliphatic, araliphatic or aromatic radical andR.sup.3 and R.sup.4 are identical or different and represent a hydrogen atom, an optionally substituted aliphatic, cycloaliphatic, araliphatic, aromatic or heterocyclic radical or the amino or hydroxyl group, or together with the connecting nitrogen atom represent a five-membered or six-membered heterocyclic ring, the ring carbon atoms of which are optionally interrupted by one or more further hetero-atoms,which possess fungicidal activity.
    Type: Grant
    Filed: December 15, 1981
    Date of Patent: May 10, 1983
    Assignee: Bayer Aktiengesellschaft
    Inventors: Engelbert Kuhle, Volker Paul, Wilhelm Brandes