Patents by Inventor Alain P. Lacour

Alain P. Lacour has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4831051
    Abstract: New aromatic derivatives having an activity antagonistic to calcium and corresponding to formula: ##STR1## in which: A represents a chain having any one of the following structures: ##STR2## Ar represents a group of structure: ##STR3## n takes the value 1 or 2 when R is different from H; m takes the value 2 or 3.
    Type: Grant
    Filed: January 22, 1988
    Date of Patent: May 16, 1989
    Assignee: Delande S.A.
    Inventors: Guy R. Bourgery, Alain P. Lacour, Bernard M. Pourrias, Raphael Santamaria
  • Patent number: 4732896
    Abstract: New aromatic derivatives having an activity antagonistic to calcium and corresponding to formula: ##STR1## in which: A represents a chain having any one of the following structures: ##STR2## Ar represents a group of structure: ##STR3## n takes the value 1 or 2 when R is different from H; m takes the value 2 or 3.
    Type: Grant
    Filed: June 26, 1985
    Date of Patent: March 22, 1988
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Alain P. Lacour, Bernard M. Pourrias, Raphael Santamaria
  • Patent number: 4536500
    Abstract: New aromatic derivatives having an activity antagonistic to calcium and corresponding to formula: ##STR1## in which: A represents a chain having any one of the following structures: ##STR2## Ar represents a group of structure: ##STR3## n takes the value 1 or 2 when R is different from H; m takes the value 2 or 3.
    Type: Grant
    Filed: December 21, 1982
    Date of Patent: August 20, 1985
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Alain P. Lacour, Bernard M. Pourrias, Raphael Santamaria
  • Patent number: 4528380
    Abstract: New tetrazole derivatives, characterized in that they correspond to the formula: ##STR1## in which R.sub.1 represents: either a hydrogen atom in any one of the positions 1 to 5 of the tetrazole nucleus, R designating a branched alkyl group comprising at least 5 carbon atoms or a branched alkenyl group, or a methyl group in position 2(3) of the tetrazole nucleus, R representing the (1-propyl)n butyl chain.These new derivatives are useful as medicaments, more especially for their anti-epileptic action.
    Type: Grant
    Filed: December 6, 1982
    Date of Patent: July 9, 1985
    Assignee: Delalande S.A.
    Inventors: Alain P. Lacour, Michel Langlois, Maurice F. Jalfre, Bernard P. Bucher
  • Patent number: 4526786
    Abstract: N-aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones are disclosed. These compounds possess antidepressant activity.
    Type: Grant
    Filed: June 16, 1982
    Date of Patent: July 2, 1985
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Colette A. Douzon, Jean-Francois R. Ancher, Alain P. Lacour, Patrick G. Guerret, Michel Langlois, Phillippe L. Dostert
  • Patent number: 4517197
    Abstract: A compound of the formula ##STR1## where R is selected from the group consisting of CH.sub.3 --CO--(CH.sub.2).sub.2 --O--, ##STR2## The compounds are useful in treating depression.
    Type: Grant
    Filed: July 29, 1983
    Date of Patent: May 14, 1985
    Assignee: Delalande S.A.
    Inventors: Jean-Francois R. Ancher, Guy R. Bourgery, Philippe L. Dostert, Colette A. Douzon, Patrick G. Guerret, Alain P. Lacour, Michel Langlois
  • Patent number: 4500531
    Abstract: A class of known (1-cinnamoyl or 1-phenylethylcarbonyl) piperazine derivatives have been found to be central nervous system stimulants effective to improve the mental alertness and to brighten the spirits of human beings.
    Type: Grant
    Filed: July 27, 1983
    Date of Patent: February 19, 1985
    Assignee: Delalande S.A.
    Inventors: Alain Y. Platel, Alain P. Lacour, Guy R. Bourgery
  • Patent number: 4476136
    Abstract: Derivatives corresponding to the general formula: ##STR1## in which Ar represents a phenyl group; a phenyl group substituted by a halogen atom or by a trifluoromethyl group; or the (chloro-3 fluoro-4) phenyl group and n is either equal to zero or equal to 1 in which case X is a chain chosen from the following: --CH.sub.2 --CH.sub.2 --, --CH.dbd.CH--, --C.tbd.C--, --CH.sub.2 --O-- whose CH.sub.2 group is linked to Ar.These compounds are useful as medicaments more especially for the treatment of troubles of the central nervous system and senescence.
    Type: Grant
    Filed: February 24, 1982
    Date of Patent: October 9, 1984
    Assignee: Delalande S.A.
    Inventors: Philippe L. Dostert, Alain P. Lacour, Michel Langlois, Margherita Strolin-Benedetti
  • Patent number: 4470993
    Abstract: Method of treating the central nervous system troubles such as the Parkinson's disease and the senescence troubles, generally treated by the B type monoamine oxidase inhibitors, which comprises administering internally to a human being requiring such treatment a therapeutically effective amount of N-aryl 5-aminomethyl oxazolidine-2-one derivatives.
    Type: Grant
    Filed: March 3, 1983
    Date of Patent: September 11, 1984
    Assignee: Delalande S.A.
    Inventors: Jean-Francois R. Ancher, Guy R. Bourgery, Philippe L. Dostert, Colette A. Douzon, Patrick G. Guerret, Alain P. Lacour, Michel Langlois, Margherita Strolin-Benedetti
  • Patent number: 4435415
    Abstract: N-aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones are disclosed. These compounds possess antidepressant activity.
    Type: Grant
    Filed: June 16, 1982
    Date of Patent: March 6, 1984
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Colette A. Douzon, Jean-Francois R. Ancher, Alain P. Lacour, Patrick G. Guerret, Michel Langlois, Philippe L. Dostert
  • Patent number: 4413001
    Abstract: N-aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones are disclosed. These compounds possess antidepressant activity.
    Type: Grant
    Filed: June 16, 1982
    Date of Patent: November 1, 1983
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Colette A. Douzon, Jean-Francois R. Ancher, Alain P. Lacour, Patrick G. Guerret, Michel Langlois, Philippe L. Dostert
  • Patent number: 4395416
    Abstract: Derivatives of formula: ##STR1## in which Z< represents: either an amino group of struture >N-R.sub.1 where R.sub.1 represents a linear or branched alkyl group with 1 to 5 carbon atoms or a phenyl group possibly substituted by a chlorine atom, in which case:n=1 or 2,the pair (A, C X) assumes the following values: (S, C.dbd.O), (S, CH.sub.2), (O, CH.sub.2), (O, CH--C.sub.6 H.sub.5), andR represents a hydrogen or halogen atom, one or more methoxy groups or the butadiene-1,3 ylene chain ##STR2## fixed in position 5,6 of the phenyhl nucleus and thus forming with this latter a naphthyl nucleus;or a methylene group (--CH.sub.2 --), in which case:n=1 or 2,A represents the oxygen atom,>C X represents a carbonyl group (>C.dbd.O) or thiocarbonyl group (>C.dbd.S), andR has the same meanings as previously,as well as the mineral or organic acid addition salts thereof. The compounds exhibit anti-convulsion and analgesic activity.
    Type: Grant
    Filed: January 21, 1982
    Date of Patent: July 26, 1983
    Assignee: Delalande S.A.
    Inventors: Michel Langlois, Bernard P. Bucher, Philippe L. Dostert, Alain P. Lacour, Gerard H. Moinet
  • Patent number: 4372967
    Abstract: Derivatives of 5H-furanone-2 and 3H-dihydrofuranone-2, substituted at the 3 position with substituted phenyl and at the 5 position with substituted methyl, are prepared by various processes. The derivatives are inhibitors of monoamine oxidase and are useful for treating depression.
    Type: Grant
    Filed: February 26, 1982
    Date of Patent: February 8, 1983
    Assignee: Delalande S.A.
    Inventors: Michel Langlois, Alain P. Lacour, Bernard P. Bucher, Gisele C. Mocquet
  • Patent number: 4368199
    Abstract: 1-substituted-4-(3,4,5-trimethoxy) cinnamoyl piperazine compounds are disclosed. The compounds exhibit a substantial activity of stimulating cardiac contractile force, without affecting the cardiac frequency, and they also exhibit coronary vasodilatory and hypotensive effects.
    Type: Grant
    Filed: January 16, 1981
    Date of Patent: January 11, 1983
    Assignee: Delalande S.A.
    Inventors: Jean-Francois R. Ancher, Alain P. Lacour, Gerard H. Moinet, Jacky A. Tisne-Versailles
  • Patent number: 4348393
    Abstract: N-aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones are disclosed. These compounds possess antidepressant activity.
    Type: Grant
    Filed: June 4, 1979
    Date of Patent: September 7, 1982
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Colette A. Douzon, Jean-Francois R. Ancher, Alain P. Lacour, Patrick G. Guerret, Michel Langlois, Phillippe L. Dostert
  • Patent number: 4346102
    Abstract: Derivatives of 5H-furanone-2 and 3H-dihydrofuranone-2, substituted at the 3 position with substituted phenyl and at the 5 position with substituted methyl, are prepared by various processes. The derivatives are inhibitors of monoamine oxidase and are useful for treating depression.
    Type: Grant
    Filed: April 28, 1980
    Date of Patent: August 24, 1982
    Assignee: Delalande S.A.
    Inventors: Michel Langlois, Alain P. Lacour, Bernard P. Bucher, Gisele C. Mocquet
  • Patent number: 4287351
    Abstract: N-aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones are disclosed. These compounds possess antidepressant activity.
    Type: Grant
    Filed: February 6, 1980
    Date of Patent: September 1, 1981
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Colette A. Douzon, Jean-Francois R. Ancher, Alain P. Lacour, Patrick G. Guerret, Michel Langlois, Phillippe L. Dostert
  • Patent number: 4248788
    Abstract: Alcohol, thiol, epoxylated alcohol, epoxylated thiol and benzyloxy derivatives of benzodioxane, benzodioxole and benzodioxepine are useful as intermediates for preparing certain useful cinnamoyl piperazines and homopiperazines.
    Type: Grant
    Filed: April 13, 1979
    Date of Patent: February 3, 1981
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Alain P. Lacour, Gerard H. Moinet, Bernard M. Pourrias, Anne-Marie P. Ruch
  • Patent number: 4178442
    Abstract: Cinnamoyl piperazine and homopiperazine derivatives which possess antiangorous activity and activities on the peripheral and cerebral circulation.
    Type: Grant
    Filed: April 10, 1978
    Date of Patent: December 11, 1979
    Assignee: Delalande S. A.
    Inventors: Guy R. Bourgery, Alain P. Lacour, Gerard H. Moinet, Bernard M. Pourrias, Anne-Marie P. Ruch
  • Patent number: 4153620
    Abstract: Aminoalkoxybenzofurans having the formula ##STR1## wherein ##STR2## are either (1) ##STR3## is monoalkylamino, dialkylamino, cycloalkylamino or heterocyclic amino, or (2) ##STR4## (H, 1, 4-methyl piperazino), ##STR5## is piperidino. The compounds possess antidysrhythmic properties.
    Type: Grant
    Filed: June 12, 1978
    Date of Patent: May 8, 1979
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Alain P. Lacour, Bernard M. Pourrias, Genevieve C. Bregeon