Abstract: Substituted 3-aminosydnone imines of the formula I ##STR1## and their pharmacologically acceptable acid addition salts, in which R.sup.1 denotes e.g. hydrogen;R.sup.2 denotes e.g. an alkyl radical;at least two of the radicals R.sup.3, R.sup.4, R.sup.5 and R.sup.6 denote alkyl radicals and the others denote hydrogen, are prepared by cyclization of a compound of the formula II ##STR2## and, if appropriate, subsequent acylation, and have useful pharmacological properties.
Type:
Grant
Filed:
June 7, 1990
Date of Patent:
January 12, 1993
Assignee:
Cassella Aktiengellschaft
Inventors:
Eckard Kujath, Christian Baumgartner, Karl Schonafinger, Rudi Beyerle, Melitta Just, Helmut Bohn, Jorg Ostrowski
Abstract: The 1,2,3,4-oxatriazolium-5-olates of the formula I ##STR1## in which R.sup.1 denotes, for example, (C.sub.2 to C.sub.4)alkyl,R.sup.2 and R.sup.3 denotes (C.sub.1 to C.sub.4)alkyl have useful pharmacological properties.
Type:
Grant
Filed:
April 6, 1990
Date of Patent:
February 25, 1992
Assignee:
Cassella Aktiengellschaft
Inventors:
Karl Schonafinger, Helmut Bohn, Rudi Beyerle, Melitta Just