Abstract: Novel 4-dedimethylamino-4-arylsulfonamido-5a,6-anhydrotetracyclines of the general formula I ##STR1## wherein R stands for C.sub.1 -C.sub.3 -alkyl, halogen or --NHCOR.sup.1, R.sup.1 being C.sub.1 -C.sub.3 -alkyl.
Abstract: Corrosion inhibitors and preservatives of the following formula ##SPC1##WhereinR.sub.1 is hydrogen;R.sub.2 is selected from the group which consists of hydrogen, the diacetoxypropionic acid methyl ester and the diacetoxypropionic acid dialkylaminoethylamide with 1 to 4 carbon atoms in the alkyl group;R.sub.3 is hydrogen, unbranches or branched alkyl with 1 to 10 carbon atoms, carboxyl or alkoxycarbonyl wherein the alkoxy contains from 1 to 4 carbon atoms; andR.sub.4 is hydrogen, unbranched or branched alkyl with 1 to 4 carbon atoms; or acid addition or quaternary ammonium salts thereof.
Abstract: The new antibiotic compounds N-(4-R-benzenesulfonyl)-erythromycylamine, wherein R is a lower alkyl group having 1-5 carbon atoms, an acylamino group wherein the acyl has 2-4 carbon atoms, or a halo group.
Abstract: N-(4-R.sup.2 -benzenesulfonyl)-5-O-desosaminyl-erythromycilamine, wherein R.sup.2 is a C.sub.1 -C.sub.5 alkyl radical, halogen or NH.sub.2. The compounds possess antibacterial activity.
Type:
Grant
Filed:
January 10, 1975
Date of Patent:
February 17, 1976
Assignee:
Pliva, Pharmaceutical and Chemical Works