Abstract: A compound with anti-drug resistant bacteria activity having the following formula (I): is disclosed. R1 and R2 are each independently H, alkyl, or phenyl, or R1 and R2 form —(CH2)3—, —(CH2)4—, or —(CH2)5—, and R3 is —COOCH2CH3, or CN. A method of preparing the compound of formula (I) is also disclosed.