Patents by Inventor Erik WEIS

Erik WEIS has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • PCSK9 INHIBITORS AND METHODS OF USE THEREOF
    Publication number: 20240239767
    Abstract: A compound with the Formula (I): wherein A is of the following formula: and X1 is selected from O, S or NH; X2 is either N or C—H X3 is either N or C—RA3; wherein if X1 is NH and X2 is C—H then X3 is C—RA3; B is of formula (B-1) or (B-2) C is selected from the group consisting of optionally substituted C6-10 carboaryl, C5-6 heteroaryl or C5-10 heterocyclyl, and their use as PCSK9 inhibitors.
    Type: Application
    Filed: December 14, 2023
    Publication date: July 18, 2024
    Inventors: Gavin Donal O’MAHONY, Olaf PANKNIN, Andrey FROLOV, Anna TOMBERG, Mateusz Piotr PLESNIAK, Jens Peter BRANDT, Erik WEIS, Jens Patrik JOHANSSON, Emma BRATT
  • PCSK9 INHIBITORS AND METHODS OF USE THEREOF
    Publication number: 20240228469
    Abstract: A compound with the Formula (I): A-B-C??(I) wherein A is of the following formula: where X1 is N B is of formula (B-1) or (B-2) and C is selected from the group consisting of optionally substituted C6-10 carboaryl, C5-6 heteroaryl and C5-10 heterocyclyl and their use as PCSK9 inhibitors.
    Type: Application
    Filed: September 20, 2023
    Publication date: July 11, 2024
    Inventors: Gavin Donal O’MAHONY, Olaf PANKNIN, Andrey FROLOV, Anna TOMBERG, Erik WEIS, Hans Frederik BERGSTRÖM, Karl Thomas ANTONSSON, Jan Åke LINDBERG, Jens Patrik JOHANSSON
  • Scalable process for the preparation of a GlyT-1 Inhibitor
    Publication number: 20240083889
    Abstract: This invention relates to a synthetic method for the preparation of Compound 1 and precursors thereof. Compound 1 is prepared via reaction of isoxazole 2 with phenylether (R)-3-ONa.
    Type: Application
    Filed: August 24, 2023
    Publication date: March 14, 2024
    Inventors: Katrin BAER, Gisela BODENBACH, Jack Delbert BROWN, Rosemarie Karoline COLLET, Daniel HERKOMMER, Rogelio P. FRUTOS, Joe Ju GAO, Julia Regina GRIMM, Sandra KOCH, Sonia RODRIGUEZ, Svetlana SEHL-OLLENBERGER, Joshua Daniel SIEBER, Thomas G. TAMPONE, Ulrich THEIS, Dirk WEBER, Erik WEIS, Anke WILD