Patents by Inventor Antonella Ursini

Antonella Ursini has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Methods for the treatment of sleep disorders
    Patent number: 7625904
    Abstract: The invention relates to methods for the treatment of a sleep disorder in a mammal comprising administering to said mammal an effective amount of a compound of formula (I): wherein all variables are as defined herein.
    Type: Grant
    Filed: December 13, 2007
    Date of Patent: December 1, 2009
    Assignee: SmithKline Beecham Corporation
    Inventors: Giuseppe Alvaro, Romano Di Fabio, Riccardo Giovannini, Giuseppe Guercio, Yves St-Denis, Antonella Ursini
  • Chemical Compounds
    Publication number: 20080249108
    Abstract: The invention relates to methods for the treatment of medical conditions comprising administering an effective amount of a compound of formula (I): wherein all variables are as defined herein.
    Type: Application
    Filed: December 13, 2007
    Publication date: October 9, 2008
    Inventors: Giuseppe Alvaro, Romano DI FABIO, Riccardo GIOVANNINI, Giuseppe GUERCIO, Yves ST-DENIS, Antonella URSINI
  • Chemical compounds
    Patent number: 7345041
    Abstract: The invention relates to methods for the treatment of a sleep disorder comprising administering a compound of formula (I): wherein all variables are as defined herein.
    Type: Grant
    Filed: January 18, 2006
    Date of Patent: March 18, 2008
    Assignee: SmithKline Beecham Corporation
    Inventors: Giuseppe Alvaro, Romano Di Fabio, Riccardo Giovannini, Giuseppe Guercio, Yves St-Denis, Antonella Ursini
  • Chemical compounds
    Patent number: 7071196
    Abstract: The invention relates to piperazine derivatives, to processes for their preparation, to pharmaceutical compositions containing them, and to their medical use. The novel compounds are antagonists of tachykinins, including substance P and other neurokinins.
    Type: Grant
    Filed: August 8, 2003
    Date of Patent: July 4, 2006
    Assignee: SmithKline Beecham Croporation
    Inventors: Giuseppe Alvaro, Romano Di Fabio, Riccardo Giovannini, Giuseppe Guercio, Yves St-Denis, Antonella Ursini
  • Chemical compounds
    Publication number: 20060122192
    Abstract: The invention relates to piperazine derivatives, to processes for their preparation, to pharmaceutical compositions containing them, and to their medical use. The novel compounds are antagonists of tachykinins, including substance P and other neurokinins.
    Type: Application
    Filed: January 18, 2006
    Publication date: June 8, 2006
    Inventors: Giuseppe Alvaro, Romano Di Fabio, Riccardo Giovannini, Giuseppe Guercio, Yves St-Denis, Antonella Ursini
  • Chemical compounds
    Patent number: 6951861
    Abstract: The invention relates to piperazine derivatives, to processes for their preparation, to pharmaceutical compositions containing them, and to their medical use. The novel compounds are antagonists of tachykinins, including substance P and other neurokinins.
    Type: Grant
    Filed: October 5, 2000
    Date of Patent: October 4, 2005
    Assignee: SmithKline Beechan Corporation
    Inventors: Giuseppe Alvaro, Romano Di Fabio, Riccardo Giovannini, Giuseppe Guercio, Yves St-Denis, Antonella Ursini, Mauro Corsi, Sergio Melotto
  • Chemical compounds
    Publication number: 20040209893
    Abstract: The invention relates to piperazine derivatives, to processes for their preparation, to pharmaceutical compositions containing them, and to their medical use. The novel compounds are antagonists of tachykinins, including substance P and other neurokinins.
    Type: Application
    Filed: May 4, 2004
    Publication date: October 21, 2004
    Inventors: Giuseppe Alvaro, Romano Di Fabio, Riccardo Giovannini, Giuseppe Guercio, Yves St-Denis, Antonella Ursini
  • Chemical compounds
    Publication number: 20040048862
    Abstract: The invention relates to piperazine derivatives, to processes for their preparation, to pharmaceutical compositions containing them, and to their medical use. The novel compounds are antagonists of tachykinins, including substance P and other neurokinins.
    Type: Application
    Filed: August 8, 2003
    Publication date: March 11, 2004
    Inventors: Giuseppe Alvaro, Romano Di Fabio, Riccardo Giovannini, Giuseppe Guercio, Yves St-Denis, Antonella Ursini
  • Treating emesis in a mammal
    Patent number: 6642240
    Abstract: The invention relates to piperazine derivatives, to processes for their preparation, to pharmaceutical compositions containing them, and to their medical use. The novel compounds are antagonists of tachykinins, including substance P and other neurokinins.
    Type: Grant
    Filed: July 3, 2002
    Date of Patent: November 4, 2003
    Assignee: SmithKline Beecham Corporation
    Inventors: Giuseppe Alvaro, Romano Di Fabio, Riccardo Giovannini, Giuseppe Guercio, Yves St-Denis, Antonella Ursini
  • Chemical compounds
    Publication number: 20030028021
    Abstract: The invention relates to piperazine derivatives, to processes for their preparation, to pharmaceutical compositions containing them, and to their medical use. The novel compounds are antagonists of tachykinins, including substance P and other neurokinins.
    Type: Application
    Filed: July 3, 2002
    Publication date: February 6, 2003
    Inventors: Giuseppe Alvaro, Romano Di Fabio, Riccardo Giovannini, Giuseppe Guercio, Yves St-Denis, Antonella Ursini
  • 1,5-benzodiazepine derivatives
    Patent number: 5716953
    Abstract: Compounds of formula (I) ##STR1## wherein the substituents are defined in the specification are antagonists of gastrin and CCK.
    Type: Grant
    Filed: March 22, 1996
    Date of Patent: February 10, 1998
    Assignee: Glaxo Wellcome S.p.A.
    Inventors: Daniele Donati, Antonella Ursini, Mauro Corsi
  • 1,5-benzodiazepines useful as gastrinor CCK-antagonists
    Patent number: 5686449
    Abstract: The invention relates to compounds of formula (I) ##STR1## and pharmaceutically acceptable salts thereof having gastrin and/or CCK-B antagonist activity.
    Type: Grant
    Filed: October 23, 1995
    Date of Patent: November 11, 1997
    Assignee: Glaxo Wellcome S.p.A.
    Inventors: Maria Elvira Tranquillini, Gabriella Finizia, Antonella Ursini
  • 10(1-hydroxyethyl)-11-oxo-1-azatricyclo/7.2.0.0..sup.3.8/ undec-2-ene-2-carboxylic acid esters and a process for preparing thereof
    Patent number: 5587374
    Abstract: A compound of the formula 1-cyclohexyloxycarbonyloxethyl (4S, 8S, 9R 10S, 12R)-4-methoxy-10-(1-hydroxyethyl)-11-oxo-1-azatricyclo[7.2.0.0..sup.3,8 ]undec-2-ene-2-carboxylate which is useful as a pharmaceutical composition to treat bacterial infection.
    Type: Grant
    Filed: February 14, 1995
    Date of Patent: December 24, 1996
    Assignee: Glaxo SpA
    Inventors: Alcide Perboni, Tino Rossi, Giovanni Gaviraghi, Giorgio Tarzia, Antonella Ursini
  • Carbamate derivatives
    Patent number: 5486514
    Abstract: The present invention relates to compound of formula (I) which are antagonists of gastrin and CCK-B receptors. The compounds of formula (I) are carbamate derivatives.
    Type: Grant
    Filed: July 20, 1994
    Date of Patent: January 23, 1996
    Assignee: Glaxo SpA
    Inventors: David Trist, Giorgio Pentassuglia, Maria E. Tranquillini, Antonella Ursini
  • Chemical compounds
    Patent number: RE39921
    Abstract: The invention relates to piperazine derivatives, to processes for their preparation, to pharmaceutical compositions containing them, and to their medical use. The novel compounds are antagonists of tachykinins, including substance P and other neurokinins.
    Type: Grant
    Filed: October 5, 2004
    Date of Patent: November 13, 2007
    Assignee: SmithKline Beecham Corporation
    Inventors: Giuseppe Alvaro, Romano DiFabio, Riccardo Giovannini, Giuseppe Guercio, Yves St-Denis, Antonella Ursini