Patents by Inventor Jacques Lannoy

Jacques Lannoy has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
    Patent number: 8288560
    Abstract: The invention relates to thiazole, oxazole, imidazole, isoxazole and isoxazoline derivatives of general formula (I) wherein Het is thiazole, oxazole, imidazole, isoxazole or isoxazoline, n is an integer from 0 to 6, A is notably selected from various optionally substituted aromatic radicals, B is notably hydrogen, alkyl or phenyl, R1 and R2 are notably independently hydrogen, alkyl or cycloalkyl and ? is —NR46R47 or —OR48, R46 and R47 are notably independently hydrogen, alkyl, cycloalkyl or —(CH2)k—COOR51, R51 is notably alkyl or haloalkyl and R48 is notably hydrogen or alkyl. These compounds have advantageous pharmacological properties which allow their use in therapeutics, notably for treating neurodegenerative disorders or pain.
    Type: Grant
    Filed: March 21, 2011
    Date of Patent: October 16, 2012
    Assignee: Ipsen Pharma S.A.S.
    Inventors: Pierre-Etienne Chabrier De Lassauniere, Jeremiah Harnett, Dennis Bigg, Anne-Marie Liberatore, Jacques Pommier, Jacques Lannoy, Christophe Thurieau
  • DERIVATIVES OF HETEROCYCLES WITH 5 MEMBERS, THEIR PREPARATION AND THEIR USE AS MEDICAMENTS
    Publication number: 20110172434
    Abstract: The invention relates to thiazole, oxazole, imidazole, isoxazole and isoxazoline derivatives of general formula (I) wherein Het is thiazole, oxazole, imidazole, isoxazole or isoxazoline, n is an integer from 0 to 6, A is notably selected from various optionally substituted aromatic radicals, B is notably hydrogen, alkyl or phenyl, R1 and R2 are notably independently hydrogen, alkyl or cycloalkyl and ? is —NR46R47 or —OR48, R46 and R47 are notably independently hydrogen, alkyl, cycloalkyl or —(CH2)k—COOR51, R51 is notably alkyl or haloalkyl and R48 is notably hydrogen or alkyl. These compounds have advantageous pharmacological properties which allow their use in therapeutics, notably for treating neurodegenerative disorders or pain.
    Type: Application
    Filed: March 21, 2011
    Publication date: July 14, 2011
    Applicant: Ipsen Pharma S.A.S.
    Inventors: Pierre-Etienne CHABRIER DE LASSAUNIERE, Jeremiah Harnett, Dennis Bigg, Anne-Marie Liberatore, Jacques Pommier, Jacques Lannoy, Christophe Thurieau
  • Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
    Patent number: 7956075
    Abstract: The invention relates to thiazole, oxazole, imidazole, isoxazole and isoxazoline derivatives of general formula (I) wherein Het is thiazole, oxazole, imidazole, isoxazole or isoxazoline, n is an integer from 0 to 6, A is notably selected from various optionally substituted aromatic radicals, B is notably hydrogen, alkyl or phenyl, R1 and R2 are notably independently hydrogen, alkyl or cycloalkyl and ? is —NR46R47 or —OR48, R46 and R47 are notably independently hydrogen, alkyl, cycloalkyl or —(CH2)k—COOR51, R51 is notably alkyl or haloalkyl and R48 is notably hydrogen or alkyl. These compounds have advantageous pharmacological properties which allow their use in therapeutics, notably for treating neurodegenerative disorders or pain.
    Type: Grant
    Filed: December 11, 2007
    Date of Patent: June 7, 2011
    Assignee: Ipsen Pharma S.A.S.
    Inventors: Pierre-Etienne Chabrier De Lassauniere, Jeremiah Harnett, Dennis Bigg, Anne-Marie Liberatore, Jacques Pommier, Jacques Lannoy, Christophe Thurieau
  • Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
    Publication number: 20080146627
    Abstract: The invention relates to thiazole, oxazole, imidazole, isoxazole and isoxazoline derivatives of general formula (I) wherein Het is thiazole, oxazole, imidazole, isoxazole or isoxazoline, n is an integer from 0 to 6, A is notably selected from various optionally substituted aromatic radicals, B is notably hydrogen, alkyl or phenyl, R1 and R2 are notably independently hydrogen, alkyl or cycloalkyl and Q is —NR46R47 or —OR48, R46 and R47 are notably independently hydrogen, alkyl, cycloalkyl or —(CH2)k—COOR51, R51 is notably alkyl or haloalkyl and R48 is notably hydrogen or alkyl. These compounds have advantageous pharmacological properties which allow their use in therapeutics, notably for treating neurodegenerative disorders or pain.
    Type: Application
    Filed: December 11, 2007
    Publication date: June 19, 2008
    Inventors: Pierre-Etienne Chabrier De Lassauniere, Jeremiah Harnett, Dennis Bigg, Anne-Marie Liberatore, Jacques Pommier, Jacques Lannoy, Christophe Thurieau
  • Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
    Patent number: 7291641
    Abstract: Thiaxozle, oxazole, imidazole, isoxazole and isoxazoline compounds of the formula wherein Het is thiazole, oxazole, imidazole, isoxazole or isoxazoline, n is an integer from 0 to 6, A is selected from the various optionally substituted aromatic radicals defined in the specification, B is hydrogen, alkyl or phenyl, R1 and R2 are independently hydrogen, alkyl or cycloalkyl or R1 and R2 taken together with the carbon atom which carries them, form a carbocycle with 3 to 7 members and ? is —NH46R47 or —OR48, R46 and R47 are independently hydrogen, alkyl, cycloalkyl or —(CH2)kCOOR51, R51 is alkyl or haloalkyl and R48 is hydrogen or alkyl having advantageous pharmacological properties which allow their use in therapeutics, for treating neurodegenerative disorders or pain.
    Type: Grant
    Filed: August 10, 2004
    Date of Patent: November 6, 2007
    Assignee: Societe de Conseils de Recherches et d'Applications Scientifiques (S.C.R.A.S.)
    Inventors: Pierre-Etienne Chabrier De Lassauniere, Jermiah Harnett, Dennis Bigg, Ann-Marie Liberatore, Jacques Pommier, Jacques Lannoy, Christophe Thurieau, Zheng Xin Dong
  • Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
    Publication number: 20070179153
    Abstract: A method of treating Parkinson's disease in warm-blooded animals comprising administering to warm-blooded animals in need thereof an effective amount of a compound of the formula wherein the substituents are defined as in the specification
    Type: Application
    Filed: February 20, 2007
    Publication date: August 2, 2007
    Inventors: Pierre Chabrier de Lassauniere, Anne-Marie Liberatore, Christophe Thurieau, Jeremiah Harnett, Denis Bigg, Jacuqes Pommier, Jacques Lannoy
  • Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
    Publication number: 20070021390
    Abstract: A method of treating Parkinson's disease in warm-blooded animals comprising administering to warm-blooded animals in need thereof an amount of a compound of the formula in racemic, enantiomeric form or any combination of these forms, wherein the substituents are as defined in the specification.
    Type: Application
    Filed: October 24, 2005
    Publication date: January 25, 2007
    Inventors: Pierre Chabrier de Lassauniere, Jeremiah Harnett, Denis Bigg, Jacuqes Pommier, Jacques Lannoy, Anne-Marie Liberatore, Christophe Thurieau
  • Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
    Publication number: 20050038087
    Abstract: The invention relates to thiazole, oxazole, imidazole, isoxazole and isoxazoline derivatives of general formula (I) wherein Het is thiazole, oxazole, imidazole, isoxazole or isoxazoline, n is an integer from 0 to 6, A is notably selected from various optionally substituted aromatic radicals, B is notably hydrogen, alkyl or phenyl, R1 and R2 are notably independently hydrogen, alkyl or cycloalkyl or R1 and R2, taken together with the carbon atom which carries them, form a carbocycle with 3 to 7 members and ? is —NR46R47 or —OR48, R46 and R47 are notably independently hydrogen, alkyl, cycloalkyl or —(CH2)k—COOR51, R51 is notably alkyl or haloalkyl and R48 is notably hydrogen or alkyl. These compounds have advantageous pharmacological properties which allow their use in therapeutics, notably for treating neurodegenerative disorders or pain.
    Type: Application
    Filed: August 10, 2004
    Publication date: February 17, 2005
    Inventors: Pierre-Etienne Chabrier De Lassauniere, Jermiah Harnett, Dennis Bigg, Ann-Marie Liberatore, Jacques Pommier, Jacques Lannoy, Christophe Thurieau, Zheng Xin Dong
  • Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
    Publication number: 20040132788
    Abstract: The invention relates to thiazole, oxazole, imidazole, isoxazole and isoxazoline derivatives of general formula (I) 1
    Type: Application
    Filed: October 8, 2003
    Publication date: July 8, 2004
    Inventors: Pierre-Etienne Chabrier De Lassauniere, Jeremiah Harnett, Dennis Bigg, Anne-Marie Liberatore, Jacques Pommier, Jacques Lannoy, Christophe Thurieau