Patents by Inventor Daniel Coussediere

Daniel Coussediere has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4873256
    Abstract: A compound in all possible racemic and optically active forms of the formula ##STR1## wherein .dbd.X is .dbd.O or imino having antiandrogenic activity and novel intermediates and processes for their preparations.
    Type: Grant
    Filed: August 10, 1988
    Date of Patent: October 10, 1989
    Assignee: Roussel Uclaf
    Inventors: Daniel Coussediere, Giuseppe Gigliotti, Martine Moguilewsky
  • Patent number: 4273771
    Abstract: Novel .DELTA..sup.4,9 -gonadiene-21-ol-3,20-diones of the formula ##STR1## wherein X is selected from the group consisting of hydrogen and tritium, R.sub.1 is alkyl of 1 to 3 carbon atoms, R.sub.2 is alkyl of 1 to 12 carbon atoms and R.sub.3 is alkyl of 1 to 4 carbon atoms in the form of 21R or 21S epimers or mixtures thereof having progestomimetic and antiestrogenic properties, their preparation and novel intermediates.
    Type: Grant
    Filed: July 5, 1979
    Date of Patent: June 16, 1981
    Assignee: Roussel Uclaf
    Inventor: Daniel Coussediere
  • Patent number: 4064339
    Abstract: There are disclosed pharmaceutically-active aminoglycosides comprising 4-O-(2',6'-diamino 2',6'-didesoxy .alpha.,D-glucopyrannosyl) 6-O-(3"-amino 3",4",6"-tridesoxy .alpha., D-xylohexopyrannosyl) 2-desoxy streptamine of the formula: ##STR1## and the addition salts thereof with mineral acids or organic acids. Also disclosed are methods for preparation of the novel products as well as certain novel intermediate products. There are also disclosed pharmaceutical compositions in which the novel products are the active agents as well as methods for use of compositions as antibiotic agents.
    Type: Grant
    Filed: March 11, 1975
    Date of Patent: December 20, 1977
    Assignee: Roussel UCLAF
    Inventors: Daniel Coussediere, Jean-Claude Gasc
  • Patent number: 3981861
    Abstract: There are disclosed pharmaceutically-active aminoglycosides comprising 4-0-(2',6'-diamino 2', 3', 4', 6'-tetradesoxy .alpha.,D-erythrohexopyrannosyl) 6-0-(3"-methylamino 3", 4", 6"-tridesoxy .alpha.,D-xylohexopyrannosyl) 2-desoxystreptamine of the formula: ##SPC1##And the addition salts thereof with mineral acids or organic acids. Also disclosed are methods for preparation of the novel products as well as certain novel intermediate products. There are also disclosed pharmaceutical compositions in which the novel products are the active agents as well as methods for use of compositions as antibiotic agents.
    Type: Grant
    Filed: March 7, 1975
    Date of Patent: September 21, 1976
    Assignee: Roussel-UCLAF
    Inventors: Jean Bernard Chazan, Daniel Coussediere, Jean-Claude Gasc
  • Patent number: 3975413
    Abstract: Novel haptenes of the formula ##SPC1##Wherein X is ##EQU1## when Y is ##EQU2## in the .alpha.- or .beta.-position and R' is selected from the group of p-phenylene and --(CH.sub.2).sub.a --and a is a whole number from 1 to 18 with the proviso that a is other than 2 when Y is in the .alpha.-position and when Y is hydrogen, X is selected from the group consisting of ##EQU3## and =N--O--(CH.sub.2).sub.c --COOH, b is a whole number from 1 to 18 and c is a whole number from 1 to 12 useful for the preparation of antigens formed therefrom.
    Type: Grant
    Filed: July 2, 1975
    Date of Patent: August 17, 1976
    Inventors: Andre Pierdet, Daniel Coussediere
  • Patent number: 3959255
    Abstract: There are disclosed pharmaceutically-active aminoglycosides comprising 4-O-[2',6'-diamino-2',6'-didesoxy-.alpha.-D-glucopyranosyl] 6-O-[3"-methylamino-3",4",6"-tridesoxy-.alpha.-D-xylohexopyranosyl] 2-desoxy streptamine of the formula: ##SPC1##And the addition salts thereof with mineral acids or organic acids. Also disclosed are methods for preparation of the novel products as well as certain novel intermediate products. There are also disclosed pharmaceutical compositions in which the novel products are the active agents as well as methods for use of compositions as antibiotic agents.
    Type: Grant
    Filed: April 29, 1974
    Date of Patent: May 25, 1976
    Assignee: Roussel-UCLAF
    Inventors: Jean-Bernard Chazan, Daniel Coussediere, Jean-Claude Gasc