Abstract: The invention provides cyclodextrin inclusion complex delivery vehicles, in which the cyclodextrin inclusion complex comprising acetaminophen and N-acetylcysteine is provided together with enzyme having a cyclodextrin-degrading activity capable of digesting the cyclodextrin, so that upon oral delivery of the vehicle to a target the enzyme is activated and releases acetaminophen and N-acetylcysteine from the cyclodextrin cavity. In alternative aspects, these cyclodextrin inclusion complex delivery vehicles are for example provided in the form of medicaments, food ingredients, medical food ingredients, nutritional supplement ingredients, dietary supplement ingredients, herbicides, insecticides, fungicides, animal repellents, pheromones, plant growth regulators, fragrances, fabrics or packaging materials.