Abstract: A composition of matter is described herein which has herbicidal activity and methods of use. The composition is defined by the following generic formula ##STR1## wherein X and Y are independently selected from the group consisting of chloro, bromo, and trifluoromethyl; n is either 0 or 1; m is either 0 or 1; and R and R.sub.1 are independently selected from the group consisting of lower alkyl from C.sub.1 to C.sub.3, inclusive, and lower alkoxy from C.sub.1 to C.sub.3, inclusive, or R and R.sub.
Abstract: A heart and vasotropic pharmaceutical of the formula: ##STR1## wherein R represents a hydrogen atom or an acyl group, preferably a C.sub.1-15 alkylcarbonyl, C.sub.2-6 alkenylcarbonyl, or a phenyl- (C.sub.1-5)-alkylcarbonyl group or a benzoyl group optionally substituted with halogen, trihalomethyl, C.sub.1-4 or nitroAnd pharmaceutically acceptable acid addition and quaternary salts thereof.
Type:
Grant
Filed:
June 9, 1976
Date of Patent:
December 27, 1977
Assignee:
Richter Gedeon Vegyeszeti Gyar Rt.
Inventors:
Csaba Lorincz, Kalman Szasz, Maria Bolyos, Karola Jovanovics, Laszlo Szporny, Egon Karpati, Eva Palosi
Abstract: Compounds of the formula ##STR1## IN WHICH R is aminocarbonylphenyl in which amino is --NH.sub.2, pyrrolidino, piperidino or morpholino, and Ar is phenyl substituted with chloro, fluoro, trifluoromethyl, methylenedioxy or one or more methoxy. The compounds are prepared by reacting 2-Ar-4-chloropyrimidin-6-yl ethylacetate with ##STR2## and then reacting that reaction product with hydroxylamine hydrochloride. The compounds possess vasodilatatory, anti-ulcerous, respiratory analeptic, hypotensive, diuretic, anti-depressive, analgesic, anti-inflammatory and neurotropic properties.
Type:
Grant
Filed:
December 10, 1976
Date of Patent:
December 6, 1977
Assignee:
Delalande S.A.
Inventors:
Claude P. Fauran, Jeannine A. Eberle, Guy R. Bourgery, Guy R. Raynaud, Claude J. Gouret