Abstract: This invention provides a novel crystalline sitagliptin ethanedisulfonate salt having the structure set forth below, and a method for using same to treat type 2 diabetes.
Type:
Grant
Filed:
March 29, 2012
Date of Patent:
March 5, 2013
Assignee:
Corporacion Medichem, S.L.
Inventors:
Stephen Benedict David Winter, Monica Benito Velez, Ernesto Duran Lopez
Abstract: This invention provides improved methods for making solifenacin and pharmaceutically acceptable salts thereof. The instant methods are unexpectedly advantageous in their simplicity and efficiency.