Patents by Inventor Helmut Heitzer

Helmut Heitzer has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 5708180
    Abstract: The reaction of cyanoolefins, aminocarbonylolefins or hydroxyiminoolefins with a Vilsmeier reagent leads to 2-halogenopyridines which bear aldehyde groups in the 3 and/or 5 position. These pyridinealdehydes are valuable intermediates for the preparation of pharmaceuticals and crop protection agents.
    Type: Grant
    Filed: November 27, 1996
    Date of Patent: January 13, 1998
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer
  • Patent number: 5258394
    Abstract: 1-Trifluoromethyl-1-nitro-2-alkoxy-2-aryl-ethanes of the formula ##STR1## in which R.sup.1 represents a straight-chain or branched alkyl radical andR.sup.2 represents an optionally substituted aryl or hetaryl radical,their preparation from an aldehyde of the formula R.sup.2 --CHO, an alcohol of the formula R.sup.1 --OH and trifluoromethylnitromethane in the presence of a compound containing basic groups and antimycotic agents containing these compounds.
    Type: Grant
    Filed: January 23, 1992
    Date of Patent: November 2, 1993
    Assignee: Bayer Aktiengesellschaft
    Inventors: Bernd Baasner, Gunther Beck, Helmut Heitzer, Klaus Schaller
  • Patent number: 5221681
    Abstract: The present invention relates to new substituted benzoxazepines and benzothiazepines of the general formula I ##STR1## in which X, R.sup.1, R.sup.2 and R.sup.3 have the meaning given in the description, processes for their preparation and their use in medicaments having vaso- and muscle-relaxing properties, in particular as circulatory agents.
    Type: Grant
    Filed: January 16, 1992
    Date of Patent: June 22, 1993
    Assignee: Bayer Aktiengesellschaft
    Inventors: Hans-Joachim Kabbe, Helmut Heitzer, Andreas Knorr, Claudia Hirth-Dietrich
  • Patent number: 5175336
    Abstract: The invention relates to new fluoromethylated polycyanobenzenes of the formula ##STR1## in which X represents hydrogen, fluorine or chlorine,m is 1 or 2 andn is (6-m),to a process for their preparation and to the salt-like alkali metal cyanide adducts of the fluoromethylated polycyanobenzenes formed as intermediates in this preparation process and to the use of the fluoromethylated polycyanobenzenes for the detection of anions.
    Type: Grant
    Filed: May 16, 1991
    Date of Patent: December 29, 1992
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Wolfgang von der Emden, Helmut Heitzer, Friedrich W. Krock, Ernst Kysela, Albrecht Marhold
  • Patent number: 5066681
    Abstract: 1-Trifluoromethyl-1-nitro-2-alkoxy-2-aryl-ethanes of the formula ##STR1## in which R.sup.1 represents a straight-chain or branched alkyl radical andR.sup.2 represents an optionally substituted aryl or hetaryl radical,their preparation from an aldehyde of the formula R.sup.2 -CHO, an alcohol of the formula R.sup.1 -OH and trifluoromethylnitromethane in the presence of a compound containing basic groups and antimycotic agents containing these compounds.
    Type: Grant
    Filed: September 20, 1989
    Date of Patent: November 19, 1991
    Assignee: Bayer Aktiengesellschaft
    Inventors: Bernd Baasner, Gunther Beck, Helmut Heitzer, Klaus Scaller
  • Patent number: 4748243
    Abstract: A process for the preparation of 2-chloro-5-chloromethyl-thiazole of the formula: ##STR1## comprising reacting allyl isothiocyanate of the formulaCH.sub.2 .dbd.CH--CH.sub.2 --NCSwith about 2 to 20 times its molar amount of chlorine at a temperature from above 0.degree. to 150.degree. C.
    Type: Grant
    Filed: August 31, 1987
    Date of Patent: May 31, 1988
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer
  • Patent number: 4369186
    Abstract: 4,5-Dichloroimidazole-2-carboxylic acid derivatives of the formula ##STR1## in which the group ##STR2## represents a carbon atom which has three bonds to hetero-atoms, and their salts with bases, possess insecticidal, acaricidal, fungicidal, nematicidal and herbicidal properties.
    Type: Grant
    Filed: May 17, 1979
    Date of Patent: January 18, 1983
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Klaus Sasse, Helmut Heitzer, Ludwig Eue, Robert R. Schmidt, Hans Scheinpflug, Ingeborg Hammann, Wilhelm Brandes
  • Patent number: 4350520
    Abstract: The imidazole-2-carboxylic acid amides of the general formula ##STR1## in which R represents alkyl, have powerful growth-regulating properties.The invention provides a method of regulating the growth of plants, which comprises applying to the plants, or to a habitat thereof, a compound of the formula (I) alone or in the form of a composition containing as active ingredient a compound of the formula (I) in admixture with a diluent or carrier.
    Type: Grant
    Filed: December 5, 1980
    Date of Patent: September 21, 1982
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer, Klaus Lurssen
  • Patent number: 4293331
    Abstract: Acyloxamide compounds of the formula ##STR1## in which R is chlorine, alkyl of from 1 or 2 carbon atoms or chloroalkyl of from 1 or 2 carbon atoms and 1 to 5 chlorine atomse.g., 2,2-dichloropropionyl-oxamide and trichloroacetyl-oxamide are outstandingly effective as plant growth regulants. spThis is a continuation of application Ser. No. 964,223 filed Nov. 27, 1978, abandoned.
    Type: Grant
    Filed: December 7, 1979
    Date of Patent: October 6, 1981
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer, Klaus Lurssen
  • Patent number: 4187306
    Abstract: The invention covers compounds of the formula ##STR1## in which R.sup.1 and R.sup.5 each represents 0, 1, 2, 3 or 4 of the following substituents: alkyl, hydroxyl, acyloxy, alkoxy, nitro, amino, alkylamino, dialkylamino, acylamino, acylalkylamino, alkoxycarbonylamino, halogen, trifluoromethyl, cyano, carboxyl, alkoxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, aminosulphonyl, alkylaminosulphonyl, dialkylaminoamino, R.sup.2 is hydrogen, optionally substituted alkyl, aralkyl or aryl or heterocyclo-alkyl, acyl or alkoxycarbonyl, and R.sup.3 and R.sup.4 are each hydrogen, or optionally substituted alkyl, aralkyl, aryl or hetero-aryl, are useful as medicaments which have an action on the central nervous system, in particular as, for example, tranquilizers and/or antiamnesics. Also included in the invention are methods for preparing said compounds, compositions containing them and methods for the use of said compounds and compositions.
    Type: Grant
    Filed: July 6, 1978
    Date of Patent: February 5, 1980
    Assignee: Bayer Aktiengesellschaft
    Inventors: Karl H. Mayer, Helmut Heitzer, Friedrich Hoffmeister, Arend Heise, Stanislav Kazda
  • Patent number: 4179277
    Abstract: 4,5-Dichloroimidazole-2-carboxylic acid derivatives of the formula ##STR1## in which the group ##STR2## represents a carbon atom which has three bonds to hetero-atoms, and their salts with bases,possess insecticidal, acaricidal, fungicidal, nematicidal and herbicidal properties.
    Type: Grant
    Filed: February 18, 1977
    Date of Patent: December 18, 1979
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Klaus Sasse, Helmut Heitzer, Ludwig Eue, Robert R. Schmidt, Hans Scheinpflug, Ingeborg Hammann, Wilhelm Brandes
  • Patent number: 4171442
    Abstract: Process for the preparation of 2,4,5-trichloropyrimidine, characterized in that compounds of the formula ##STR1## wherein R a radical which can be split off under the reaction conditions andR' an optionally substituted lower alkyl radical,Are reacted at temperatures from 0.degree. to 50.degree. C. with less than 7.5 mols of chlorine, in particular 3.5 to 7.0 mols of chlorine, and the reaction products are then after-heated to temperatures of 100.degree.-150.degree. C., in particular 110.degree.-140.degree. C., in the absence of chlorine.
    Type: Grant
    Filed: June 6, 1978
    Date of Patent: October 16, 1979
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer
  • Patent number: 4140857
    Abstract: Process for the preparation of 2,4,5-trichloropyrimidine, characterized in that compounds of the formula ##STR1## wherein R = a radical which can be split off under the reaction conditionsAre reacted with more than 7 and less than 13 mols of chlorine, in particular 11 mols of chlorine, at temperatures from 0 - 40.degree. C. and the reaction mixture is then subsequently heated in the absence of chlorine to temperatures from about 100 - 150.degree. C., in particular 110 - 140.degree. C.
    Type: Grant
    Filed: January 11, 1978
    Date of Patent: February 20, 1979
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer
  • Patent number: 4125722
    Abstract: Process for the preparation of tetrachloropyrimidine, characterized in that compounds of the formula ##STR1## wherein R = a radical which can be split off under the reaction conditions,Are reacted with chlorine or agents which release chlorine, preferably at temperatures from 0.degree.-150.degree. C and using more than 7 mols of chlorine, in particular using 11-13 mols of chlorine.
    Type: Grant
    Filed: October 17, 1977
    Date of Patent: November 14, 1978
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer
  • Patent number: 4125723
    Abstract: Process for the preparation of tetrachloropyrimidine, characterized in that compounds of the formula ##STR1## wherein R = a radical which can be split off under the reaction conditions andR' = optionally substituted lower allyl radical, are reacted with chlorine or agents which release chlorine, preferably at temperatures from 0.degree. to 150.degree. C and using more than 7.5 mols of chlorine, preferably 8 to 9 mols of chlorine.
    Type: Grant
    Filed: November 14, 1977
    Date of Patent: November 14, 1978
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer
  • Patent number: 4067721
    Abstract: New imidazolidinedione compounds of the formula ##STR1## in which R is chlorine, alkyl of 1 or 2 carbon atoms or chloroalkyl of 1 or 2 carbon atoms and 1 to 5 chlorine atomsAre outstandingly effective as plant growth regulants and have surprisingly been found to exhibit substantially greater activity than conventional materials of this type.
    Type: Grant
    Filed: October 20, 1976
    Date of Patent: January 10, 1978
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer, Klaus Lurssen
  • Patent number: 4021443
    Abstract: Perchlorodiazafulvene having the formula ##STR1## IS PREPARED BY REACTING 2,4,5-TRICHLORO-2-TRICHLOROMETHYL-2H-imidazole having the formula ##STR2## WITH DECHLORINATING AGENTS AT ELEVATED TEMPERATURES AND IS USEFUL AS A FUNGICIDE.
    Type: Grant
    Filed: October 29, 1975
    Date of Patent: May 3, 1977
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Fritz Doring, Helmut Heitzer, Hans Holtschmidt
  • Patent number: 4013674
    Abstract: The new compound N-(1,2,2,2-tetrachloroethyl)-formimide chloride of the formula ##STR1## is produced by reacting a substituted formamide of the formula ##STR2## wherein X is OH or Cl,With approximately the stoichiometrically required amount of a highly reactive inorganic acid chloride, e.g. phosphorus pentachloride. The compound (I) can be reacted with sulfur at about 150.degree. to 250.degree. C to produce trichlorothiazole of the formula ##STR3## which is known to have insecticidal activity.
    Type: Grant
    Filed: December 9, 1975
    Date of Patent: March 22, 1977
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer
  • Patent number: 3994913
    Abstract: 2,5-Dichloro-thiazolo[4,5-d]thiazole, which is useful as a fungicide, is prepared by reacting compounds having the formula ##EQU1## wherein X.sub.1 is Cl, andX.sub.2 is H or Cl orX.sub.1 and X.sub.2 together form a C-C bondIn the temperature range of 150.degree. to 300.degree. C, with at least the stoichiometrically required amount of sulphur.
    Type: Grant
    Filed: October 28, 1975
    Date of Patent: November 30, 1976
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gunther Beck, Helmut Heitzer, Hans Holtschmidt