Patents by Inventor Jean-Christophe GAUVIN

Jean-Christophe GAUVIN has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 10106544
    Abstract: The invention relates to antibacterial compounds of formula I wherein R1 is one of the groups represented below wherein A is a bond, CH?CH or C?C; U is N or CH; V is N or CH; W represents N or CH; and R1A, R2A, R3A, R1B and R1C are as defined in the claims; and salts thereof.
    Type: Grant
    Filed: March 3, 2015
    Date of Patent: October 23, 2018
    Assignee: IDORSIA PHARMACEUTICALS LTD
    Inventors: Gaelle Chapoux, Jean-Christophe Gauvin, Azely Mirre, Philippe Panchaud, Christine Schmitt, Jean-Luc Specklin, Jean-Philippe Surivet
  • Publication number: 20180251434
    Abstract: The invention relates to antibacterial compounds of formula I wherein R1, M, R2, R3, and V are as described in the description, to their preparation, to salts thereof, and to their use as pharmaceuticals, to pharmaceutical compositions containing one or more compounds of formula I, and especially to their use as antibacterial agents.
    Type: Application
    Filed: August 30, 2016
    Publication date: September 6, 2018
    Inventors: Stefan DIETHELM, Jean-Christophe GAUVIN, Gaelle MATHIEU, Philippe PANCHAUD, Jean-Philippe SURIVET
  • Patent number: 9802901
    Abstract: The invention relates to antibacterial compounds of formula I wherein R1 is H or halogen; R2 is alkynyloxy or the group M; R3 is H or halogen; M is one of the groups wherein A is a bond, CH2CH2, CH?CH or C?C and R1A, R2A, R3A, R1B and R1C are as defined in claim 1; and salts thereof.
    Type: Grant
    Filed: September 12, 2014
    Date of Patent: October 31, 2017
    Assignee: IDORSIA PHARMACEUTICALS LTD
    Inventors: Jean-Christophe Gauvin, Azely Mirre, Etienne Ochala, Jean-Philippe Surivet
  • Patent number: 9796686
    Abstract: The invention relates to antibacterial compounds of formula I wherein R1 is H or halogen; R2 is the group M; R3 is H or halogen; M is MA or MB wherein A is a bond or C?C; R1A is H or halogen; R2A is H, alkoxy or halogen; R3A is H, alkoxy, hydroxyalkoxy, hydroxyalkyl, 1,2-dihydroxyethyl, dialkylamino, 1-hydroxymethyl-cycloprop-1-yl, 1-((dimethylglycyl)oxy)methyl-cycloprop-1-yl, 3-hydroxyoxetan-3-yl, morpholin-4-ylalkyl or morpholin-4-ylalkoxy; and R1B is a group as defined in claim 1; and salts thereof.
    Type: Grant
    Filed: May 13, 2015
    Date of Patent: October 24, 2017
    Assignee: IDORSIA PHARMACEUTICALS LTD
    Inventors: Gaëlle Chapoux, Jean-Christophe Gauvin, Azely Mirre, Jean-Philippe Surivet
  • Publication number: 20170107223
    Abstract: The invention relates to antibacterial compounds of formula I wherein R1 is one of the groups represented below wherein A is a bond, CH?CH or C?C; U is N or CH; V is N or CH; W represents N or CH; and R1A, R2A, R3A, R1B and R1C are as defined in the claims; and salts thereof.
    Type: Application
    Filed: March 3, 2015
    Publication date: April 20, 2017
    Inventors: Gaelle CHAPOUX, Jean-Christophe GAUVIN, Azely MIRRE, Philippe PANCHAUD, Christine SCHMITT, Jean-Luc SPECKLIN, Jean-Philippe SURIVET
  • Patent number: 9624206
    Abstract: The invention relates to antibacterial compounds of formula I wherein X is N or CH; R1 is H or halogen; R2 is alkynyloxy or the group M; R3 is H or halogen; M is one of the groups MA and MB represented below wherein A is a bond, CH2CH2, CH?CH or C?C; R1A is H or halogen; R2A is H, alkoxy or halogen; R3A is H, alkoxy, hydroxyalkoxy, alkoxyalkoxy, thioalkoxy, trifluoromethoxy, amino, hydroxyalkyl, 2-hydroxyacetamido, 1-aminocyclopropyl, 1-hydroxymethyl-cycloprop-1-yl, 1-((phosphonooxy)methyl)cyclopropyl, 1-(((dimethylglycyl)oxy)methyl)cyclopropyl, trans-2-hydroxymethyl-cycloprop-1-yl, 1,2-dihydroxyethyl, 3-hydroxyoxetan-3-yl, 3-(hydroxyalkyl)oxetan-3-yl, 3-aminooxetan-3-yl, 3-hydroxythietan-3-yl, morpholin-4-ylalkoxy, morpholin-4-yl-alkyl, oxazol-2-yl or [1,2,3]triazol-2-yl; and R1B is hydroxyalkyl, dihydroxyalkyl, aminoalkyl, 1-hydroxymethyl-cycloprop-1-yl, 1-aminomethyl-cycloprop-1-yl, trans-2-hydroxymethyl-cycloprop-1-yl, 3-hydroxyoxetan-3-yl, 3-hydroxythietan-3-yl, 1-(2-hydroxyacetyl)azetidin-3-yl,
    Type: Grant
    Filed: December 18, 2014
    Date of Patent: April 18, 2017
    Assignee: ACTELION PHARMACEUTICALS LTD
    Inventors: Gaelle Chapoux, Jean-Christophe Gauvin, Christian Hubschwerlen, Azely Mirre, Etienne Ochala, Jean-Luc Specklin, Jean-Philippe Surivet
  • Publication number: 20170081292
    Abstract: The invention relates to antibacterial compounds of formula I wherein R1 is H or halogen; R2 is the group M; R3 is H or halogen; M is MA or MB wherein A is a bond or C?C; R1A is H or halogen; R2A is H, alkoxy or halogen; R3A is H, alkoxy, hydroxyalkoxy, hydroxyalkyl, 1,2-dihydroxyethyl, dialkylamino, 1-hydroxymethyl-cycloprop-1-yl, 1-((dimethylglycyl)oxy)methyl-cycloprop-1-yl, 3-hydroxyoxetan-3-yl, morpholin-4-ylalkyl or morpholin-4-ylalkoxy; and R1B is a group as defined in claim 1; and salts thereof.
    Type: Application
    Filed: May 13, 2015
    Publication date: March 23, 2017
    Inventors: Gaëlle CHAPOUX, Jean-Christophe GAUVIN, Azely MIRRE, Jean-Philippe SURIVET
  • Publication number: 20170029411
    Abstract: The invention relates to antibacterial compounds of formula I wherein X is N or CH; R1 is H or halogen; R2 is alkynyloxy or the group M; R3 is H or halogen; M is one of the groups MA and MB represented below wherein A is a bond, CH2CH2, CH?CH or C?C; R1A is H or halogen; R2A is H, alkoxy or halogen; R3A is H, alkoxy, hydroxyalkoxy, alkoxyalkoxy, thioalkoxy, trifluoromethoxy, amino, hydroxyalkyl, 2-hydroxyacetamido, 1-aminocyclopropyl, 1-hydroxymethyl-cycloprop-1-yl, 1-((phosphonooxy)methyl)cyclopropyl, 1-(((dimethylglycyl)oxy)methyl)cyclopropyl, trans-2-hydroxymethyl-cycloprop-1-yl, 1,2-dihydroxyethyl, 3-hydroxyoxetan-3-yl, 3-(hydroxyalkyl)oxetan-3-yl, 3-aminooxetan-3-yl, 3-hydroxythietan-3-yl, morpholin-4-ylalkoxy, morpholin-4-yl-alkyl, oxazol-2-yl or [1,2,3]triazol-2-yl; and R1B is hydroxyalkyl, dihydroxyalkyl, aminoalkyl, 1-hydroxymethyl-cycloprop-1-yl, 1-aminomethyl-cycloprop-1-yl, trans-2-hydroxymethyl-cycloprop-1-yl, 3-hydroxyoxetan-3-yl, 3-hydroxythietan-3-yl, 1-(2-hydroxyacetyl)azetidin-3-yl,
    Type: Application
    Filed: December 18, 2014
    Publication date: February 2, 2017
    Applicant: ACTELION PHARMACEUTICALS LTD
    Inventors: Gaelle CHAPOUX, Jean-Christophe GAUVIN, Christian HUBSCHWERLEN, Azely MIRRE, Etienne OCHALA, Jean-Luc SPECKLIN, Jean-Philippe SURIVET
  • Publication number: 20160221959
    Abstract: The invention relates to antibacterial compounds of formula I wherein R1 is H or halogen; R2 is alkynyloxy or the group M; R3 is H or halogen; M is one of the groups wherein A is a bond, CH2CH2, CH?CH or C?C and R1A, R2A, R3A, R1B and R1C are as defined in claim 1; and salts thereof.
    Type: Application
    Filed: September 9, 2014
    Publication date: August 4, 2016
    Inventors: Jean-Christophe GAUVIN, Azely MIRRE, Etienne OCHALA, Jean-Philippe SURIVET