Patents by Inventor Andre Szente

Andre Szente has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4005085
    Abstract: Benzophenone derivatives are produced which have the formula ##STR1## wherein R.sub.1 signifies hydrogen, nitro, halogen or trifluoromethyl; R.sub.2 represents hydrogen or halogen; R.sub.3, R.sub.4 and R.sub.5 are the same or different and signify hydrogen or lower alkyl; R.sub.6 and R.sub.7 each represent lower alkyl or together with the nitrogen atom form a morpholino, 4-(lower alkyl)-1-piperazinyl, 1-pyrrolidinyl or piperidino group, A signifies an alkylene group with 2 to 8 C atoms and Y represents oxygen or a group ##STR2## R.sub.8 and R.sub.9 each signifying lower alkyl or together signifying lower alkylene.The benzophenone derivatives and their pharmaceutically acceptable salts exhibit sedative, anti-convulsant, muscle relaxant and anxiolytic activities.Also provided are methods for the preparation of these compounds.
    Type: Grant
    Filed: November 22, 1974
    Date of Patent: January 25, 1977
    Assignee: Hoffmann-La Roche Inc.
    Inventors: Joseph Hellerbach, Andre Szente