Patents by Inventor Colin Keith SKEPPER

Colin Keith SKEPPER has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • COMPOUNDS AND COMPOSITIONS FOR MODULATING THE ACTIVITY OF ERK
    Publication number: 20250092036
    Abstract: The invention relates to compounds which modulate the activity of ERK. The present invention also relates to processes for the preparation of said compounds, pharmaceutical compositions comprising said compounds, and use of said compounds in the treatment of conditions, diseases and disorders mediated by ERK.
    Type: Application
    Filed: August 12, 2024
    Publication date: March 20, 2025
    Inventors: Erich W. BAUM, Thomas A. DINEEN, JR., Jonathan Edward HEMPEL, Matthew James HESSE, Robert KOENIG, Matthew James LAMARCHE, Jay Francis LARROW, Ruowei MO, Henrik MOEBITZ, Rukundo NTAGANDA, Keith Bruce PFISTER, Martin SENDZIK, Colin Keith SKEPPER, Joseph WZOREK, JR., Frédéric ZECRI
  • Quinolone derivatives as antibacterials
    Patent number: 10160726
    Abstract: This invention is in the field of medicinal chemistry and relates to compounds, and pharmaceutical compositions thereof, that inhibit bacterial gyrase. The compounds are useful as inhibitors of bacterial gyrase activity and bacterial infections, and have the structure of Formula (I) as further described herein. The invention further provides pharmaceutical compositions comprising a compound of Formula (I) and methods of using the compounds and compositions to treat bacterial infections.
    Type: Grant
    Filed: August 3, 2015
    Date of Patent: December 25, 2018
    Assignee: Novartis AG
    Inventors: Javier de Vicente Fidalgo, Haiying He, Cheng Hu, Zhigan Jiang, Xiaolin Li, Peichao Lu, Wosenu Mergo, Daniel Mutnick, Folkert Reck, Alexey Rivkin, Colin Keith Skepper, Xiaojing Michael Wang, Jianhua Xia, Yongjin Xu
  • TRICYCLIC 2-QUINOLINONES AS ANTIBACTERIALS
    Publication number: 20180318311
    Abstract: This invention is in the field of medicinal chemistry and relates to compounds, and pharmaceutical compositions thereof that are useful as antibacterial agents. The compounds are useful as inhibitors of bacterial gyrase activity and of bacterial infections, and have the structure of Formula (I): as further described herein. The invention further provides pharmaceutical compositions comprising a compound of Formula (I) and methods of using the compounds and compositions to treat bacterial infections.
    Type: Application
    Filed: May 4, 2018
    Publication date: November 8, 2018
    Inventors: Guillaume LAPOINTE, Wosenu MERGO, Heinz Ernst MOSER, Alexey RIVKIN, Colin Keith SKEPPER, Sarah Louise Williams
  • QUINOLONE DERIVATIVES AS ANTIBACTERIALS
    Publication number: 20170217897
    Abstract: This invention is in the field of medicinal chemistry and relates to compounds, and pharmaceutical compositions thereof, that inhibit bacterial gyrase. The compounds are useful as inhibitors of bacterial gyrase activity and bacterial infections, and have the structure of Formula (I) as further described herein. The invention further provides pharmaceutical compositions comprising a compound of Formula (I) and methods of using the compounds and compositions to treat bacterial infections.
    Type: Application
    Filed: August 3, 2015
    Publication date: August 3, 2017
    Inventors: Javier de Vicente FIDALGO, Haiying HE, Cheng HU, Zhigan JIANG, Xiaolin LI, Peichao LU, Wosenu MERGO, Daniel MUTNICK, Folkert RECK, Alexey RIVKIN, Colin Keith SKEPPER, Xiaojing Michael WANG, Jianhua XIA, Yongjin XU