Patent number: 6806264
Abstract: The present invention relates to novel arylphenyl-substituted cyclic ketoenols of the formula (I)
in which
X represents halogen, alkyl, alkoxy, alkenyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro, cyano or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio,
Y represents in each case optionally substituted cycloalkyl, aryl or hetaryl,
W and Y independently of one another each represent hydrogen, halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano,
CKE represents one of the groups
in which
A, B, D, G and Q1 to Q6 are each as defined in the description,
to a plurality of processes for their preparation and to their use as pesticides and herbicides.
Type:
Grant
Filed:
December 8, 2003
Date of Patent:
October 19, 2004
Assignee:
Bayer Aktiengesellschaft
Inventors:
Folker Lieb, Reiner Fischer, Alan Graff, Udo Schneider, Thomas Bretshneider, Christoph Erdelen, Wolfram Andersch, Mark Wilhelm Drewes, Markus Dollinger, Ingo Wetcholowsky, Randy Allen Myers
Patent number: 6797707
Abstract: Disclosed are compounds having the formula:
where
R1=H, C1-C6 alkyl, cycloalkyl,
R2=H, C1-C6 alkyl, cycloalkyl
W=CnH2n-m—NH (n=1-6, m=0, 2, or 4),
Z=CONR8(CH2)n, CONR8(CH2)nCO, P(CH3)OCHR8OCOR9, SO2, SO2(CH2)n, SO2(CH2)nCO, SO2NR8(CH2)n, SO2NR8(CH2)nCO, n=1-4
R4=H, (CH2)nOH, (CH2)nOCOR10, (CH2)nNR10R11, (CH2)nCONR10R11, n=0-4
R5=H, (CH2)nNR12R13, n=0-4
R6=H, (CH2)nNR14R15, n=0-4
R7=H, C1-C6 alkyl, cycloalkyl; R8=H, C1-C6 alkyl, cycloalkyl; R9=H, C1-C6 alkyl, cycloalkyl;
R10=H, C1-C6 alkyl, cycloalkyl; R11=H, C1-C6 alkyl, cycloalkyl; R12=H, C1-C6 alkyl, cycloalkyl;
R13=H, C1-C6 alkyl, cycloalkyl; R14=H, C1-C6 alkyl, cycloalkyl; R15=H, C1-C6 alkyl, cycloalkyl
Dashed lines: optional; conformational constraint by (CH2)n, n=1-3, R′=H or O(═)
as well as pharmaceuticals c
Type:
Grant
Filed:
March 29, 2002
Date of Patent:
September 28, 2004
Assignee:
University of Florida
Inventor:
Laszlo Prokai
Patent number: 6797706
Abstract: A nitrogen-containing six-membered heterocyclic compound having substituents —X—A—R3, —N(R1)-(Ph substituted by R2), and —CONH2, a salt thereof, a prodrug thereof, and a Syk inhibitor containing the same as an active ingredient. (In the formula, A: a (substituted) lower alkylene, a (substituted) arylene, or the like; X: NR4, CONR4, NR4CO, O, or S; R1, R4: H, a lower alkyl, —CO-lower alkyl, or —SO2-lower alkyl; R2: H, a (substituted) lower alkyl, —O-lower alkyl, —S-lower alkyl, —O-aryl, nitro, cyano, or the like; R3: —CO2H, —CO2-lower alkyl, -lower alkylene-CO2H, —NH2, -alkylene-NH2 or the like.
Type:
Grant
Filed:
December 10, 2001
Date of Patent:
September 28, 2004
Assignee:
Yamanouchi Pharmaceutical Co., Ltd.
Inventors:
Hiroyuki Hisamichi, Souichirou Kawazoe, Kazuhito Tanabe, Atsushi Ichikawa, Akiko Orita, Takayuki Suzuki, Kenichi Onda, Makoto Takeuchi