Patents by Inventor GERD-VOLKER ROSCHENTHALER

GERD-VOLKER ROSCHENTHALER has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Publication number: 20070154537
    Abstract: A bisphosphonic acid of the general formula (I) wherein R1 is H, OH, C1-C6 alkyl C1-C6 alkoxy, C1-C6 hydroxyalkyl, C1-C6 aminoalkyl, C1-C6 halogen alkyl X is a direct bond, alkylen group with 1 to 20 carbon atoms, (CH3)m—(OCR3HCH2)n—(O)o— wherein R3 is H or CH3 and m is 0 or a number from 1 to 6, n is a number from 1 to 10, preferably 1 to 6, and o is 0 or 1, ?—(CR4HCH2O)p— wherein R4 is H or CH3, p is a number from 1 to 10, preferably 1 to 6, ?(CH3)q—(OCR5HCH2)r—(O)s—(CH3)t—, wherein R5 is H or CH3 and q is 0 or a number from 1 to 6, r is a number from 1 to 10, preferably 1 to 6, and s is 0 or 1, and t is a number from 1 to 6, R2 is a group of the formula (II) as well as their physiologically compatible derivatives, in particular salts and trimethyl silyl derivatives.
    Type: Application
    Filed: January 24, 2005
    Publication date: July 5, 2007
    Applicant: MCS MICRO CARRIER SYSTEMS GMBH
    Inventors: Wolfgang Greb, Oleg Shyhskov, Gerd-Volker Roschenthaler, Verena Hengst
  • Patent number: 7078393
    Abstract: In a method for preparing 1-hydroxy-1,1-diphosphonic acid compounds of the general formula I and/or of their pharmacologically compatible salts a compound of the formula II is reacted with a compound P(OSiR53)3-pR6p and the reaction product is hydrolyzed.
    Type: Grant
    Filed: March 12, 2002
    Date of Patent: July 18, 2006
    Assignee: EUCRO European Contract Research GmbH & Co. KG
    Inventors: Helmut Blum, Wolfgang Greb, Yurii Pustovit, Gerd-Volker Röschenthaler
  • Patent number: 7045662
    Abstract: The present invention relates to a process for preparing ?,?-difluoroamines, difluoromethylene-?,?-diazo compounds and fluorination reagents containing ?,?-difluoroamines and/or difluoromethylene-?,?-diazo compounds.
    Type: Grant
    Filed: January 5, 2004
    Date of Patent: May 16, 2006
    Assignee: Bayer Chemicals AG
    Inventors: Wolfgang Ebenbeck, Albrecht Marhold, Alexander Kolomeitsev, Gerd-Volker Röschenthaler
  • Publication number: 20050085474
    Abstract: The present invention relates to ?,?-difluoroamines, fluorinating reagents comprising ?,?-difluoroamines and also processes for preparing ?,?-difluoroamines and fluorinating reagents comprising ?,?-difluoroamines.
    Type: Application
    Filed: January 5, 2004
    Publication date: April 21, 2005
    Inventors: Wolfgang Ebenbeck, Petra Hilgers, Albrecht Marhold, Jan Barten, Alexander Kolomeitsev, Gerd-Volker Roschenthaler
  • Patent number: 6875894
    Abstract: The invention relates to bis(alkylthio)carbenium salts of the formula I with the stated definitions for R1, R2, R3 and Y?, and to a process for the preparation thereof. The compounds according to the invention are advantageously suitable as electrophilic reagents for the transfer of fluorinated alkyl and acyl radicals onto nucleophilic compounds.
    Type: Grant
    Filed: February 11, 2002
    Date of Patent: April 5, 2005
    Assignee: Merck Patent GmbH
    Inventors: Peer Kirsch, Andreas Ruhl, Gerd-Volker Röschenthaler, Dmitrii Sevenard
  • Patent number: 6872861
    Abstract: The invention relates to a process for preparing polyfluoroalkyl-lithium compounds by deprotonation of polyfluoroalkyl compounds by means of lithium bases.
    Type: Grant
    Filed: June 7, 2002
    Date of Patent: March 29, 2005
    Assignee: Bayer Aktiengesellschaft
    Inventors: Marielouise Schneider, Albrecht Marhold, Alexander Kolomeitsev, Alexander Kadyrov, Gerd-Volker Röschenthaler, Jan Barten
  • Publication number: 20040198975
    Abstract: The present invention relates to a process for preparing &agr;,&agr;-difluoroamines, difluoromethylene-&agr;,&agr;-diazo compounds and fluorination reagents containing &agr;,&agr;-difluoroamines and/or difluoromethylene-&agr;,&agr;-diazo compounds.
    Type: Application
    Filed: January 5, 2004
    Publication date: October 7, 2004
    Inventors: Wolfgang Ebenbeck, Albrecht Marhold, Alexander Kolomeitsev, Gerd-Volker Roschenthaler
  • Publication number: 20040087554
    Abstract: The invention relates to a method of producing the 1-hydroxy-1,1-diphosphonic acid compounds of general formula (I), and/or the pharmacologically acceptable salts thereof, in which formula R1 represents hydrogen, OH, NO2, Cl, F, Br, C1-C6 alkyl that may be substituted with halogen, amine and/or aminoalkyl, C1-6 alkoxy, aryl, heteroaryl, a group NR3R4, wherein R3 and R4 may be the same or different and represent hydrogen, C1-C6 alkyl, halogen-substituted alkyl, hydroxy-C1-alkyl; R2 represents hydrogen, halogen, amine that may be substituted, C1-C6 alkyl that may be substituted with halogen, amine and/or aminoalkyl, C1-C6 alkoxy, aryl, heteroaryl; Y represents O, S or NH; Z represents C1-C5 alkylene that may be substituted with amine groups, and m and n are 0 or 1, with the proviso that if n=1, m=1.
    Type: Application
    Filed: September 15, 2003
    Publication date: May 6, 2004
    Inventors: Helmut Blum, Wolfgang Greb, Yurii Pustovit, Gerd-Volker Roschenthaler
  • Publication number: 20040063985
    Abstract: The invention relates to bis(alkylthio)carbenium salts of the formula I 1
    Type: Application
    Filed: August 13, 2003
    Publication date: April 1, 2004
    Inventors: Peer Kirsch, Andreas Ruhl, Gerd-Volker Roschenthaler, Dmitrii Sevenard
  • Publication number: 20030065135
    Abstract: The invention relates to a process for preparing polyfluoroalkyl-lithium compounds by deprotonation of polyfluoroalkyl compounds by means of lithium bases.
    Type: Application
    Filed: June 7, 2002
    Publication date: April 3, 2003
    Inventors: Marielouise Schneider, Albrecht Marhold, Alexander Kolomeitsev, Alexander Kadyrov, Gerd-Volker Roschenthaler, Jan Barten
  • Publication number: 20020160261
    Abstract: The invention relates to borate salts and to their use in electro-chemical cells.
    Type: Application
    Filed: January 24, 2002
    Publication date: October 31, 2002
    Applicant: Merck GmbH
    Inventors: Michael Schmidt, Andreas Kuhner, Klaus-Dieter Franz, Gerd-Volker Roschenthaler, German Bissky, Alexander Kolomeitsev, Alexander Kadyrov