Patents by Inventor Ikutaro Saji
Ikutaro Saji has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).
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Publication number: 20110183993Abstract: The present invention relates to a novel cycloalkane derivative which has an excellent psychotropic action.Type: ApplicationFiled: January 28, 2011Publication date: July 28, 2011Applicant: Dainippon Sumitomo Pharma Co., Ltd.Inventors: Ryu Nagata, Mayumi Oda, Norihiko Tanno, Masayuki Muto, Ikutaro Saji
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Patent number: 5780632Abstract: An imide compound of the formula: ##STR1## wherein Z is a group of the formula: ##STR2## in which B is a carbonyl group or a sulfonyl group, R.sup.1, R.sup.2, R.sup.3 and R.sup.4 are each a hydrogen atom or a lower alkyl group, or R.sup.1 and R.sup.2 or R.sup.1 and R.sup.3 may be combined together to make a non-aromatic hydrocarbon ring or R.sup.1 and R.sup.3 may be combined together to make an aromatic ring, said non-aromatic hydrocarbon ring being optionally bridged with a lower alkylene group or an oxygen atom therein and said aromatic ring, said non-aromatic hydrocarbon ring and said lower alkylene group being each optionally substituted with at least one lower alkyl, and n is an integer of 0 or 1;D is a group of the formula:--(CH.sub.2).sub.p --A--(CH.sub.2).sub.Type: GrantFiled: April 18, 1996Date of Patent: July 14, 1998Assignee: Sumitomo Pharmaceuticals Company, LimitedInventors: Ikutaro Saji, Masayuki Muto, Norihiko Tanno, Mayumi Yoshigi
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Patent number: 5532372Abstract: An imide compound of the formula: ##STR1## wherein Z is a group of the formula: ##STR2## in which the substituents are defined herein, and n is an integer of 0 to 1;D is a group of the formula:--(CH.sub.2).sub.p --A--(CH.sub.2).sub.q --in which A is a non-aromatic hydrocarbon ring optionally bridged with a lower alkylene group or an oxygen atom, said non-aromatic hydrocarbon ring and said lower alkylene group being each optionally substituted with at least one lower alkyl, and p and q are each an integer of 0, 1 or 2; andAr is an aromatic group, a heterocyclic aromatic group, a benzoyl group, a phenoxy group or a phenylthio group and G is >N--, >CH-- or >COH-- or Ar is a biphenylmethylidene group and G is >C.dbd., all of the above groups being each optionally substituted with at least one of lower alkyl, lower alkoxy and halogen; and its acid addition salts, useful as an antipsycotic agent.Type: GrantFiled: August 30, 1993Date of Patent: July 2, 1996Assignee: Sumitomo Pharmaceuticals Company, Ltd.Inventors: Ikutaro Saji, Masayuki Muto, Norihiko Tanno, Mayumi Yoshigi
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Patent number: 5258396Abstract: A novel thiazole derivative represented by the following general formula [1] and a pharmaceutically acceptable salt thereof: ##STR1## wherein A is a single bond, a straight-chained or branched lower alkylene group or a straight-chained or branched lower alkenylene group; B is a single bond or --CO--; R.sup.1 is a carboxy group or --CON(R.sup.7)OR.sup.8 (R.sup.7 and R.sup.8 are independently of each other a hydrogen atom or a lower alkyl group); R.sup.2 is a lower alkyl group; R.sup.3 and R.sup.4 are independently of each other a hydrogen atom, a lower alkyl group or a lower alkoxycarbonyl group; R.sup.5 is a hydrogen atom or a halogen atom; and R.sup.6 is a hydrogen atom, a halogen atom, a lower alkyl group, a hydroxy group, a lower alkoxy group, a thiol group, a lower alkylthio group, a lower alkylsulfinyl group, a lower alkylsulfonyl group, a nitro group, an amino group, a substituted amino group, a cyano group, a carboxy group or an acyl group.Type: GrantFiled: April 21, 1992Date of Patent: November 2, 1993Assignee: Sumitomo Pharmaceuticals Company, LimitedInventors: Hiroaki Masumori, Norihiko Tanno, Ikutaro Saji, Yoshihiko Kimura
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Patent number: 5081139Abstract: An N-substituted triazole compound of the formula: ##STR1## wherein Ph is a phenyl group or a phenyl group substituted with one or two halogen atoms, R.sup.1 is a C.sub.1 -C.sub.3 alkyl group, R.sup.2 is a hydrogen atom or a C.sub.1 -C.sub.3 alkyl group, R.sup.3 is a C.sub.1 -C.sub.8 alkyl group, a C.sub.4 -C.sub.8 cycloalkylalkyl group or a C.sub.3 -C.sub.6 cycloalkyl group and n is 0, 1 or 2, or an acid addition salt thereof, which is useful as an antifungal agent.Type: GrantFiled: October 2, 1985Date of Patent: January 14, 1992Assignee: Sumitomo Pharmaceuticals Company, LimitedInventors: Ikutaro Saji, Yoshihiro Tanaka, Katsuaki Ichise, Tomoharu Tanio, Takao Okuda, Toshio Atsumi
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Patent number: 4948799Abstract: An imide derivative of the formula: ##STR1## or a pharmaceutically acceptable salt, which is useful as an antipsychotic drug.Type: GrantFiled: January 4, 1989Date of Patent: August 14, 1990Assignee: Sumitomo Pharmaceuticals Company, LimitedInventors: Fujio Antoku, Mayumi Yoshigi, Ikutaro Saji, Atsuyuki Kojima, Kukuo Ishizumi
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Patent number: 4937249Abstract: A compound of the formula: ##STR1## or its acid addition salt, which is useful as a psychotic drug.Type: GrantFiled: October 25, 1988Date of Patent: June 26, 1990Assignee: Sumitomo Pharmaceuticals Company, LimitedInventors: Fujio Antoku, Mayumi Yoshigi, Ikutaro Saji, Kikuo Ishizumi
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Patent number: 4812461Abstract: An imide derivative of the formula: ##STR1## or a pharmaceutically acceptable salt, which is useful as an antipsychotic drug.Type: GrantFiled: September 25, 1987Date of Patent: March 14, 1989Assignee: Sumitomo Pharmaceuticals Company, LimitedInventors: Fujio Antoku, Mayumi Yoshigi, Ikutaro Saji, Atsuyuki Kojima, Kukuo Ishizumi
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Patent number: 4526983Abstract: An optically active imidazolylpropanol compound of the formula: ##STR1## wherein n is an integer of 3 or 4, and its acid addition salts, which is useful as an antifungal agent, prepared by reacting an imidazolylthiol of the formula: ##STR2## with an alkylating agent of the formula:CH.sub.3 --(CH.sub.2).sub.n --X (III)wherein n is as defined above and X is a halogen atom, an alkylsulfonyloxy group or an arylsulfonyloxy group.Type: GrantFiled: May 24, 1983Date of Patent: July 2, 1985Assignee: Sumitomo Chemical Company, LimitedInventors: Ikutaro Saji, Renzo Sato, Noritaka Hanma, Yasuo Motoike
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Patent number: 4461774Abstract: An imidazolylcarboxylic acid compound of the formula: ##STR1## wherein Ph is a phenyl group or a phenyl group substituted with one or two halogen atoms, R is a hydrogen atom or a C.sub.1 -C.sub.8 alkyl group and n is an integer of 1 to 8, which is useful as an antifungal agent.Type: GrantFiled: September 29, 1982Date of Patent: July 24, 1984Assignee: Sumitomo Chemical Company, LimitedInventors: Ikutaro Saji, Hiroshi Yamazaki, Shunji Aono, Katsuaki Ichise, Takao Okuda
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Patent number: 4288448Abstract: An N-substituted imidazole compound of the formula: ##STR1## wherein R and R' are independently a phenyl group optionally substituted with one or more halogen, C.sub.1 -C.sub.8 alkyl, C.sub.1 -C.sub.8 alkoxy, C.sub.1 -C.sub.8 alkylthio, phenyl, phenoxy, phenylthio, hydroxyl, trifluoromethyl, amino, carbamoyl, di(C.sub.1 -C.sub.8) alkylamino, C.sub.1 -C.sub.8 alkanoylamino, nitro, cyano, carboxy, C.sub.1 -C.sub.8 alkoxycarbonyl, C.sub.1 -C.sub.8 alkylsulfonyloxy or C.sub.1 -C.sub.8 alkanoylpiperazino groups; a C.sub.1 -C.sub.15 alkyl group or a phenyl (C.sub.1 -C.sub.2) alkyl group optionally bearing halogen on the benzene ring, and its acid-addition salts, which is useful as an antifungal agent.Type: GrantFiled: November 26, 1980Date of Patent: September 8, 1981Assignee: Sumitomo Chemical Company, LimitedInventors: Ikutaro Saji, Shunji Aono, Takao Okuda, Hideo Agui
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Patent number: 4216333Abstract: A process for preparing N-tritylimidazole compounds of the formula: ##STR1## by the reaction between a tritylcarbinol derivative of the formula: ##STR2## and an imidazole derivative of the formula: ##STR3## , characterized in that the reaction is effected in the presence of a phosphorus compound of the formula: ##STR4##Type: GrantFiled: January 30, 1979Date of Patent: August 5, 1980Assignee: Sumitomo Chemical Company, LimitedInventors: Hideo Agui, Ikutaro Saji, Mitsuo Nakashita