Patents by Inventor Hermann Rempfler

Hermann Rempfler has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 5998636
    Abstract: Substituted N-phenyl- and N-heteroarylalkylcarbamates of the formula I ##STR1## in which Q is a group ##STR2## R is halogen, trifluoromethyl, cyano, nitro or C.sub.1 -C.sub.3 haloalkoxy;Z is hydrogen or halogen; orZ and R together in the 2- and 3-position of the phenyl ring form a group --OCF.sub.2 O--;R.sub.1 is C.sub.1 -C.sub.5 alkyl;R.sub.2, R.sub.3, R.sub.4 and R.sub.5, independently of one another, are hydrogen, methyl or ethyl;X is oxygen, sulfur, --SO-- or --SO.sub.2 --;Y is hydrogen, halogen, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy or cyano;n is 0, 1 or 2;n.sub.1 is 0 or 1; andm is 0 or 1,with the proviso that m is 1 if Q is group (1) or (2);and the diastereomers and enantiomers thereof,exhibit pre- and post-emergence herbicidal properties. The preparation of these compounds and their use as herbicidally active ingredients are described.
    Type: Grant
    Filed: August 4, 1998
    Date of Patent: December 7, 1999
    Assignee: Novartis Finance Corporation
    Inventors: Hermann Rempfler, Fredrik Cederbaum, Felix Spindler, Willy Urs Lottenbach
  • Patent number: 5831114
    Abstract: Substituted N-phenyl- and N-heteroarylalkylcarbamates of formula (I), in which Q is a group (1), (2) or (3); R is halogen, trifluoromethyl, cyano, nitro or C.sub.1 -C.sub.3 haloalkoxy; Z is hydrogen or halogen; or Z and R together in the 2- and 3-position of the phenyl ring form a group --OCF.sub.2 O--; R.sub.1 is C.sub.1 -C.sub.5 alkyl; R.sub.2, R.sub.3, R.sub.4 and R.sub.5, independently of one another, are hydrogen, methyl or ethyl; X is oxygen, sulfur, --SO-- or --SO.sub.2 --, Y is hydrogen, halogen, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy or cyano; n is 0, 1 or 2; n.sub.1 is 0 or 1; and m is 0 or 1, with the proviso that m is 1 if Q is group (1) or (2); and the diastereomers and enantiomers thereof, exhibit pre- and post-emergence herbicidal properties. The preparation of these compounds and their use as herbicidally active ingredients are described.
    Type: Grant
    Filed: May 28, 1997
    Date of Patent: November 3, 1998
    Assignee: Novartis Finance Corporation
    Inventors: Hermann Rempfler, Fredrik Cederbaum, Felix Spindler, Willy Urs Lottenbach
  • Patent number: 5500407
    Abstract: Triazolo pyrimidines of the formula ##STR1## wherein R.sub.1 is hydrogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 haloalkyl; and R.sub.2 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 haloalkylthio, C.sub.1 -C.sub.4 alkoxy-C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 -alkoxy-C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkoxy-C.sub.1 -C.sub.4 alkylthio, halogen, amino, C.sub.1 -C.sub.4 alkylamino or C.sub.1 -C.sub.4 dialkylamino, have pre- and postemergence herbicidal properties. Their preparation use thereof as herbicides are described.
    Type: Grant
    Filed: November 21, 1994
    Date of Patent: March 19, 1996
    Assignee: Ciba-Geigy Corporation
    Inventor: Hermann Rempfler
  • Patent number: 5399545
    Abstract: Substituted benzyl carbamates of formula I ##STR1## wherein R is halogen, trifluoromethyl, cyano, nitro or C.sub.1 -C.sub.3 haloalkoxy;Z is hydrogen or halogen; orZ and R together in 2- and 3-position of the phenyl ring form the group --OCF.sub.2 O--;R.sub.1 is C.sub.1 -C.sub.5 alkyl; wherein in caseR and Z together in 2- and 3-position of the phenyl ring form the group --OCF.sub.2 --,R.sub.2 and R.sub.3 are each independently of the other hydrogen, methyl or ethyl; and in case R is halogen, trifluoromethyl, cyano, nitro or C.sub.1 -C.sub.3 haloalkoxy,R.sub.2 is methyl or ethyl; and R.sub.3 is hydrogen, methyl or ethyl;X is oxygen, sulfur, --SO-- or --SO.sub.2 --;Y is hydrogen, halogen, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy or cyano; andn is 0, 1 or 2;and the diastereoisomers thereof, have pre- and postemergence herbicidal properties. The preparation of these compounds and the use thereof as herbicides are described.
    Type: Grant
    Filed: October 22, 1993
    Date of Patent: March 21, 1995
    Assignee: Ciba-Geigy Corporation
    Inventor: Hermann Rempfler
  • Patent number: 5312800
    Abstract: Pyrrolidinones of formula I ##STR1## wherein R is hydrogen, C.sub.1 -C.sub.4 alkyl, or phenyl unsubstituted or substituted by halogen, C.sub.1 -C.sub.4 alkyl or by C.sub.1 -C.sub.4 haloalkyl, or is fluorine, chlorine or bromine;R.sub.0 is hydrogen or halogen;R.sub.1 and R.sub.2 independently of one another are hydrogen or C.sub.1 -C.sub.4 alkyl;X is hydrogen, flourine, chlorine, bromine, cyano, --COOR.sub.1, --CONR.sub.1 R.sub.2, --NH.sub.2 or --NHCOR.sub.3, wherein R.sub.1 and R.sub.2 are as defined, and R.sub.3 is C.sub.1 -C.sub.4 alkyl; andY is hydrogen, chlorine or bromine; andthe diastereoisomeric forms thereof, exhibit pre- and post-emergence herbicidal properties. The preparation of those compounds and their use as herbicidal active ingredients are described.
    Type: Grant
    Filed: May 20, 1993
    Date of Patent: May 17, 1994
    Assignee: Ciba-Geigy Corporation
    Inventor: Hermann Rempfler
  • Patent number: 5159078
    Abstract: The present invention relates to novel N-phenyl-N-pyrimidin-2-ylureas having a herbicidal and plant growth-regulating activity, to agrochemical compositions containing those substances as active ingredients, to the use of the novel ureas for controlling weeds or for regulating plant growth, and to processes for the preparation of the novel compounds. The invention also relates to novel intermediates and to processes for the preparation thereof.The novel compounds correspond to formula I ##STR1## in which R.sup.1, R.sup.2 and R.sup.3 are each, independently of the others, hydrogen; halogen; C.sub.1 -C.sub.4 alkyl; C.sub.1 -C.sub.4 alkoxy; C.sub.1 -C.sub.4 haloalkyl; C.sub.1 -C.sub.4 haloalkoxy; C.sub.1 -C.sub.4 alkyl-S(O).sub.n -; nitro; cyano; C.sub.1 -C.sub.4 alkoxycarbonyl; C.sub.1 -C.sub.4 alkylcarbonyl; di-(C.sub.1 -C.sub.4 alkylamino)-carbonyl; mono-(C.sub.1 -C.sub.4 alkylamino)carbonyl; carbamoyl; C.sub.1 -C.sub.4 -haloalkyl-S(O).sub.n -; or -PO[O-(C.sub.1 -C.sub.4)-alkyl].sub.2 ;R.sup.4 is C.sub.1 -C.
    Type: Grant
    Filed: August 17, 1990
    Date of Patent: October 27, 1992
    Assignee: Ciba-Geigy Corporation
    Inventors: Hermann Rempfler, Dieter Durr, Rudolf C. Thummel
  • Patent number: 5154751
    Abstract: The invention relates to novel compositions having herbicidal and plant growth regulating properties and containing, as active ingredient, a compound of formula I ##STR1## wherein R.sub.1 to R.sub.6 are as defined in the description, to novel compounds of formula I and intermediates, and to the preparation thereof.
    Type: Grant
    Filed: May 30, 1990
    Date of Patent: October 13, 1992
    Assignee: Ciba-Geigy Corporation
    Inventor: Hermann Rempfler
  • Patent number: 5002604
    Abstract: There are described novel 2-[4-(5-chloro-3-fluoropyridin-2-yloxy)-phenoxy]-propionic acids esters and -thio-esters having a herbicidal action and an action reducing the growth of grasses, which compounds correspond to the formula I ##STR1## wherein Q is oxygen or sulfur,R.sub.1 is hydrogen or methylR.sub.2 is hydrogen or C.sub.1 -C.sub.4 alkylThe salts and enantiomers of these compounds are also part of the invention.These compounds are suitable for selectively controlling weeds in crops of cultivated plants, and for reducing the growth of grasses.
    Type: Grant
    Filed: December 16, 1988
    Date of Patent: March 26, 1991
    Assignee: Ciba-Geigy Corporation
    Inventors: Rolf Schurter, Hermann Rempfler
  • Patent number: 4999046
    Abstract: The present invention relates to novel N-(2-nitrophenyl)-N-pyrimidin-2-ylureas having a herbicidal and plant growth-regulating activity, to agrochemical compositions containing those substances as active ingredients, to the use of the novel ureas for controlling weeds or for regulating plant growth, and to processes for the preparation of the novel compounds. The invention also relates to novel intermediates and to processes for the preparation thereof.The novel compounds correspond to formula I ##STR1## in which R.sup.1 is hydrogen, methyl, fluorine, chlorine or bromine,R.sup.2 is C.sub.1 -C.sub.2 haloalkyl having at least 2 fluorine atoms, andR.sup.3 is C.sub.1 -C.sub.4 alkyl,with the proviso that R.sup.2 is not trifluoromethyl when R.sup.3 is methyl.
    Type: Grant
    Filed: April 5, 1989
    Date of Patent: March 12, 1991
    Assignee: Ciba-Geigy Corporation
    Inventor: Hermann Rempfler
  • Patent number: 4973690
    Abstract: The present invention relates to novel N-phenyl-N-pyrimidin-2-ylureas having a herbicidal and plant growth-regulating activity, to agrochemical compositions that contain those substances as active ingredients, to the use of the novel ureas for controlling weeds or for regulating plant growth, and to processes for the preparation of the novel compounds. The invention also relates to novel intermediates and to processes for the preparation thereof.The novel compounds correspond to formula I ##STR1## in which the radicals R.sup.1 to R.sup.6 have the meanings given in the text.
    Type: Grant
    Filed: April 3, 1989
    Date of Patent: November 27, 1990
    Assignee: Ciba-Geigy Corporation
    Inventors: Hermann Rempfler, Dieter Durr
  • Patent number: 4966622
    Abstract: The present invention relates to novel N-phenyl-N-pyrimidin-2-ylureas having a herbicidal and plant growth-regulating activity, to agrochemical compositions containing those substances as active ingredients, to the use of the novel ureas for controlling weeds or for regulating plant growth, and to processes for the preparation of the novel compounds. The invention also relates to novel intermediates and to processes for the preparation thereof.The novel compounds correspond to formula I ##STR1## in which R.sup.1, R.sup.2 and R.sup.3 are each, independently of the others, hydrogen; halogen; C.sub.1 -C.sub.4 alkyl; C.sub.1 -C.sub.4 alkoxy; C.sub.1 -C.sub.4 haloalkyl; C.sub.1 -C.sub.4 haloalkoxy; C.sub.1 -C.sub.4 alkyl-S(O).sub.n -; nitro; cyano; C.sub.1 -C.sub.4 alkoxycarbonyl; C.sub.1 -C.sub.4 alkylcarbonyl; di-(C.sub.1 -C.sub.4 alkylamino)-carbonyl; mono-(C.sub.1 -C.sub.4 alkylamino)carbonyl; carbamoyl; C.sub.1 -C.sub.4 haloalkyl-S(O).sub.n -; or -PO[O-(C.sub.1 -C.sub.4)-alkyl].sub.2 ;R.sup.4 is C.sub.1 -C.
    Type: Grant
    Filed: April 3, 1989
    Date of Patent: October 30, 1990
    Assignee: Ciba-Geigy Corporation
    Inventors: Hermann Rempfler, Dieter Durr, Rudolf C. Thummel
  • Patent number: 4940481
    Abstract: The invention relates to azolylpropane derivatives of the general formula I ##STR1## wherein R.sub.1 is an azolyl group,R.sub.2 and R.sub.3, each independently of the other, is hydrogen, alkyl, alkenyl, alkynyl, aralkyl, cyanoalkyl or alkoxycarbonylalkyl, and one of R.sub.2 and R.sub.3 always has a meaning other than hydrogen,R.sub.4 is C.sub.3 -C.sub.8 cycloalkyl, unsubstituted or substituted by alkyl; unsubstituted or substituted phenyl; or is C.sub.1 -C.sub.10 alkyl, unsubstituted or substituted by phenyl or substituted phenyl,R.sub.5 is an unsubstituted or a mono- or polysubstituted radical selected from the group consisting of C.sub.1 -C.sub.8 alky, C.sub.3 -C.sub.8 cycloalkyl, C.sub.3 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl, phenyl, naphthyl, biphenyl, benzylphenyl, benzyloxyphenyl, phenoxyphenyl and aralkyl,R.sub.
    Type: Grant
    Filed: February 22, 1983
    Date of Patent: July 10, 1990
    Assignee: Ciba-Geigy Corporation
    Inventors: Urs Muller, Hans Tobler, Hermann Rempfler, Alfred Meyer
  • Patent number: 4935051
    Abstract: There is described the novel 2-[4-(5-Chloro-3-fluoropyridin-2-yloxy)-phenoxy]-propionic acid methyl ester and its (R)-enantiomer. ##STR1## These compounds are suitable for selectively controlling weeds in crops of cultivated plants, and for reducing the growth of grasses.
    Type: Grant
    Filed: May 2, 1986
    Date of Patent: June 19, 1990
    Assignee: Ciba-Geigy Corporation
    Inventors: Rolf Schurter, Hermann Rempfler
  • Patent number: 4904778
    Abstract: The invention relates to ureas having a herbicidal and plant growth-regulating action of the formula ##STR1## in which R.sup.1 and R.sup.2 each represent, independently of the other, hydrogen, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkoxycarbonyl, C.sub.1 -C.sub.4 -alkoxy-(C.sub.1 -C.sub.4)-alkyl, nitro or cyano, andR.sup.3 and R.sup.4 each represents, independently of the other, hydrogen, halogen, cyano, OH, SH, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkylthio, amino, mono-C.sub.1 -C.sub.4 -alkylamino, di-C.sub.1 -C.sub.4 -alkylamino, C.sub.1 -C.sub.4 -alkoxycarbonyl or C.sub.1 -C.sub.4 -alkoxy-(C.sub.1 -C.sub.4)-alkyl,processes and intermediates for the preparation thereof, and herbicidal and plant growth-regulating compositions containing a compound of the formula I.
    Type: Grant
    Filed: October 24, 1988
    Date of Patent: February 27, 1990
    Assignee: Ciba-Geigy Corp.
    Inventors: Hermann Rempfler, Erich Stamm, Rudolph C. Thummel
  • Patent number: 4894083
    Abstract: The invention relates to a herbicidal and plant growth regulating composition which contains as active ingredient a 2-benzoyl-2-phenyloxirane of formula I ##STR1## wherein each of m and n independently of the other is 0, 1, 2 or 3 and each of R and R' independently of the other is a halogen atom, a C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkyl or C.sub.1 -C.sub.4 haloalkoxy group or the nitro or cyano group or a phenoxy group which is substituted by (R).sub.m, in the form of a racemate or an optically active enantiomer.Some oxiranes are known as intermediates for the preparation of fungicides and others are novel. The herbicidal composition has selective action in rice crops and is active against grasses.
    Type: Grant
    Filed: February 29, 1988
    Date of Patent: January 16, 1990
    Assignee: Ciba-Geigy Corporation
    Inventors: Hermann Rempfler, Walter Kunz
  • Patent number: 4849007
    Abstract: The invention relates to a herbicidal and plant growth regulating composition which contains as active ingredient a 2-benzoyl-2-phenyloxirane of formula I; ##STR1## wherein each of m and n independently of the other is 0, 1, 2 or 3 and each of R and R' independently of the other is a halogen atom, a C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkyl or C.sub.1 -C.sub.4 haloalkoxy group or the nitro or cyano group or a phenoxy group which is substituted by (R).sub.m, in the form of a racemate or an optically active enantiomer.Some oxiranes are known as intermediates for the preparation of fungicides and others are novel. The herbicidal composition has selective action in rice crops and is active against grasses.
    Type: Grant
    Filed: November 24, 1986
    Date of Patent: July 18, 1989
    Assignee: Ciba-Geigy Corporation
    Inventors: Hermann Rempfler, Walter Kunz
  • Patent number: 4831148
    Abstract: In accordance with a novel process, 2,3-difluoropyridines of formula I ##STR1## wherein X is halogen or trifluoromethyl, are prepared by diazotising a 3-amino-2-halopyridine of formula II ##STR2## wherein X is as defined for formula I and Y is bromine, chlorine or fluorine, in the presence of hydrogen fluroide, to give a 3-fluoro-2-halopyridine of formula III ##STR3## wherein X and Y are as defined for formula II, and treating resultant 3-fluoro-2-halopyridines of formula III, wherein Y is bromine or chlorine, with a fluorinating agent.The 2,3-difluoropyridines prepared by the novel process are valuable intermediates for the preparation of 2-[4-(3-fluoropyridin-2-yloxy)-phenoxy]propionic acid derivatives which are known as herbicides.
    Type: Grant
    Filed: October 4, 1985
    Date of Patent: May 16, 1989
    Assignee: Ciba-Geigy Corporation
    Inventors: Rolf Schurter, Urs Siegrist, Hermann Rempfler, Peter Baumeister
  • Patent number: 4802909
    Abstract: The invention relates to ureas having a herbicidal and plant growth-regulating action of the formula ##STR1## in which R.sup.1 and R.sup.2 each represents, independently of the other, hydrogen, halogen, C.sub.1 -C.sub.6 -alkyl C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkoxycarbonyl, C.sub.1 -C.sub.4 -alkoxy-(C.sub.1 -C.sub.4)-alkyl, nitro or cyano, andR.sup.3 and R.sup.4 each represents, independently of the other, hydrogen, halogen, cyano, OH, SH, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkylthio, amino, mono-C.sub.1 -C.sub.4 -alkylamino, di-C.sub.1 -C.sub.4 -alkylamino, C.sub.1 -C.sub.4 -alkoxycarbonyl or C.sub.1 -C.sub.4 -alkoxy-(C.sub.1 -C.sub.4)-alkyl,processes and intermediates for the preparation thereof, and herbicidal and plant growth-regulating compositions containing a compound of the formula I.
    Type: Grant
    Filed: October 9, 1987
    Date of Patent: February 7, 1989
    Assignee: Ciba-Geigy Corporation
    Inventors: Hermann Rempfler, Erich Stamm, Rudolph C. Thummel
  • Patent number: 4759796
    Abstract: 2-Phenoxypropionic acid cyanamides of the formula ##STR1## have a useful selective herbicidal activity against weeds, preferably grass weeds, in crops of useful plants.In this formulaR is hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.3 -C.sub.4 alkenyl, C.sub.3 -C.sub.4 alkynyl or C.sub.2 -C.sub.4 alkoxyalkyl, andT is a radical ##STR2## wherein A is oxygen or sulfur,X is fluorine, chlorine, bromine, iodine or trifluoromethyl,Y is hydrogen, fluorine, chlorine, bromine or trifluoromethyl, andZ is nitrogen or the methine bridge.
    Type: Grant
    Filed: October 16, 1986
    Date of Patent: July 26, 1988
    Assignee: Ciba-Geigy Corporation
    Inventors: Beat Bohner, Hermann Rempfler, Rolf Schurter
  • Patent number: 4758670
    Abstract: Fluoroazolylpropane derivatives of the formula I ##STR1## are described, in which Az is imidazolyl or triazolyl, R.sup.1 is hydrogen, alkyl or aralkyl which is unsubstituted or substituted by halogen, alkyl, alkoxy, halogenoalkyl, nitro, cyano, carboxyl or alkoxycarbonyl, R.sup.2 is C.sub.1 -C.sub.10 -alkyl which is unsubstituted or substituted by alkoxy, aralkoxy or phenyl, it being possible for the aromatic nuclei of aralkoxy and phenyl in turn to be unsubstituted or substituted by halogen, alkyl, alkoxy, halogenoalkyl, cyano, carboxyl or alkoxycarbonyl, R.sup.3 is hydrogen, alkyl, alkylcarbonyl or aralkyl which is unsubstituted or substituted by halogen, alkoxy, alkyl, halogenoalkyl, cyano, carboxyl or alkoxycarbonyl, R.sup.5 is an unsubstituted or monosubstituted or polysubstituted radical selected from the series comprising C.sub.1 -C.sub.8 -alkyl, C.sub.3 -C.sub.8 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.
    Type: Grant
    Filed: January 4, 1984
    Date of Patent: July 19, 1988
    Assignee: Ciba-Geigy Corporation
    Inventors: Urs Muller, Hermann Rempfler, Hans Tobler