Abstract: Certain novel acyl saccharins and acyl 3-oxo-1,2-benzisothiazolines, their preparation, pharmaceutical compositions and novel methods of inhibiting elatase and treating emphysema are disclosed.
Type:
Grant
Filed:
August 20, 1975
Date of Patent:
March 25, 1980
Assignee:
Merck & Co., Inc.
Inventors:
Dennis Mulvey, Howard Jones, Morris Zimmerman