Patents by Inventor Jag Paul Heer

Jag Paul Heer has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • OXADIAZOLE DERIVATIVES ACTIVE ON SPHINGOSINE-1-PHOSPHATE (S1P)
    Publication number: 20100152235
    Abstract: The present invention relates to a novel oxadiazole derivative having pharmacological activity, processes for its preparation, pharmaceutical compositions containing it and its use in the treatment of various disorders.
    Type: Application
    Filed: February 24, 2010
    Publication date: June 17, 2010
    Inventors: Jag Paul Heer, Thomas Daniel Heightman
  • XANTHINE DERIVATIVES AS SELECTIVE HM74A AGONISTS
    Publication number: 20100099690
    Abstract: The present invention relates to compounds which are xanthine derivatives, processes for the manufacture of said derivatives, pharmaceutical formulations containing the active compounds and the use of the compounds in therapy, for example, in the treatment of diseases where under-activation of the HM74A receptor contributes to the disease or where activation of the receptor will be beneficial.
    Type: Application
    Filed: August 8, 2006
    Publication date: April 22, 2010
    Inventors: Jag Paul Heer, Ian Edward David Smith
  • Novel Derivatives
    Publication number: 20100022555
    Abstract: The present invention relates to novel piperazine derivatives; to processes for their preparation; to pharmaceutical compositions containing the derivatives; and to the use of the derivatives in therapy to treat diseases for which blocking the Cav2.2 calcium channels is beneficial.
    Type: Application
    Filed: July 15, 2009
    Publication date: January 28, 2010
    Inventors: Paul John Beswick, Alister Campbell, Andrew Cridland, Robert James Gleave, Jag Paul Heer, Neville Hubert Nicholson, Lee William Page, Sadie Vile
  • Novel Derivatives
    Publication number: 20100016330
    Abstract: The present invention relates to novel piperazine derivatives; to processes for their preparation; to pharmaceutical compositions containing the derivatives; and to the use of the derivatives in therapy to treat diseases for which blocking the Cav2.2 calcium channels is beneficial.
    Type: Application
    Filed: July 15, 2009
    Publication date: January 21, 2010
    Inventors: Jag Paul Heer, David Norton, Simon E. Ward
  • Thiazolyl substituted triazoles as alk5 inhibitors
    Publication number: 20040266842
    Abstract: Thiazolyl substituted triazoles of formula (I) 1
    Type: Application
    Filed: May 13, 2004
    Publication date: December 30, 2004
    Inventors: Laramie Mary Gaster, John David Harling, Jag Paul Heer, Thomas David Heightman, Andrew Hele Payne
  • Pyridinylimidazoles
    Publication number: 20040220230
    Abstract: Compounds of formula (I) and pharmaceutically acceptable salts thereof: 1
    Type: Application
    Filed: January 29, 2004
    Publication date: November 4, 2004
    Applicant: SmithKline Beecham p.l.c.
    Inventors: Laramie Mary Gaster, Michael Stewart Hadley, John David Harling, Frank Peter Harrington, Jag Paul Heer, Thomas Daniel Heightman, Andrew Hele Payne
  • Pyridyl-substituted triazoles as tgf inhibitors
    Publication number: 20040152738
    Abstract: Pyridyl substituted triazoles of formula (I) 1
    Type: Application
    Filed: March 22, 2004
    Publication date: August 5, 2004
    Inventors: Laramie Mary Gaster, John David Harling, Jag Paul Heer, Thomas Daniel Heightman, Andrew Hele Payne
  • Pyridinylimidazoles
    Publication number: 20030166633
    Abstract: Compounds of formula (I) and pharmaceutically acceptable salts thereof wherein R1, R2 and R3 represent various functional groups, and one of X1 and X2 is N and the other is NR10; and their use as pharmaceuticals.
    Type: Application
    Filed: October 29, 2002
    Publication date: September 4, 2003
    Inventors: Laramie Mary Gaster, Michael Stewart Hadley, John David Harling, Frank Peter Harrington, Jag Paul Heer, Thomas Daniel Heightman, Andrew Hele Payne
  • Substituted isoquinoline derivatives and their use as anticonvulsivants
    Patent number: 6492378
    Abstract: This invention relates to novel substituted isoquinoline derivatives and their use as anticonvulsants.
    Type: Grant
    Filed: February 9, 2001
    Date of Patent: December 10, 2002
    Assignee: SmithKline Beecham p.l.c.
    Inventors: John David Harling, Jag Paul Heer, Mervyn Thompson