Patents by Inventor Jacques Bure

Jacques Bure has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Enantiomers derived from (S)-2-amino-2-(3,4-dichlorobenzyl)-1-propanol, their use and method of preparation
    Patent number: 5348980
    Abstract: Enantiomers of (S) configuration of formula (I) ##STR1## in which R is H or methyl, with antiallergic and in particular antihistaminic activity, useful as medicinal products.
    Type: Grant
    Filed: May 3, 1993
    Date of Patent: September 20, 1994
    Assignee: Institute de Recherche Jouveinal
    Inventors: Gilbert Aubard, Jacques Bure, Alain Calvet, Claude J. Gouret, Agnes Grouhel, Jean-Louis Junien
  • Aminoalcohols, their preparation process and their applications, particularly in therapeutics
    Patent number: 4994617
    Abstract: Aminoalcohols of formula: ##STR1## in which R.sub.1 is alkyl, R.sub.2 H or alkyl, R.sub.3 in particularly H, alkyl, phenylakyl, alkanoyl, phenylalkanoyl, in which N, R.sub.2 and R.sub.3 together form a heterocycle saturated with 5 to 7 chain links.Analgesic medicaments.
    Type: Grant
    Filed: December 26, 1989
    Date of Patent: February 19, 1991
    Assignee: Jouveinal S.A.
    Inventors: Gilbert Aubard, Jacques Bure, Alain P. Calvet, Claude Gouret, Agnes G. Grouhel, Jean-Louis Junien
  • Aminoethylimidazole and cytoprotective and gastric antisecretory composition containing the same
    Patent number: 4734428
    Abstract: Aminoethyl imidazole of formula: ##STR1## in which R.sub.1 is a lower alkyl, R.sub.2 is a phenyl or phenoxy radical, optionally substituted by a halogen atom or a lower alkoxy radical, R.sub.3,R.sub.4 and R.sub.5 are a hydrogen atom or a lower alkyl radical and x, y and z have the value 0 or 1, but the values of y and z cannot be the same, together with their acid addition salts with acids.Cytoprotective medicament.
    Type: Grant
    Filed: June 10, 1986
    Date of Patent: March 29, 1988
    Assignee: Jouveinal S.A.
    Inventors: Gilbert G. Aubard, Jacques Bure, Agnes G. Grouhel, Jean-Louis Junien, Veronique J. Lelievre, Xavier B. Pascaud, Claude P. Roux
  • Thieno[2,3-b] pyrrole compounds and analgesic use thereof
    Patent number: 4608384
    Abstract: New thieno[2,3-b] pyrrole compounds of the formula: ##STR1## in which: R.sub.1 is hydrogen or lower alkyl,R.sub.2 is cyano, carboxy, COOM in which M is alkali alkaline-earth metal, ammonium mono-, di-, or tri-, (C.sub.1 -C.sub.5) alkylammonium optionally substituted by hydroxy, COOR in which R is lower alkyl, or ##STR2## in which R' and R" are hydrogen or lower alkyl; R.sub.3 is lower alkyl; andR.sub.4 is lower alkyl, phenyl, halophenyl, lower alkylphenyl, lower alkoxy-phenyl nitrophenyl and di-lower-alkylamino,and enatiomers thereof.These new compounds may be used as medicines especially in the treatment of acute and chronic pains.
    Type: Grant
    Filed: December 12, 1983
    Date of Patent: August 26, 1986
    Assignee: Adir, S.A.R.L.
    Inventors: Michel Wierzbicki, Jacques Bure
  • Piperidyl phenyl trifluoroethanols
    Patent number: 4404215
    Abstract: This invention relates to novel arylethanol and to process for producing the said compounds.The arylethanols of the invention have valuable pharmacological properties and find a use in human or animal therapy.
    Type: Grant
    Filed: November 18, 1981
    Date of Patent: September 13, 1983
    Assignee: Science Union et Cie
    Inventors: Michel Vincent, Georges Remond, Jacques Bure
  • Thiosubstituted amino acids
    Patent number: 4315031
    Abstract: This invention relates to thiosubstituted cyclic amino acids, to a process for their preparation and to pharmaceutical compositions containing them together with an inert non toxic pharmaceutical carrier.
    Type: Grant
    Filed: August 28, 1978
    Date of Patent: February 9, 1982
    Assignee: Science Union et Cie
    Inventors: Michel Vincent, Georges Remond, Jacques Bure
  • Monosubstituted piperazines
    Patent number: 4312869
    Abstract: Biphenylalkylene-thiazolyl-piperazines of the formula ##STR1## wherein Ar and A are as defined herein, e.g., 1-[4-(4-phenylsulfinylbenzyl)-2-thiazolyl]piperazine, and 1-[4-(4-biphenylylmethyl)-2-thiazolyl]piperazine, and their physiologically tolerable salts are provided. These compounds are useful as medicines for the treatment of inflammation with an immunological component, and are useful as hypolipemic and hypocholesterolemic agents and to assist lowering of lipid and cholesterol content in the blood.
    Type: Grant
    Filed: September 11, 1980
    Date of Patent: January 26, 1982
    Assignee: Science Union et Cie
    Inventors: Gilbert Regnier, Jacques Bure
  • Novel pharmaceutical compositions incorporating an aryltrifluoroethanol
    Patent number: 4285943
    Abstract: This invention relates to pharmaceutical compositions containing as active ingredient an aryltrifluoroethanol, and a process for producing the same.These pharmaceutical compositions are useful for treating or alleviating pain, hyperpyretic conditions and/or inflammatory states.
    Type: Grant
    Filed: November 2, 1979
    Date of Patent: August 25, 1981
    Assignee: Science Union Et Cie
    Inventors: Michel Vincent, Georges Remond, Jacques Bure
  • 1-Methyl-4-piperidinol esters of 4-quinolinylamino benzoates and antiinflammatory and analgesic compositions and methods employing them
    Patent number: 4259335
    Abstract: 1-methyl-4-piperidinol esters of the formula: ##STR1## in which R is 7-chloro-4-quinolyl, 7-trifluoromethyl-4-quinolyl or 8-trifluoromethyl-4-quinolyl.These compounds and physiologically tolerable acid addition salts thereof may be used as medicines especially in the treatment of inflammatory processes and painful syndroms.
    Type: Grant
    Filed: August 6, 1979
    Date of Patent: March 31, 1981
    Assignee: Science Union et Cie, Societe Francaise de Recherche Medicale
    Inventors: Laszlo Beregi, Pierre Hugon, Jacques Bure, Francoise Degrand