Patents Examined by Carolyn S. Greason
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Patent number: 4690950Abstract: The present invention relates to new derivatives selected from the group consisting of:(i) 1-[N-(.alpha.-alkylamino-.alpha.-methylacetyl)aminophenyl]-2-alkylaminopro panones of the general formula: ##STR1## in which R represents a C.sub.1 -C.sub.4 alkyl group and R' represents H or a C.sub.1 -C.sub.4 alkyl group; and(ii) addition salts thereof.These new derivatives are useful as CNS-active substances, in particular as stimulants and antidepressants.The invention also relates to the method for their preparation.Type: GrantFiled: August 16, 1985Date of Patent: September 1, 1987Assignee: Laboratoire L. LafonInventor: Louis Lafon
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Patent number: 4685962Abstract: A compound of the formula ##STR1## wherein Y represents a halogen atom, a lower alkyl group, a lower alkoxy group or a trifluoromethyl group and R represents a lower alkyl group. This compound can be produced by reacting a compound of the formula ##STR2## or a reactive derivative thereof with an aniline derivative of the formula ##STR3## and is useful as a herbicide.Type: GrantFiled: December 17, 1984Date of Patent: August 11, 1987Assignee: Yashima Chemical Industrial Co., Ltd.Inventors: Tetsuo Takematsu, Akinori Suzuki, Kazuya Toda, Masuo Goto
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Patent number: 4684748Abstract: This invention provides certain benzamide derivatives, their pharmaceutical formulations, and their use as anticonvulsant agents.Type: GrantFiled: July 26, 1985Date of Patent: August 4, 1987Assignee: Eli Lilly and CompanyInventor: David W. Robertson
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Patent number: 4663481Abstract: Bromoacetamides of the formula ArCONHCH(Br)CONH.sub.2 are obtained by addition to bromine of a solution of ArCONHCH.sub.2 CN in a saturated aliphatic carboxylic acid preferably glacial acetic or propionic acid. This is an improvement in a process described in European Patent Specification No. 0059536 in which the bromine is added to a solution of the cyanomethylbenzamide, enabling consistently high yields (e.g. 75 to 90%) to be obtained.Type: GrantFiled: November 19, 1984Date of Patent: May 5, 1987Inventor: John D. Jones
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Patent number: 4634558Abstract: .alpha.-Substituted acrylamides of the general formula I ##STR1## where R.sup.1 is a straight-chain, branched or cyclic alkyl radical of not more than 15 carbon atoms which can be unsubstituted or further substituted, are prepared by a process in which the corresponding .alpha.-substituted acrolein oximes are heated at from 40.degree. to 250.degree. C. in the presence of a copper(II) carboxylate and of an unsubstituted or substituted acrylonitrile as cocatalyst.Type: GrantFiled: November 30, 1984Date of Patent: January 6, 1987Assignee: BASF AktiengesellschaftInventors: Franz Merger, Wolfgang Schwarz
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Patent number: 4632939Abstract: This invention provides certain benzamide derivatives of the formula: ##STR1## wherein Z is bond, --CH.sub.2 --, or CHCH.sub.3 ; A is --CH.sub.2 --, or CH.sub.2 CH.sub.2 --; and represents a single or double bond; and their pharmaceutical formulations and their use as anticonvulsant agents.Type: GrantFiled: March 15, 1985Date of Patent: December 30, 1986Assignee: Eli Lilly and CompanyInventors: Edward E. Beedle, David W. Robertson
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Patent number: 4632938Abstract: New insecticidal or/and ovicidal benzoylurea derivatives of the formula: ##STR1## wherein X.sup.1 is hydrogen or halogen; X.sup.2 is halogen; Y.sup.1, Y.sup.2 and Y.sup.3 are hydrogen, halogen or alkyl, whereby at least one of Y.sup.1, Y.sup.2 and Y.sup.3 is other than hydrogen; and R is hydrogen or a group represented by the formula --CF.sub.a Z.sub.b H.sub.(3-a-b) wherein a and b are 0, 1, 2 or 3, with a+b.ltoreq.3 and Z is halogen, their production and use.Type: GrantFiled: February 27, 1985Date of Patent: December 30, 1986Assignee: Takeda Chemical Industries, Ltd.Inventors: Hiroshi Nagase, Yasuo Sato
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Patent number: 4633016Abstract: Compounds corresponding to the general formula ##STR1## wherein R.sup.3 represents H, CH.sub.3R.sup.4 represents H, C.sub.1-12 alkyl, C.sub.1-4 alkoxy, C.sub.1-12 alkylamino, C.sub.7-8 aralkylamino, arylamino, or C.sub.7-20 aralkyl,A represents a two-bonded group having the structure ##STR2## X may represent a single bond or --CO-- if it is attached to a carbon atom but only --CO-- if it is attached to a hetero atom,R.sup.1 represents R.sup.2, H or C.sub.1-4 alkyl,m represents 1 or 2 andn represents an integer from 1 to 12 are suitable as age resisters which can be built into polymers, in particular nitrile rubber.Type: GrantFiled: August 6, 1985Date of Patent: December 30, 1986Assignee: Bayer AktiengesellschaftInventors: Hans-Josef Buysch, Josef Witt, Zsolt Szentivanyi
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Patent number: 4632983Abstract: Compounds of the general formula I ##STR1## where R is hydrogen or an aliphatic, alkenyl, cycloaliphatic, araliphatic, aromatic or heteroaromatic radical, R.sup.1 is hydrogen, amino, hydroxyl or C.sub.1 -C.sub.3 -alkyl, R.sup.2 is hydrogen, unsubstituted or substituted alkyl, allyl, aralkyl or aryl or alkylamino or arylamino, X is hydrogen, chlorine, bromine, nitro, methyl, phenoxy, tolyloxy, dimethylphenoxy, chlorophenoxy or C.sub.1 -C.sub.8 -alkoxy, Y is hydrogen, chlorine or bromine, and Z is hydrogen, acetyl, carbamyl or cyano, are useful for dyeing and/or printing textile material.Type: GrantFiled: December 5, 1983Date of Patent: December 30, 1986Assignee: BASF AktiengesellschaftInventor: Gunther Lamm
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Patent number: 4623719Abstract: This invention relates to disazo dyestuffs for cellulose or cellulose-containing fibers represented by the formula: ##STR1## wherein R.sup.1 represents a hydrogen atom, a nitro group, a halogen atom, an alkyl group of 1 or 2 carbon atoms or an acetylamino group; R.sup.2 and R.sup.3 each represents a hydrogen atom, an alkyl group of 1 or 2 carbon atoms, and alkoxy group or an acetylamino group; Y.sup.1 and Y.sup.2 each represents a hydrogen atom or an alkyl group, and alkenyl group, a cyclohexyl group, an aryl group or an aralkyl group which group ma optionally be substituted by cyano, hydroxyl, lower alkoxy or dialkylamino, or NY.sup.1 Y.sup.2 represents a 5-membered or 6-membered nitrogen-containing heretocyclic ring formed by combination of Y.sup.1 and Y.sup.2, and the total carbon atoms in Y.sup.1 and Y.sup.2 is 18 or less.Type: GrantFiled: March 24, 1986Date of Patent: November 18, 1986Assignee: Mitsubishi Chemical Industries LimitedInventors: Toshio Niwa, Kiyoshi Himeno, Toshio Hihara
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Patent number: 4623383Abstract: The present invention relates to novel N- and optionally N'-substituted (N-dichloroacetyl)glycine amides of the formula I with antidote action, to antidote compositions containing such compounds, to selective herbicide compositions containing these antidotes together with herbicidally active compounds and to a method for treating cultivated plants with said compositions.Type: GrantFiled: July 23, 1984Date of Patent: November 18, 1986Assignee: Eszakmagyarorszagi VegyimuvekInventors: Erzsebet Grega nee Toth, Jozsef Nagy, Gyula Tarpai, Erno Lorik, Istvan Toth, Karoly Pasztor, Zsuzsanna Bartfai nee Harsanyi, Ilona Beres, Laszlo Tasi, Eszter Urszin nee Simon, Zsolt Dombay, Judit Bajusz nee Olah, Karoly Balogh
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Patent number: 4622426Abstract: N,N'-bis(2-hydroxyethyl)oxamide is facilely prepared, e.g., in finely divided crystalline form, by reacting an alkyl oxalate with ethanolamine in an aqueous reaction medium.Type: GrantFiled: November 9, 1984Date of Patent: November 11, 1986Assignee: Rhone-Poulenc Specialites ChimiquesInventor: Michel Crochemore
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Patent number: 4613695Abstract: The invention concerns N-nitroso compounds having the general formula: ##STR1## wherein A is lower alkyl or halolower alkyl;B is hydrogen; lower alkenyl; lower alkynyl; 3-6 C cycloalkyl; --RSO.sub.2 NR.sup.3 R.sup.4, or lower alkyl optionally monosubstituted with lower alkoxy, or 3-6 C cycloalkyl;R is straight or branched 2-5 C alkylene, optionally monosubstituted with SO.sub.2 NR.sup.3 R.sup.4 or CONR.sup.3 R.sup.4, said alkylene always containing at least two carbon atoms separating the nitrogen atom of the urea from any SO.sub.2 NR.sup.1 R.sup.2 or SO.sub.2 NR.sup.3 R.sup.4 ;R.sup.1 and R.sup.2 are the same or different and selected from hydrogen, 5-6 C cycloalkyl, lower alkoxy, phenyl, benzyl, and straight or branched 1-6 C alkyl, optionally monosubstituted with hydroxy, lower alkoxy, SO.sub.2 NR.sup.3 R.sup.4, or CONR.sup.3 R.sup.4 ; R.sup.1 and R.sup.2 may also together form a 4-5 C alkylene; and R.sup.3 and R.sup.4 are the same or different and selected from hydrogen or lower alkyl, or R.sup.3 and R.Type: GrantFiled: September 6, 1983Date of Patent: September 23, 1986Assignee: Aktiebolaget LeoInventors: Jan-Inge L. Carlsson, Herta G. Jensen Petersen, Anders R. Stamvik
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Patent number: 4603195Abstract: A composition obtained by interracting a quinone diazo compound and an organosilicon compound; and use thereof in lithography.Type: GrantFiled: December 30, 1983Date of Patent: July 29, 1986Assignee: International Business Machines CorporationInventors: Edward D. Babich, Michael Hatzakis, Jurij R. Paraszczak, Jane M. Shaw
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Patent number: 4600796Abstract: A process for preparing a class of polyols resulting from the reaction of a bicyclic amide acetal with an alkanolamine is described.Type: GrantFiled: June 3, 1985Date of Patent: July 15, 1986Assignee: Ashland Oil, Inc.Inventor: Anil B. Goel
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Patent number: 4597907Abstract: .alpha.-substituted acrylamides of the general formula I ##STR1## where R.sup.1 is a straight-chain, branched or cyclic alkyl radical of not more than 15 carbon atoms which can be unsubstituted or further substituted, are prepared by a process in which the corresponding .alpha.-substituted acrolein oximes are heated at from 40.degree. to 250.degree. C. in the presence of a copper(II) carboxylate.Type: GrantFiled: December 3, 1984Date of Patent: July 1, 1986Assignee: BASF AktiengesellschaftInventors: Franz Merger, Wolfgang Schwarz
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Patent number: 4595779Abstract: The present invention provides a nonpyrophoric and thermally stable form of lithium diisopropylamide which is useful as a reagent in the preparation of pharmaceuticals and specialty chemicals. The preferred composition includes lithium diisopropylamide, a limited amount of tetrahydrofuran in an amount not exceeding one mole per mole of lithium diisopropylamide, and at least one C.sub.2 to C.sub.18 amine.Type: GrantFiled: December 24, 1984Date of Patent: June 17, 1986Assignee: Lithium Corporation of America, Inc.Inventors: Robert C. Morrison, Randy W. Hall, Terry L. Rathman
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Patent number: 4593123Abstract: Process for the production of acrylamide or methacrylamide wherein acrylonitrile or methacrylonitrile is reacted with water and/or a water donor in the presence of Raney copper catalyst, which is protected from contact with oxygen.Type: GrantFiled: November 28, 1984Date of Patent: June 3, 1986Assignee: Mitsui Toatsu Chemicals, IncorporatedInventor: Fujio Matsuda
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Patent number: 4579938Abstract: Thiophen-2-ylazopyrazole dyes useful for dyeing polyesters, cellulose acetate esters, and polyamides in fast yellow shades have the general formula ##STR1## wherein: X is a substituent such as alkyl, allyloxy, alkoxy, aryl, aryloxy, amino, alkylamino, arylamino, cyclohexyloxy, thienyl, cycloalkylamino, or the like; Y is hydrogen, alkyl, or aryl; Z is alkyl, aryl, alkylsulfonyl, 2-benzothiazolyl, cyano or COX; R and R.sub.1 are alkyl or aryl; R.sub.2 is hydrogen, or a substituent such as alkyl, aryl, acyl, benzothiazolyl, pyridyl, sulfolanyl, thiocarbamyl, carbamyl, alkoxycarbonyl, aroyl, or the like; wherein the hydrocarbon moieties of the above radicals may be substituted with up to three of --OH, alkoxy, hydroxyalkoxy, carbamyl, or the like; and wherein the dye molecule contains at least one SO.sub.3 M, OSO.sub.3 M, or SSO.sub.3 M water-solubilizing group.Type: GrantFiled: April 9, 1984Date of Patent: April 1, 1986Assignee: Eastman Kodak CompanyInventor: Max A. Weaver
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Patent number: 4564638Abstract: Fungicidally active novel benzylurea derivatives of the formula ##STR1## in which R.sup.1 is a halogen atom or a lower alkyl group,X is an oxygen or sulfur atom, andR.sup.2 is an alkyl group, a cycloalkyl group having 5 to 8 carbon atoms, or a phenyl group which may be substituted by at least one member of the class consisting of halogen atoms, lower alkyl groups, lower alkoxy groups and hydroxyl groups.Type: GrantFiled: June 10, 1983Date of Patent: January 14, 1986Assignee: Nihon Tokushu Boyaku Seizo K.K.Inventors: Yasuo Yamada, Junichi Saito, Tatsuo Tamura, Shinji Sakawa