Abstract: The present invention relates to a process for preparing 1-O-acyl-2-deoxy-2-fluoro-4-thio-?-D-arabinofuranoses having formula I and intermediates thereof: wherein R1 represents —C(O)—C1-C6-alkyl or —C(O)-aryl; and R2 represents C1-C6-alkyl, C1-C4-perfluoroalkyl or aryl.
Type:
Grant
Filed:
September 7, 2012
Date of Patent:
April 16, 2013
Assignee:
LIBRAMEDICINA, Inc.
Inventors:
David Voigtländer, Michael Sander, Michael Harre
Abstract: The present invention relates to a process for preparing 1-O-acyl-2-deoxy-2-fluoro-4-thio-?-D-arabinofuranoses having formula I and intermediates thereof: wherein R1 represents —C(O)—C1-C6-alkyl or —C(O)-aryl; and R2 represents C1-C6-alkyl, C1-C4-perfluoroalkyl or aryl.
Type:
Application
Filed:
September 7, 2012
Publication date:
January 3, 2013
Applicant:
LibraMedicina, Inc.
Inventors:
David VOIGTLÄNDER, Michael SANDER, Michael HARRE
Abstract: The present invention relates to a process for preparing 1-O-acyl-2-deoxy-2-fluoro-4-thio-?-D-arabinofuranoses having formula I and intermediates thereof: wherein R1 represents —C(O)—C1-C6-alkyl or —C(O)-aryl; and R2 represents C1-C6-alkyl, C1-C4-perfluoroalkyl or aryl.
Type:
Grant
Filed:
December 3, 2010
Date of Patent:
December 11, 2012
Assignee:
Libramedicina, Inc.
Inventors:
David Voigtländer, Michael Sander, Michael Harre