Patents Examined by Carolyn S. Greason
  • Patent number: 4690950
    Abstract: The present invention relates to new derivatives selected from the group consisting of:(i) 1-[N-(.alpha.-alkylamino-.alpha.-methylacetyl)aminophenyl]-2-alkylaminopro panones of the general formula: ##STR1## in which R represents a C.sub.1 -C.sub.4 alkyl group and R' represents H or a C.sub.1 -C.sub.4 alkyl group; and(ii) addition salts thereof.These new derivatives are useful as CNS-active substances, in particular as stimulants and antidepressants.The invention also relates to the method for their preparation.
    Type: Grant
    Filed: August 16, 1985
    Date of Patent: September 1, 1987
    Assignee: Laboratoire L. Lafon
    Inventor: Louis Lafon
  • Patent number: 4685962
    Abstract: A compound of the formula ##STR1## wherein Y represents a halogen atom, a lower alkyl group, a lower alkoxy group or a trifluoromethyl group and R represents a lower alkyl group. This compound can be produced by reacting a compound of the formula ##STR2## or a reactive derivative thereof with an aniline derivative of the formula ##STR3## and is useful as a herbicide.
    Type: Grant
    Filed: December 17, 1984
    Date of Patent: August 11, 1987
    Assignee: Yashima Chemical Industrial Co., Ltd.
    Inventors: Tetsuo Takematsu, Akinori Suzuki, Kazuya Toda, Masuo Goto
  • Patent number: 4684748
    Abstract: This invention provides certain benzamide derivatives, their pharmaceutical formulations, and their use as anticonvulsant agents.
    Type: Grant
    Filed: July 26, 1985
    Date of Patent: August 4, 1987
    Assignee: Eli Lilly and Company
    Inventor: David W. Robertson
  • Patent number: 4663481
    Abstract: Bromoacetamides of the formula ArCONHCH(Br)CONH.sub.2 are obtained by addition to bromine of a solution of ArCONHCH.sub.2 CN in a saturated aliphatic carboxylic acid preferably glacial acetic or propionic acid. This is an improvement in a process described in European Patent Specification No. 0059536 in which the bromine is added to a solution of the cyanomethylbenzamide, enabling consistently high yields (e.g. 75 to 90%) to be obtained.
    Type: Grant
    Filed: November 19, 1984
    Date of Patent: May 5, 1987
    Inventor: John D. Jones
  • Patent number: 4634558
    Abstract: .alpha.-Substituted acrylamides of the general formula I ##STR1## where R.sup.1 is a straight-chain, branched or cyclic alkyl radical of not more than 15 carbon atoms which can be unsubstituted or further substituted, are prepared by a process in which the corresponding .alpha.-substituted acrolein oximes are heated at from 40.degree. to 250.degree. C. in the presence of a copper(II) carboxylate and of an unsubstituted or substituted acrylonitrile as cocatalyst.
    Type: Grant
    Filed: November 30, 1984
    Date of Patent: January 6, 1987
    Assignee: BASF Aktiengesellschaft
    Inventors: Franz Merger, Wolfgang Schwarz
  • Patent number: 4632939
    Abstract: This invention provides certain benzamide derivatives of the formula: ##STR1## wherein Z is bond, --CH.sub.2 --, or CHCH.sub.3 ; A is --CH.sub.2 --, or CH.sub.2 CH.sub.2 --; and represents a single or double bond; and their pharmaceutical formulations and their use as anticonvulsant agents.
    Type: Grant
    Filed: March 15, 1985
    Date of Patent: December 30, 1986
    Assignee: Eli Lilly and Company
    Inventors: Edward E. Beedle, David W. Robertson
  • Patent number: 4632938
    Abstract: New insecticidal or/and ovicidal benzoylurea derivatives of the formula: ##STR1## wherein X.sup.1 is hydrogen or halogen; X.sup.2 is halogen; Y.sup.1, Y.sup.2 and Y.sup.3 are hydrogen, halogen or alkyl, whereby at least one of Y.sup.1, Y.sup.2 and Y.sup.3 is other than hydrogen; and R is hydrogen or a group represented by the formula --CF.sub.a Z.sub.b H.sub.(3-a-b) wherein a and b are 0, 1, 2 or 3, with a+b.ltoreq.3 and Z is halogen, their production and use.
    Type: Grant
    Filed: February 27, 1985
    Date of Patent: December 30, 1986
    Assignee: Takeda Chemical Industries, Ltd.
    Inventors: Hiroshi Nagase, Yasuo Sato
  • Patent number: 4633016
    Abstract: Compounds corresponding to the general formula ##STR1## wherein R.sup.3 represents H, CH.sub.3R.sup.4 represents H, C.sub.1-12 alkyl, C.sub.1-4 alkoxy, C.sub.1-12 alkylamino, C.sub.7-8 aralkylamino, arylamino, or C.sub.7-20 aralkyl,A represents a two-bonded group having the structure ##STR2## X may represent a single bond or --CO-- if it is attached to a carbon atom but only --CO-- if it is attached to a hetero atom,R.sup.1 represents R.sup.2, H or C.sub.1-4 alkyl,m represents 1 or 2 andn represents an integer from 1 to 12 are suitable as age resisters which can be built into polymers, in particular nitrile rubber.
    Type: Grant
    Filed: August 6, 1985
    Date of Patent: December 30, 1986
    Assignee: Bayer Aktiengesellschaft
    Inventors: Hans-Josef Buysch, Josef Witt, Zsolt Szentivanyi
  • Patent number: 4632983
    Abstract: Compounds of the general formula I ##STR1## where R is hydrogen or an aliphatic, alkenyl, cycloaliphatic, araliphatic, aromatic or heteroaromatic radical, R.sup.1 is hydrogen, amino, hydroxyl or C.sub.1 -C.sub.3 -alkyl, R.sup.2 is hydrogen, unsubstituted or substituted alkyl, allyl, aralkyl or aryl or alkylamino or arylamino, X is hydrogen, chlorine, bromine, nitro, methyl, phenoxy, tolyloxy, dimethylphenoxy, chlorophenoxy or C.sub.1 -C.sub.8 -alkoxy, Y is hydrogen, chlorine or bromine, and Z is hydrogen, acetyl, carbamyl or cyano, are useful for dyeing and/or printing textile material.
    Type: Grant
    Filed: December 5, 1983
    Date of Patent: December 30, 1986
    Assignee: BASF Aktiengesellschaft
    Inventor: Gunther Lamm
  • Patent number: 4623719
    Abstract: This invention relates to disazo dyestuffs for cellulose or cellulose-containing fibers represented by the formula: ##STR1## wherein R.sup.1 represents a hydrogen atom, a nitro group, a halogen atom, an alkyl group of 1 or 2 carbon atoms or an acetylamino group; R.sup.2 and R.sup.3 each represents a hydrogen atom, an alkyl group of 1 or 2 carbon atoms, and alkoxy group or an acetylamino group; Y.sup.1 and Y.sup.2 each represents a hydrogen atom or an alkyl group, and alkenyl group, a cyclohexyl group, an aryl group or an aralkyl group which group ma optionally be substituted by cyano, hydroxyl, lower alkoxy or dialkylamino, or NY.sup.1 Y.sup.2 represents a 5-membered or 6-membered nitrogen-containing heretocyclic ring formed by combination of Y.sup.1 and Y.sup.2, and the total carbon atoms in Y.sup.1 and Y.sup.2 is 18 or less.
    Type: Grant
    Filed: March 24, 1986
    Date of Patent: November 18, 1986
    Assignee: Mitsubishi Chemical Industries Limited
    Inventors: Toshio Niwa, Kiyoshi Himeno, Toshio Hihara
  • Patent number: 4623383
    Abstract: The present invention relates to novel N- and optionally N'-substituted (N-dichloroacetyl)glycine amides of the formula I with antidote action, to antidote compositions containing such compounds, to selective herbicide compositions containing these antidotes together with herbicidally active compounds and to a method for treating cultivated plants with said compositions.
    Type: Grant
    Filed: July 23, 1984
    Date of Patent: November 18, 1986
    Assignee: Eszakmagyarorszagi Vegyimuvek
    Inventors: Erzsebet Grega nee Toth, Jozsef Nagy, Gyula Tarpai, Erno Lorik, Istvan Toth, Karoly Pasztor, Zsuzsanna Bartfai nee Harsanyi, Ilona Beres, Laszlo Tasi, Eszter Urszin nee Simon, Zsolt Dombay, Judit Bajusz nee Olah, Karoly Balogh
  • Patent number: 4622426
    Abstract: N,N'-bis(2-hydroxyethyl)oxamide is facilely prepared, e.g., in finely divided crystalline form, by reacting an alkyl oxalate with ethanolamine in an aqueous reaction medium.
    Type: Grant
    Filed: November 9, 1984
    Date of Patent: November 11, 1986
    Assignee: Rhone-Poulenc Specialites Chimiques
    Inventor: Michel Crochemore
  • Patent number: 4613695
    Abstract: The invention concerns N-nitroso compounds having the general formula: ##STR1## wherein A is lower alkyl or halolower alkyl;B is hydrogen; lower alkenyl; lower alkynyl; 3-6 C cycloalkyl; --RSO.sub.2 NR.sup.3 R.sup.4, or lower alkyl optionally monosubstituted with lower alkoxy, or 3-6 C cycloalkyl;R is straight or branched 2-5 C alkylene, optionally monosubstituted with SO.sub.2 NR.sup.3 R.sup.4 or CONR.sup.3 R.sup.4, said alkylene always containing at least two carbon atoms separating the nitrogen atom of the urea from any SO.sub.2 NR.sup.1 R.sup.2 or SO.sub.2 NR.sup.3 R.sup.4 ;R.sup.1 and R.sup.2 are the same or different and selected from hydrogen, 5-6 C cycloalkyl, lower alkoxy, phenyl, benzyl, and straight or branched 1-6 C alkyl, optionally monosubstituted with hydroxy, lower alkoxy, SO.sub.2 NR.sup.3 R.sup.4, or CONR.sup.3 R.sup.4 ; R.sup.1 and R.sup.2 may also together form a 4-5 C alkylene; and R.sup.3 and R.sup.4 are the same or different and selected from hydrogen or lower alkyl, or R.sup.3 and R.
    Type: Grant
    Filed: September 6, 1983
    Date of Patent: September 23, 1986
    Assignee: Aktiebolaget Leo
    Inventors: Jan-Inge L. Carlsson, Herta G. Jensen Petersen, Anders R. Stamvik
  • Patent number: 4603195
    Abstract: A composition obtained by interracting a quinone diazo compound and an organosilicon compound; and use thereof in lithography.
    Type: Grant
    Filed: December 30, 1983
    Date of Patent: July 29, 1986
    Assignee: International Business Machines Corporation
    Inventors: Edward D. Babich, Michael Hatzakis, Jurij R. Paraszczak, Jane M. Shaw
  • Patent number: 4600796
    Abstract: A process for preparing a class of polyols resulting from the reaction of a bicyclic amide acetal with an alkanolamine is described.
    Type: Grant
    Filed: June 3, 1985
    Date of Patent: July 15, 1986
    Assignee: Ashland Oil, Inc.
    Inventor: Anil B. Goel
  • Patent number: 4597907
    Abstract: .alpha.-substituted acrylamides of the general formula I ##STR1## where R.sup.1 is a straight-chain, branched or cyclic alkyl radical of not more than 15 carbon atoms which can be unsubstituted or further substituted, are prepared by a process in which the corresponding .alpha.-substituted acrolein oximes are heated at from 40.degree. to 250.degree. C. in the presence of a copper(II) carboxylate.
    Type: Grant
    Filed: December 3, 1984
    Date of Patent: July 1, 1986
    Assignee: BASF Aktiengesellschaft
    Inventors: Franz Merger, Wolfgang Schwarz
  • Patent number: 4595779
    Abstract: The present invention provides a nonpyrophoric and thermally stable form of lithium diisopropylamide which is useful as a reagent in the preparation of pharmaceuticals and specialty chemicals. The preferred composition includes lithium diisopropylamide, a limited amount of tetrahydrofuran in an amount not exceeding one mole per mole of lithium diisopropylamide, and at least one C.sub.2 to C.sub.18 amine.
    Type: Grant
    Filed: December 24, 1984
    Date of Patent: June 17, 1986
    Assignee: Lithium Corporation of America, Inc.
    Inventors: Robert C. Morrison, Randy W. Hall, Terry L. Rathman
  • Patent number: 4593123
    Abstract: Process for the production of acrylamide or methacrylamide wherein acrylonitrile or methacrylonitrile is reacted with water and/or a water donor in the presence of Raney copper catalyst, which is protected from contact with oxygen.
    Type: Grant
    Filed: November 28, 1984
    Date of Patent: June 3, 1986
    Assignee: Mitsui Toatsu Chemicals, Incorporated
    Inventor: Fujio Matsuda
  • Patent number: 4579938
    Abstract: Thiophen-2-ylazopyrazole dyes useful for dyeing polyesters, cellulose acetate esters, and polyamides in fast yellow shades have the general formula ##STR1## wherein: X is a substituent such as alkyl, allyloxy, alkoxy, aryl, aryloxy, amino, alkylamino, arylamino, cyclohexyloxy, thienyl, cycloalkylamino, or the like; Y is hydrogen, alkyl, or aryl; Z is alkyl, aryl, alkylsulfonyl, 2-benzothiazolyl, cyano or COX; R and R.sub.1 are alkyl or aryl; R.sub.2 is hydrogen, or a substituent such as alkyl, aryl, acyl, benzothiazolyl, pyridyl, sulfolanyl, thiocarbamyl, carbamyl, alkoxycarbonyl, aroyl, or the like; wherein the hydrocarbon moieties of the above radicals may be substituted with up to three of --OH, alkoxy, hydroxyalkoxy, carbamyl, or the like; and wherein the dye molecule contains at least one SO.sub.3 M, OSO.sub.3 M, or SSO.sub.3 M water-solubilizing group.
    Type: Grant
    Filed: April 9, 1984
    Date of Patent: April 1, 1986
    Assignee: Eastman Kodak Company
    Inventor: Max A. Weaver
  • Patent number: 4564638
    Abstract: Fungicidally active novel benzylurea derivatives of the formula ##STR1## in which R.sup.1 is a halogen atom or a lower alkyl group,X is an oxygen or sulfur atom, andR.sup.2 is an alkyl group, a cycloalkyl group having 5 to 8 carbon atoms, or a phenyl group which may be substituted by at least one member of the class consisting of halogen atoms, lower alkyl groups, lower alkoxy groups and hydroxyl groups.
    Type: Grant
    Filed: June 10, 1983
    Date of Patent: January 14, 1986
    Assignee: Nihon Tokushu Boyaku Seizo K.K.
    Inventors: Yasuo Yamada, Junichi Saito, Tatsuo Tamura, Shinji Sakawa