Patents by Inventor Guido Kurz

Guido Kurz has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Imidazo [2, 1-B] [1, 3, 4] Thiadiazole Derivatives
    Publication number: 20120094996
    Abstract: There is provided compounds of formula (I): wherein R1, R2 and R3 have meanings given in the description, and pharmaceutically-acceptable esters, amides, solvates or salts thereof, which compounds are useful in the treatment of diseases in which inhibition of a protein or lipid kinase (e.g. PI3-K, particularly class I PI3K) is desired and/or required, and particularly in the treatment of cancer.
    Type: Application
    Filed: April 1, 2010
    Publication date: April 19, 2012
    Applicant: Centro Nacional de Investigaciones Oncologicas (CNIO)
    Inventors: Joaquin Pastor Fernández, Guido Kurz, Sonia Martinez Gonzalez
  • INHIBITORS OF 11-BETA-HYDROXY STERIOD DEHYDROGENASE TYPE 1
    Publication number: 20100113435
    Abstract: The present invention relates to compounds with the formula (II) and also to pharmaceutical compositions comprising the compounds, to processes for their preparation, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-?-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Application
    Filed: November 16, 2009
    Publication date: May 6, 2010
    Inventors: Tjeerd BARF, Rikard Emond, Guido Kurz, Jerk Vallgarda, Marianne Nilsson
  • Inhibitors of 11-?-hydroxy steroid dehydrogenase type 1
    Patent number: 7671051
    Abstract: The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-?-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Grant
    Filed: July 13, 2005
    Date of Patent: March 2, 2010
    Assignee: Biovitrum AB
    Inventors: Tjeerd Barf, Rikard Emond, Jerk Vallgarda, Guido Kurz, Marianne Nilsson, Lian Zhang
  • Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
    Patent number: 7618961
    Abstract: The present invention relates to compounds with the formula (II) and also to pharmaceutical compositions comprising the compounds, to processes for their preparation, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-?-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Grant
    Filed: May 22, 2001
    Date of Patent: November 17, 2009
    Assignee: Biovitrum AB
    Inventors: Tjeerd Barf, Rikard Emond, Guido Kurz, Jerk Vallgårda, Marianne Nilsson
  • Use of thiazole derivatives and analogues in the treatment of cancer
    Publication number: 20090156644
    Abstract: There is provided a use of a compound of formula (I), wherein X, Y, T, W, A1, A2R1, R5 and R6 have meanings given in the description for the manufacture of a medicament for the treatment of cancer.
    Type: Application
    Filed: July 21, 2006
    Publication date: June 18, 2009
    Inventors: Jacob Westman, Guido Kurz, Bjorn Eriksson, Christian Hedberg
  • Use of thiazole derivatives and analogues in disorders caused by free fatty acids
    Publication number: 20090136472
    Abstract: There is provided a use of a compound of formula I, wherein X, T, Y, W, A1, A2, R1, R5 and R6 have meanings given in the description, for the manufacture of a medicament for the treatment of a disorder or condition caused by, linked to, or contributed to by, free fatty acids, such as hyperinsulinemia and associated conditions, including type 2 diabetes and the like.
    Type: Application
    Filed: July 21, 2006
    Publication date: May 28, 2009
    Inventors: Jacob Westman, Guido Kurz, Bjorn Eriksson, Christian Hdberg
  • Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
    Publication number: 20060287374
    Abstract: The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, to processes for their preparation, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-?-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Application
    Filed: August 29, 2006
    Publication date: December 21, 2006
    Inventors: Tjeerd Barf, Marianne Nilsson, Jerk Vallgarda, Guido Kurz
  • Inhibitors of 11-?-hydroxy steroid dehydrogenase type 1
    Patent number: 7132436
    Abstract: The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, to processes for their preparation, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-?-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Grant
    Filed: May 22, 2001
    Date of Patent: November 7, 2006
    Assignee: Biovitrum AB
    Inventors: Guido Kurz, Marianne Nilsson
  • Inhibitors of 11-?-hydroxy steroid dehydrogenase type 1
    Patent number: 7125900
    Abstract: The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, to processes for their preparation, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-?-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Grant
    Filed: May 22, 2001
    Date of Patent: October 24, 2006
    Assignee: Biovitrum AB
    Inventors: Tjeerd Barf, Marianne Nilsson, Jerk Vallgårda, Guido Kurz
  • Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
    Patent number: 7094792
    Abstract: The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-?-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Grant
    Filed: November 22, 2002
    Date of Patent: August 22, 2006
    Assignee: Biovitrum AB
    Inventors: Tjeerd Barf, Rikard Emond, Guido Kurz, Marianne Nilsson, Jerk Vallgårda, Lian Zhang
  • Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
    Patent number: 7074788
    Abstract: The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-?-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Grant
    Filed: November 22, 2002
    Date of Patent: July 11, 2006
    Assignee: Biovitrum AB
    Inventors: Guido Kurz, Marianne Nilsson, Jerk Vallgårda, Meredith Williams
  • Inhibitors of 11-beta-hydroxy steriod dehydrogenase type 1
    Publication number: 20050250776
    Abstract: The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-?-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Application
    Filed: July 13, 2005
    Publication date: November 10, 2005
    Inventors: Tjeerd Barf, Rikard Emond, Guido Kurz, Marianne Nilsson, Jerk Vallgarda, Lian Zhang
  • New compounds
    Publication number: 20050239853
    Abstract: The present invention relates to compounds with the formula (I) wherein R1, R2, R3, X, and Y are as defined herein, and also to pharmaceutical compositions comprising the compounds, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Application
    Filed: February 3, 2005
    Publication date: October 27, 2005
    Inventors: Tjeerd Barf, Guido Kurz, Sofia Nordin, Lars Tedenborg, Jerk Vallgarda, Meredith Williams
  • Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
    Publication number: 20040224996
    Abstract: The present invention relates to compounds with the formula (II) and also to pharmaceutical compositions comprising the compounds, to processes for their preparation, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-&bgr;-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Application
    Filed: February 18, 2003
    Publication date: November 11, 2004
    Inventors: Tjeerd Barf, Rikard Emond, Guido Kurz, Jerk Vallgarda, Marianne Nilsson
  • Method for producing a milling disc and milling disc produced according to the inventive method
    Patent number: 6723277
    Abstract: A method for producing a milling disc with embedded insets of hard metal, ceramics or other similar hard materials. The milling disc has a centrical bore in the base body of the disc. The tips of the insets protrude over the circumference of the disc body. The invention also relates to a milling disc produced according to the method wherein a powdery sintered metal material is filled into the recess of a mold pertaining to a compression molding die, and the mold matches the outer contour of the disc base body. Pre-fabricated insets are inserted into the sintered metal material and are positioned in the mold of the compression molding die. A green compact is subsequently pressed in the compression molding die and then taken out of the compression molding die. The green compact is sintered with the pressed insets and is subjected to hardening and/or surface treatment, if required.
    Type: Grant
    Filed: March 21, 2002
    Date of Patent: April 20, 2004
    Assignee: Karl Simon GmbH & Co. KG
    Inventors: Guido Kurz, Herbert König, Thomas Broghammer
  • Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
    Publication number: 20030176476
    Abstract: The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, to processes for their preparation, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-&bgr;-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Application
    Filed: February 18, 2003
    Publication date: September 18, 2003
    Inventors: Tjeerd Barf, Marianne Nilsson, Jerk Vallgarda, Guido Kurz
  • Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
    Publication number: 20030166689
    Abstract: The present invention relates to compounds with the formula (I) and also to pharmaceutical compositions comprising the compounds, to processes for their preparation, as well as to the use of the compounds in medicine and for the preparation of a medicament which acts on the human 11-&bgr;-hydroxysteroid dehydrogenase type 1 enzyme.
    Type: Application
    Filed: April 1, 2003
    Publication date: September 4, 2003
    Inventors: Guido Kurz, Marianne Nilsson
  • Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
    Publication number: 20030130318
    Abstract: The present invention relates to compounds with the formula (I) 1
    Type: Application
    Filed: November 22, 2002
    Publication date: July 10, 2003
    Inventors: Tjeerd Barf, Rikard Emond, Guido Kurz, Marianne Nilsson, Jerk Vallgarda, Lian Zhang
  • Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
    Publication number: 20030130258
    Abstract: The present invention relates to compounds with the formula (I) 1
    Type: Application
    Filed: November 22, 2002
    Publication date: July 10, 2003
    Inventors: Guido Kurz, Marianne Nilsson, Jerk Vallgarda, Meredith Williams
  • Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
    Publication number: 20030130279
    Abstract: The present invention relates to compounds with the formula (I) 1
    Type: Application
    Filed: November 22, 2002
    Publication date: July 10, 2003
    Inventors: Guido Kurz, Marianne Nilsson, Jerk Vallgarda, Meredith Williams