Abstract: Disclosed are compounds of formula: that inhibiting GPBP activity, making them useful as therapeutics in antibody-mediated disorders, drug-resistant cancer, inflammation, protein misfolding and ER stress-mediated disorders, and aberrant apoptosis.
Type:
Application
Filed:
October 25, 2013
Publication date:
March 20, 2014
Applicant:
FIBROSTATIN, S.L.
Inventors:
Juan Saus, Santos Fustero, Juan F Sanz-Cervera, Enrique Pérez-Payá, Raül Blasco, Francisco Revert-Ros, Fernando Revert
Abstract: Disclosed are compounds of formula: that inhibiting GPBP activity, making them useful as therapeutics in antibody-mediated disorders, drug-resistant cancer, inflammation, protein misfolding and ER stress-mediated disorders, and aberrant apoptosis.
Type:
Grant
Filed:
November 5, 2010
Date of Patent:
November 19, 2013
Assignee:
FibroStatin, S.L.
Inventors:
Juan Saus, Santos Fustero, Juan F. Sanz-Cervera, Enrique Perez-Paya, Raul Blasco, Francisco Revert-Ros, Fernando Revert
Abstract: The present invention provides methods for the diagnosis and/or treatment of chronic kidney disease, immune complex-mediated GN, rheumatoid arthritis, and pulmonary fibrosis, and methods for identifying compounds for such therapeutic use.
Type:
Application
Filed:
February 21, 2012
Publication date:
August 23, 2012
Applicant:
Fibrostatin S.L.
Inventors:
Juan Saus, Fernando Revert, Ramón Merino, Jesús Merino, Francisco Revert-Ros
Abstract: Disclosed are compounds of formula: that inhibiting GPBP activity, making them useful as therapeutics in antibody-mediated disorders, drug-resistant cancer, inflammation, protein misfolding and ER stress-mediated disorders, and aberrant apoptosis.
Type:
Application
Filed:
November 5, 2010
Publication date:
May 5, 2011
Applicant:
FIBROSTATIN, S.L.
Inventors:
JUAN SAUS, SANTOS FUSTERO, JUAN F. SANZ-CERVERA, ENRIQUE PEREZ-PAYA, RAUL BLASCO, FRANCISCO REVERT-ROS, FERNANDO REVERT