Patents by Inventor Gerard Giblin

Gerard Giblin has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Process for preparing alpha-carboxamide pyrrolidine derivatives
    Patent number: 10421716
    Abstract: The invention relates to a novel process for preparing ?-carboxamide pyrrolidine derivatives, in particular (2S, 5R)-5-(4-((2-fluorobenzyl)oxy)phenyl)pyrrolidine-2-carboxamide, and to novel intermediates for use in said process along with processes for preparing said intermediates.
    Type: Grant
    Filed: December 23, 2015
    Date of Patent: September 24, 2019
    Assignee: Convergence Pharmaceuticals Limited
    Inventors: David MacPherson, David Witty, Gerard Giblin, Michael Williams, Donald Walker, William Kiesman, Tamera Mack
  • Process for Preparing Alpha-Carboxamide Pyrrolidine Derivatives
    Publication number: 20170369437
    Abstract: The invention relates to a novel process for preparing ?-carboxamide pyrrolidine derivatives, in particular (2S, 5R)-5-(4-((2-fluorobenzyl)oxy)phenyl)pyrrolidine-2-carboxamide, and to novel intermediates for use in said process along with processes for preparing said intermediates.
    Type: Application
    Filed: December 23, 2015
    Publication date: December 28, 2017
    Inventors: David MacPherson, David WITTY, Gerard GIBLIN, Michael WILLIAMS, Donald WALKER, William KIESMAN, Tamera MACK
  • Pyrrolopyridine Derivatives
    Publication number: 20070219229
    Abstract: The present invention relates to novel pyrrolopyridine derivatives, pharmaceutical compositions containing these compounds and their use in the treatment of diseases, particularly pain, which diseases are caused directly or indirectly by an increase or decrease in activity of the cannabinoid receptor.
    Type: Application
    Filed: June 7, 2005
    Publication date: September 20, 2007
    Applicant: GLAXO GROUP LIMITED
    Inventors: Andrew Eatherton, Gerard Giblin, Matthew Johnson, William Mitchell, Brian Slingsby, Alcide Perboni
  • Pyridine derivatives as cb2 receptor modulators
    Publication number: 20070129367
    Abstract: The present invention relates to novel pyridine derivatives, pharmaceutical compositions containing these compounds and their use in the treatment of diseases, particularly pain, which diseases are caused directly or indirectly by an increase or decrease in activity of the cannabinoid receptor.
    Type: Application
    Filed: September 25, 2003
    Publication date: June 7, 2007
    Inventors: Andrew Eatherton, Gerard Giblin, Richard Green, Jennifer Doughty, Karamjit Jandu, William Mitchell, Alan Naylor, Giovanni Palombi, Derek Rawlings, Brian Slingsby, Andrew Whittington
  • Benzo[F]Isoindole Derivatives With Affinity To The EP4 Receptor
    Publication number: 20070088068
    Abstract: A compound of formula (I) and processes for the preparation thereof.
    Type: Application
    Filed: November 8, 2006
    Publication date: April 19, 2007
    Inventors: Miles Congreve, Gerard Giblin, Andrew Mason, Neil Miller, Susan Roomans, Ann Walker
  • Pyrrole compounds for the treatment of prostaglandine mediated diseases
    Publication number: 20070082912
    Abstract: Compounds of formula (I) or a pharmaceutically acceptable derivative thereof: wherein A, R1, R2a, R2b, Rx, R8, and R9 are as defined in the specification, a process for the preparation of such compounds, pharmaceutical compositions comprising such compounds and the use of such compounds in medicine.
    Type: Application
    Filed: May 30, 2003
    Publication date: April 12, 2007
    Inventors: Gerard Giblin, Adrian Hall, Mark Healy, Xiao Lewell, Neil Miller, Riccardo Novelli
  • Pyrrole compounds
    Publication number: 20070072906
    Abstract: Compounds of formula (I) or a derivative thereof: wherein A, B, Z, R1, R2a, R2b, Rx, R6, and R9 are as defined in the specification, a process for the preparation of such compounds, pharmaceutical compositions comprising such compounds and the use of such compounds in medicine.
    Type: Application
    Filed: November 30, 2004
    Publication date: March 29, 2007
    Inventors: Gerard Giblin, Adrian Hall, Mark Healy, Francis King, Xiao Lewell, Neil Miller, Alan Naylor, Riccardo Novelli
  • Heterocyclyl compounds
    Publication number: 20070060596
    Abstract: Compounds of formula (I) or a pharmaceutically acceptable derivative thereof: wherein W, X, Y, Z, R1, R2a, R2b, and Rx, R8 and R9 are as defined in the specification, a process for the preparation of such compounds, pharmaceutical compositions comprising such compounds and the use of such compounds in medicine.
    Type: Application
    Filed: October 21, 2004
    Publication date: March 15, 2007
    Inventors: Gerard Giblin, Adrian Hall, David Hurst, Xiao Lewell, Olivier Lorthioir, Stephen Mickeown, Tiziana Scoccitti, Stephen Watson
  • Pyrimidine compounds
    Publication number: 20060247261
    Abstract: The present invention relates to novel pyrimidine derivatives, pharmaceutical compositions containing these compounds and their use in the treatment of diseases, particularly pain, which diseases are caused directly or indirectly by an increase or decrease in activity of the cannabinoid receptor.
    Type: Application
    Filed: August 19, 2003
    Publication date: November 2, 2006
    Inventors: Andrew Eatherton, Gerard Giblin, Richard Green, Jennifer Doughty, William Mitchell, Alan Naylor, Derek Rawlings, Brian Slingsby, Andrew Whittington
  • Phenyl compounds
    Publication number: 20060235057
    Abstract: Compounds of formula (I) or derivatives thereof: wherein A, B, Z, R1, R2a, R2b, Rx, R8, and R9 are as defined in the specification, a process for the preparation of such compounds, pharmaceutical compositions comprising such compounds and the use of such compounds in medicine.
    Type: Application
    Filed: October 30, 2003
    Publication date: October 19, 2006
    Inventors: Rino Bit, Gerard Giblin, Adrian Hall, David Hurst, Ian Kilford, Neil Miller, Tiziana Scoccitti
  • Benzo'fisoindole derivatives with affinity to the ep4 receptor
    Publication number: 20050080257
    Abstract: The present invention relates to a compound of formula (I): corresponding pharmaceutical compositions, preparation processes, and/or methods of using the aforementioned compounds and/or compositions.
    Type: Application
    Filed: February 7, 2002
    Publication date: April 14, 2005
    Inventors: Miles Congreve, Gerard Giblin, Neil Miller, Susan Roomans, Ann Walker, Andrew Mason