Patent number: 6696607
Abstract: Use of phenethylacrylamides of the formula I:
in which the substituents have the following meanings:
X is halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and —O—C(Ra,Rb)—C≡C—R6;
Ra,Rb and Rc have the meanings given in the description;
m,n independently of one another are 1 to 4, it being possible for the radicals X or Y to be different if m or n is greater than 1;
Y is halogen, nitro, cyano, alkyl, CF3, alkoxy and phenyl;
R1,R2 independently of one another are hydrogen, halogen, alkyl, alkoxy, haloalkoxy and CF3;
R3,R4,R5,R6 independently of one another are hydrogen, halogen, alkyl, alkoxy, or
R3 and R4 together form a cyclopropyl ring, it being possible for the C—R5— and C—R6 bonds can be in the E- or Z-position relative to each other;
for controlling phytopathogenic fungal pests, novel phenethylacrylamides, their preparation, and compositions comprising them.
Type:
Grant
Filed:
December 4, 2002
Date of Patent:
February 24, 2004
Assignee:
BASF Aktiengesellschaft
Inventors:
Wassilios Grammenos, Hubert Sauter, Oliver Cullmann, Markus Gewehr, Bernd Müller, Jordi Tormo i Blasco, Norbert Götz, Thorsten Volk, Gisela Lorenz, Eberhard Ammermann, Reinhard Stierl, Siegfried Strathmann
Patent number: 6680283
Abstract: Agrochemical compositions having fungicidal action and comprising as active compounds compounds of the formula I
where
R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-haloalkylcarbonyl;
R2 is halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halo-C1-C6-alkylsulfonyl, cyano or a radical NR13R14;
R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halo-C1-C6-alkyl, C1-C6-alkoxy, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halo-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which may be unsubstituted or substituted by halogen, C1-C6-alkyl or halo-C1-C6-alkyl,
R13 is hydrogen, C1-C6-alkyl,
R14 is C1-C6-alkyl, C1-C8-cycloalkyl or, together with R13 and the nitrogen atom to which they are attached, a saturated or unsaturated heterocyclic five- or six-membered ring which contains one or two heteroatoms selected from the group co
Type:
Grant
Filed:
April 11, 2003
Date of Patent:
January 20, 2004
Assignee:
BASF Aktiengesellschaft
Inventors:
Joachim Rheinheimer, Karl Eicken, Ingo Rose, Thomas Grote, Eberhard Ammermann, John-Bryan Speakman, Siegfried Strathmann, Gisela Lorenz
Publication number: 20030191190
Abstract: The invention relates to the use of phenethyl acrylamides of formula I for controlling phytopathogenic fungi, wherein the substituents of said phenethyl acrylamides have the following significations: X signifies halogen, alkyl, halogenalkyl, alkoxy halogenalkoxy and —O—C(Ra, Rb)—C≡C—R6; Ra, Rb and Rc have the signification given in the description; m, n independently signify 1 to 4, the radicals X or Y being potentially different if m or n is higher than 1; Y signifies halogen, nitro, cyano, alkyl, CF3, alkoxy and phenyl; R1, R2 independently signify hydrogen, halogen, alkyl, alkoxy, halogenalkoxy and CF3; R3, R4, R5, and R6 independently signify hydrogen, alkyl and alkoxy, or R3 and R4 together form a cyclopropyl ring, whereby the C—R5 and C—R6 bonds can be in position E or Z in relation to each other. The invention also relates to novel phenethyl acrylamides, a method for the productio thereof, and agents containing the same.
Type:
Application
Filed:
December 4, 2002
Publication date:
October 9, 2003
Inventors:
Wassilios Grammenos, Hubert Sauter, Oliver Cullmann, Markus Gewehr, Bernd Muller, Jordi Tormo i Blasco, Norbert Gotz, Thorsten Volk, Gisela Lorenz, Eberhard Ammermann, Reinhard Stierl, Siegfried Strathman
Patent number: 6593315
Abstract: Salicylic acid derivatives of the formula I,
where the index and the substituents have the following meanings:
X is halogen, NO2, cyano, alkyl or alkoxy;
m is 0, 1, 2 or 3, it being possible for the substituents X to be different from each other if n is greater than 1;
A is OH, alkoxy, NH2, NHCH3 or N(CH3)2;
R1 is phenyl, naphthyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, comprising one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted;
R2 is hydrogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy or alkylthio,
processes for the preparation of these compounds, compositions comprising them, and their use for controlling harmful fungi.
Type:
Grant
Filed:
July 2, 2001
Date of Patent:
July 15, 2003
Assignee:
BASF Aktiengesellschaft
Inventors:
Andreas Gypser, Thomas Grote, Joachim Rheinheimer, Ingo Rose, Oliver Cullmann, Markus Gewehr, Wassilios Grammenos, Jordi Tormo i Blasco, Bernd Müller, Hubert Sauter, Eberhard Ammermann, Siegfried Strathmann, Gisela Lorenz, Reinhard Stierl
Patent number: 6586369
Abstract: Agrochemical compositions having fungicidal action and comprising as active compounds compounds of the formula I
where
R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-haloalkylcarbonyl;
R2 is halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halo-C1-C6-alkylsulfonyl, cyano or a radical NR13R14;
R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halo-C1-C6-alkyl, C1-C6-alkoxy, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halo-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which may be unsubstituted or substituted by halogen, C1-C6-alkyl or halo-C1-C6-alkyl,
R13 is hydrogen, C1-C6-alkyl,
R14 is C1-C6-alkyl, C1-C8-cycloalkyl or, together with R13 and the nitrogen atom to which they are attached, a saturated or unsaturated heterocyclic five- or six-membered ring which contains one or two heteroatoms selected from the group co
Type:
Grant
Filed:
August 20, 2002
Date of Patent:
July 1, 2003
Assignee:
BASF Aktiengesellschaft
Inventors:
Joachim Rheinheimer, Karl Eicken, Ingo Rose, Thomas Grote, Eberhard Ammermann, John-Bryan Speakman, Siegfried Strathmann, Gisela Lorenz
Patent number: 6576595
Abstract: Xanthone derivatives of the formula I
where the index and the variables are as defined below:
n is 0, 1 or 2;
R1 is alkyl or haloalkyl;
R2,R3 are alkoxy, alkenyloxy or alkynyloxy, or R2 and R3 together form an unsubstituted or substituted oxyalkyleneoxy group;
R4 is halogen, cyano, hydroxyl, amino, mercapto, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylcarbonyloxy or alkylcarbonylthio;
R5 is a group R4, where the groups R5 may be different if n=2;
X, Y are oxygen or sulfur;
Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.
Type:
Grant
Filed:
September 23, 2002
Date of Patent:
June 10, 2003
Assignee:
BASF Aktiengesellschaft
Inventors:
Ingo Rose, Jordi Tormo i Blasco, Markus Gewehr, Wassilios Grammenos, Bernd Müller, Joachim Rheinheimer, Peter Schäfer, Frank Schieweck, Thomas Grote, Andreas Gypser, Eberhard Ammermann, Gisela Lorenz, Reinhard Stierl, Siegfried Strathmann
Patent number: 6569875
Abstract: Fungicidal mixtures comprise as active components
a) an amide compound of the formula I
A—CO—NR1R2 I
in which
A is an aryl group or an aromatic or nonaromatic, 5- or 6-membered heterocycle which has from 1 to 3 hetero atoms selected from O, N and S; where the aryl group or the heterocycle may or may not have 1, 2 or 3 substituents which are selected, independently of one another, from alkyl, halogen, CHF2, CF3, alkoxy, haloalkoxy, alkylthio, alkylsulfynyl and alkylsulfonyl;
R1 is a hydrogen atom;
R2 is a phenyl or cycloalkyl group which may or may not have 1, 2 or 3 substituents which are selected, independently of one another, from alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkyl, cycloalkenyl, cycloalkyloxy, cycloalkenyloxy, phenyl and halogen, where the aliphatic and cycloaliphatic radicals may be partially or fully halogenated and/or the cycloaliphatic radicals may be substituted by from 1 to 3 alkyl groups and where the phenyl group may have from 1 to
Type:
Grant
Filed:
June 13, 2000
Date of Patent:
May 27, 2003
Assignee:
BASF Aktiengesellschaft
Inventors:
Klaus Schelberger, Maria Scherer, Karl Eicken, Manfred Hampel, Eberhard Ammermann, Gisela Lorenz, Siegfried Strathmann
Patent number: 6562833
Abstract: 2-(N-phenylamino)pyrimidines of the formula I,
where:
R1, R3 independently of one another are cyano, C1-C8-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, where the radicals alkyl, alkenyl and alkynyl may be substituted by cyano, halogen, C1-C4-alkoxy or C1-C4-alkoxycarbonyl, or are C3-C8-cycloalkyl or a group C(═NORx)Ry
R2 is halogen, C1-C8-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, where the radicals alkyl, alkenyl and alkynyl may be substituted by cyano, halogen, C1-C4-alkoxy or C1-C4-alkoxycarbonyl, or
R1 and R2 together with the two linking carbon atoms form a fused-on partially unsaturated 4- to 8-membered ring which may be up to trisubstituted by identical or different substituents selected from the group consisting of C1-C4-alkyl, halogen and C1-C4-alkoxy-carbonyl, which may contain a carbonyl group and/or, in addition to the multiple bond of the pyrimidine ring, a double bond and/or which may be interrupted by O, S or N—(C1-C4-alkyl);
the substituents R4 to R8, Rx, Ry, Ra and Rb are
Type:
Grant
Filed:
December 5, 2000
Date of Patent:
May 13, 2003
Assignee:
BASF Aktiengesellschaft
Inventors:
Bernd Müller, Hubert Sauter, Herbert Bayer, Oliver Cullmann, Markus Gewehr, Wassilios Grammenos, Andreas Gypser, Arne Ptock, Norbert Götz, Thomas Grote, Michael Rack, Eberhard Ammermann, Gisela Lorenz, Siegfried Strathmann, John-Bryan Speakman
Patent number: 6559151
Abstract: 6-(2-Trifluoromethyl-phenyl)-triazolopyrimidines of formula I
in which
R1 and R2 independently denote hydrogen or
alkyl, alkenyl, alkynyl, alkadienyl, or haloalkyl,
cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or
5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or
where R1 and R2 radicals may be unsubstituted or substituted as defined in the specification; or
R1 and R2 together with the interjacent nitrogen atom represents a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted as defined in the specification;
R3 is hydrogen, halogen, alkyl, alkoxy and haloalkyl; and
X is halogen;
processes and intermediates for preparing these compounds, compositions comprising them a
Type:
Grant
Filed:
December 12, 2000
Date of Patent:
May 6, 2003
Assignee:
BASF Aktiengesellschaft
Inventors:
Klaus Jüergen Pees, Frank Schieweck, Jordi Tormo I Blasco, Hubert Sauter, Oliver Cullman, Bernd Müller, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Ingo Rose, Peter Schäfer, Eberhard Ammermann, Siegried Strathmann, Gisela Lorenz, Rheinhard Stierl