Patents by Inventor Annick Goergler

Annick Goergler has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Diazapane derivatives useful as antagonists of neurokinin 1 receptor and methods for their formation
    Patent number: 6452001
    Abstract: The invention relates to compounds of the formula wherein R1, R2 are independently from each other aryl or heteroaryl, wherein the heteroaryl group contains one or two heteroatoms, selected from N, O, or S, and wherein the aryl or heteroaryl groups are optionally substituted by 1 to 3 substituents, which are independently from each other halogen, CF3, lower alkoxy or lower alkyl; R3 is hydrogen, lower alkyl, —(CH2)nN(R)2, —(CH2)n-heteroaryl or is a —(CH2)n-non aromatic heterocycle, which heterocycles are optionally substituted by halogen, CF3, lower alkoxy or lower alkyl; R4 is ═O, ═N(CH2)nCH3 or ═N(CH2)nN(R)2; R3 and R4 may be together with the N and C atoms to which they are attached the group —CR5═N—N═; R5 is hydrogen, —(CH2)nN(R)2, —(CH2)n-heteroaryl or is a —(CH2)n-non aromatic heterocycle, which heterocycles are optionally substituted by halogen, CF3, lower alkoxy or lower alkyl; R is hydrogen or lower alkyl;
    Type: Grant
    Filed: May 14, 2001
    Date of Patent: September 17, 2002
    Assignee: Hoffmann-La Roche Inc.
    Inventors: Guido Galley, Annick Goergler, Thierry Godel, Reinhard Heck
  • Diazapane derivatives useful as antagonists of neurokinin 1 receptor and methods for their formation
    Publication number: 20020010174
    Abstract: The invention relates to compounds of the formula 1
    Type: Application
    Filed: May 14, 2001
    Publication date: January 24, 2002
    Inventors: Guido Galley, Annick Goergler, Thierry Godel, Reinhard Heck
  • Substituted heterocyclic siprodecane compound active as an antagonist of neurokinin 1 receptor
    Publication number: 20020006932
    Abstract: The invention relates to compounds of the formula 1
    Type: Application
    Filed: May 21, 2001
    Publication date: January 17, 2002
    Inventors: Guido Galley, Thierry Godel, Annick Goergler, Torsten Hoffmann, Sabine Kolczewski, Stephan Roever