Patents by Inventor Claude Oberlander

Claude Oberlander has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 6534515
    Abstract: A compound selected from the group consisting of all possible isomers or racemates of a compound of the formula wherein the various substituents are as defined in the specification and its non-toxic, pharmaceutically acceptable salts with acids or bases having anti-anoxic, anti-ischemic and neuronal protective anti-depressant activities.
    Type: Grant
    Filed: April 15, 1994
    Date of Patent: March 18, 2003
    Assignee: Aventis Pharma S.A.
    Inventors: François Clemence, Jean-Luc Haesslein, Claude Oberlander
  • Publication number: 20020045637
    Abstract: A compound selected from the group consisting of all possible isomers or racemates of a compound of the formula 1
    Type: Application
    Filed: April 15, 1994
    Publication date: April 18, 2002
    Inventors: FRANCOIS CLEMENCE, JEAN-LUC HAESSLEIN, CLAUDE OBERLANDER
  • Patent number: 5424314
    Abstract: A compound in all racemic or optionally active forms selected from the group consisting of a compound of the formula ##STR1## where the substituents are defined as in the specification and their non-toxic, pharmaceutically acceptable acid addition salts having anti-anoxic activity and a novel process and intermediates for their preparation.
    Type: Grant
    Filed: March 7, 1994
    Date of Patent: June 13, 1995
    Assignee: Roussel-Uclaf
    Inventors: Francois Clemence, Jean-Luc Haesslein, Claude Oberlander
  • Patent number: 5332748
    Abstract: A compound and all possible racemic or optically active isomer forms, selected from the group consisting of compound of the formula ##STR1## wherein the substituents are defined as set forth in the application as filed. Useful for treating cerebral insufficiencies of anoxic or ischemic origin.
    Type: Grant
    Filed: January 19, 1993
    Date of Patent: July 26, 1994
    Assignee: Roussel-Uclaf
    Inventors: Nurgun Aktogu, Francois Clemence, Claude Oberlander
  • Patent number: 5093337
    Abstract: The invention concerns compounds of formula (I); ##STR1## in which R.sub.1, R.sub.2 and R.sub.3, identical or different, stand for hydrogen, halogen, alkyl or alkoxy (C.sub.1-5), hydroxy, trifluoromethyl, nitro, amino, alkylamino, dialkylamino, acylamino, R.sub.1, R.sub.2 and R.sub.3 being unable to stand for hydrogen simultaneously and in which (a) stands for (b), (c), or (d), all possible isomeric forms of said products of formula (I) being racemic or optically active, as well as their additional salts with acids, their preparation and the new intermediate products obtained, their application as drugs in particular nootropes, antidepressants, neuronal protectors, anti-anoxics, anti-ischemics, and the compositions containing them.
    Type: Grant
    Filed: July 18, 1989
    Date of Patent: March 3, 1992
    Assignee: Roussel Uclaf
    Inventors: Nurgun Aktogu, Francois Clemence, Claude Oberlander
  • Patent number: 5034396
    Abstract: A compound selected from the group consisting of optically active isomers of a racemic compound of the formula ##STR1## wherein the 3-hydrogen and 16-hydrogen are trans and ##STR2## is selected from the group consisting of ##STR3## with the --OH being .alpha. or .beta. and their non-toxic, pharmaceutically acceptable acid addition salts having antidepressant activity and an affinity for alpha.sub.
    Type: Grant
    Filed: November 15, 1988
    Date of Patent: July 23, 1991
    Assignee: Roussel Uclaf
    Inventors: Nurgun Aktogu, Francois Clemence, Claude Oberlander
  • Patent number: 4975427
    Abstract: A compound selected from the group consisting of a compound of the formula ##STR1## wherein R.sub.1 and R.sub.2 are individually selected from the group consisting of hydrogen, halogen, alkyl and alkoxy of 1 to 5 carbon atoms, hydroxy, trifluoromethyl and nitro, n is 0,1 or 2 and the group: ##STR2## in all possible racemic or optically active isomer forms and their non-toxic, pharmaceutically acceptable acid addition salts having analgesic, anti-anoxic and anti-ischemic neuronal protective properties.
    Type: Grant
    Filed: September 29, 1989
    Date of Patent: December 4, 1990
    Assignee: Roussel Uclaf
    Inventors: Francois Clemence, Jean-Luc Haesslein, Claude Oberlander
  • Patent number: 4904655
    Abstract: Novel compounds selected from the group consisting of all possible racemic or optically active forms of compounds of the formula ##STR1## wherein R.sub.1 and R.sub.2 are individually selected from the group consisting of hydrogen, alkyl and alkoxy of 1 to 5 carbon atoms, -OH, -CF.sub.3 and -NO.sub.2 and ##STR2## is selected from the group consisting of ##STR3## and their non-toxic, pharmaceutically acceptable acid addition salts having a very good analgesic activity as well as antidepressive, neuronal protective, anti-anoxic, anti-ischemic and no-otropic activities.
    Type: Grant
    Filed: January 26, 1989
    Date of Patent: February 27, 1990
    Assignee: Roussel Uclaf
    Inventors: Nurgun Aktogu, Francoise Delevallee, Francois Clemence, Claude Oberlander
  • Patent number: 4736034
    Abstract: A compound selected from the group consisting of a compound of the formulae ##STR1## wherein R.sub.1 ' is selected from the group consisting of alkoxy of 1 to 5 carbon atoms, phenoxy and phenylalkoxy of 7 to 9 carbon atoms, R' is selected from the group consisting of alkyl of 1 to 5 carbon atoms, cycloalkylalkyl of 4 to 7 carbon atoms and phenyl alkyl of 7 to 12 carbon atoms optionally substituted with one or more members of the group consisting of alkyl of 1 to 5 carbon atoms, alkoxy of 1 to 5 carbon atoms, halogen and alkenyl of 3 to 5 carbon atoms and alkynyl of 3 to 5 carbon atoms with the proviso that the multiple bond is not between the carbons .alpha.- and .beta. to the nitrogen atom and B is a reversible secondary amine blocking group and their haloamines.
    Type: Grant
    Filed: March 23, 1987
    Date of Patent: April 5, 1988
    Assignee: Roussel Uclaf
    Inventors: Lucien Nedelec, Patrick Fauveau, Gilles Hamon, Claude Oberlander
  • Patent number: 4694011
    Abstract: Novel 7-hydroxy-indoles of the formula ##STR1## wherein R is selected from the group consisting of hydrogen, alkyl of 1 to 5 carbon atoms, cycloalkylalkyl of 4 to 7 carbon atoms and aralkyl of 7 to 12 carbon atoms optionally substituted by one or more members of the group consisting of alkyl and alkoxy of 1 to 5 carbon atoms, halogen and alkenyl and alkynyl of 3 to 5 carbon atoms with the multiple bond being other than between the carbons .alpha.- and .beta.- to the nitrogen atom, R.sub.1 is selected from the group consisting of --OH, alkoxy of 1 to 5 carbon atoms, phenoxy and phenylalkoxy of 7 to 9 carbon atoms and their non-toxic, pharmaceutically acceptable acid addition salts having remarkable dopaminergic properties with few central effects and a novel process and novel intermediates for their preparation.
    Type: Grant
    Filed: March 10, 1986
    Date of Patent: September 15, 1987
    Assignee: Roussel Uclaf
    Inventors: Lucien Nedelec, Gilles Hamon, Patrick Fauveau, Claude Oberlander
  • Patent number: 4661482
    Abstract: Novel pyrazolobenzoxazines of the formula ##STR1## wherein R is selected from the group consisting of hydrogen, alkyl of 1 to 5 carbon atoms, cycloalkylalkyl or 4 to 7 carbon atoms, alkenyl and alkynyl of 3 to 5 carbon atoms with the proviso that the multiple bond is not between the carbon .alpha.- and .beta.- to the nitrogen atom, aralkyl of 7 to 12 carbon atoms and aralkyl of 7 to 12 carbon atoms substituted with at least one member of the group consisting of alkyl and alkoxy of 1 to 5 carbon atoms, amino, -OH and halogen, X is selected from the group consisting of hydrogen and --CH.sub.2 --S--Alk, Alk is alkyl of 1 to 5 carbon atoms, the wavy line indicates the .alpha.- or .beta.-position and their non-toxic, pharmaceutically acceptable acid addition salts having dopaminergic agonistic, hypotensive, antihypertensive and antianoxic properties and their preparation.
    Type: Grant
    Filed: February 25, 1986
    Date of Patent: April 28, 1987
    Assignee: Roussel Uclaf
    Inventors: Lucien Nedelec, Patrick Fauveau, Gilles Hamon, Claude Oberlander
  • Patent number: 4112093
    Abstract: Novel dopaminerginic compositions comprised of an dopaminergically effective amount of at least one member of the group consisting of N-(3,4-methylenedioxy-benzyl)-N'-(2-pyridyl)-piperazine and its non-toxic, pharmaceutically acceptable acid addition salts and an inert pharmaceutical carrier and to a novel method of treating the symptoms of Parkinson disease.
    Type: Grant
    Filed: June 16, 1977
    Date of Patent: September 5, 1978
    Assignee: Roussel Uclaf
    Inventors: Claude Dumont, Claude Oberlander