Patents by Inventor Derek A. Rawlings

Derek A. Rawlings has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Pyridine derivatives as cb2 receptor modulators
    Publication number: 20070129367
    Abstract: The present invention relates to novel pyridine derivatives, pharmaceutical compositions containing these compounds and their use in the treatment of diseases, particularly pain, which diseases are caused directly or indirectly by an increase or decrease in activity of the cannabinoid receptor.
    Type: Application
    Filed: September 25, 2003
    Publication date: June 7, 2007
    Inventors: Andrew Eatherton, Gerard Giblin, Richard Green, Jennifer Doughty, Karamjit Jandu, William Mitchell, Alan Naylor, Giovanni Palombi, Derek Rawlings, Brian Slingsby, Andrew Whittington
  • Pyrimidine compounds
    Publication number: 20060247261
    Abstract: The present invention relates to novel pyrimidine derivatives, pharmaceutical compositions containing these compounds and their use in the treatment of diseases, particularly pain, which diseases are caused directly or indirectly by an increase or decrease in activity of the cannabinoid receptor.
    Type: Application
    Filed: August 19, 2003
    Publication date: November 2, 2006
    Inventors: Andrew Eatherton, Gerard Giblin, Richard Green, Jennifer Doughty, William Mitchell, Alan Naylor, Derek Rawlings, Brian Slingsby, Andrew Whittington
  • Pyridine derivatives as cb2 receptor modulators
    Publication number: 20060240048
    Abstract: The present invention relates to novel pyridine derivatives, pharmaceutical compositions containing these compounds and their use in the treatment of diseases, particularly pain, which diseases are caused directly or indirectly by an increase or decrease in activity of the cannabinoid receptor.
    Type: Application
    Filed: September 25, 2003
    Publication date: October 26, 2006
    Inventors: Andrew Eatherton, Gerard Martin Giblin, Richard Green, Jennifer Doughty, Karamjit Jandu, William Mitchell, Alan Naylor, Giovanni Palombi, Derek Rawlings, Brian Slingsby, Andrew Whittington
  • Phenylpyrimidones
    Patent number: 5118686
    Abstract: This invention relates to phenylpyrimidone derivatives which have bronchodilator activity. A compound of the invention is 4-cyano-6-hydroxy-2-(2-propoxyphenyl)pyrimidine.
    Type: Grant
    Filed: April 25, 1990
    Date of Patent: June 2, 1992
    Assignee: Smith Kline & French Laboratories Limited
    Inventors: William J. Coates, Derek A. Rawlings
  • Pyrimidone derivatives as bronchodilators
    Patent number: 5075310
    Abstract: This invention relates to fused pyrimidine derivatives which have bronchodilator activity. A compound of this invention is 2-(2-propoxyphenyl)thieno[2,3-d]pyrimidin-4(3H)-one.
    Type: Grant
    Filed: June 23, 1989
    Date of Patent: December 24, 1991
    Assignee: Smith Kline & French Laboratories, Ltd.
    Inventors: William J. Coates, Derek A. Rawlings
  • Chemical compounds
    Patent number: 5047404
    Abstract: This invention relates to fused pyrimidine derivatives which have bronchodilator and anti-allergic activities. A compound of the invention is 2-(2-propoxyphenyl)pyrido[2,3-d]pyrimid-4(3H)-one.
    Type: Grant
    Filed: June 13, 1989
    Date of Patent: September 10, 1991
    Assignee: Smith Kline & French Laboratories, Ltd.
    Inventors: William J. Coates, Sean T. Flynn, Derek A. Rawlings
  • N-Substituted pyridinones having histamine H.sub.2 -antagonist activity
    Patent number: 4540699
    Abstract: This invention relates to N-substituted pyridinone compounds which have histamine H.sub.2 -antagonist activity. A specific compound of this invention is 2-[2-(5-methyl-4-imidazolylmethylthio)ethylamino]-5-(1-methyl-2-oxopyridin -4-ylmethyl)pyrimidin-4-one.
    Type: Grant
    Filed: November 29, 1983
    Date of Patent: September 10, 1985
    Assignee: Smith Kline & French Laboratories Limited
    Inventors: Thomas H. Brown, Derek A. Rawlings