Patents Assigned to Amphaster Pharmaceuticals, Inc.
  • Patent number: 9303060
    Abstract: A method of preparing a thioic acid intermediate of fluticasone propionate includes: treating a 17?-[(N,N-dimethyl carbamoyl)thio]carbonyl compound in a solution including an alcohol and an alkali metal hydroxide, an alkaline-earth metal hydroxide, or a mixture thereof to cleave an amide from the 17?-[(N,N-dimethyl carbamoyl)thio]carbonyl compound; treating the solution to separate an aqueous portion; and adding an acid to the aqueous portion to obtain the thioic acid intermediate of fluticasone propionate. A method of preparing fluticasone propionate includes preparing the thioic acid intermediate of fluticasone propionate, and alkylating the thioic acid intermediate of fluticasone propionate to prepare the fluticasone propionate.
    Type: Grant
    Filed: April 16, 2015
    Date of Patent: April 5, 2016
    Assignee: Amphaster Pharmaceuticals, Inc.
    Inventors: Yinhua Qiu, Zhengyuan Wu, Yong Liu, Song Chen, Haoning Zhang