Patents by Inventor Jean-Pierre Tarayre

Jean-Pierre Tarayre has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Publication number: 20120088792
    Abstract: The invention concerns the use of compounds of general formula (I) for treating opioid drug dependence, hyperalgesia induced by opiate drug withdrawal and psychological craving induced by opiate drug withdrawal.
    Type: Application
    Filed: October 7, 2011
    Publication date: April 12, 2012
    Applicant: Pierre Fabre Medicament
    Inventors: Francis Colpaert, Liesbeth Bruins Slot, Gilbert Alphonse Morales, Wouter Koek, Jean-Pierre Tarayre, Bernard Vacher
  • Patent number: 8106074
    Abstract: The invention concerns the use pf compounds of general formula (I) for treating opioid drug dependence, hyperalgesia induced by opiate drug withdrawal and psychological craving induced by opiate drug withdrawal.
    Type: Grant
    Filed: December 4, 2008
    Date of Patent: January 31, 2012
    Assignee: Pierre Fabre Medicament
    Inventors: Francis Colpaert, Liesbeth Bruins Slot, Gilbert Alphonse Morales, legal representative, Wouter Koek, Jean-Pierre Tarayre, Bernard Vacher
  • Publication number: 20100099709
    Abstract: The invention concerns the use pf compounds of general formula (I) for treating opioid drug dependence, hyperalgesia induced by opiate drug withdrawal and psychological craving induced by opiate drug withdrawal.
    Type: Application
    Filed: December 4, 2008
    Publication date: April 22, 2010
    Applicant: Pierre Fabre Medicament
    Inventors: Francis COLPAERT, Liesbeth Bruins Slot, Gilbert Alphonse Morales, Wouler Koek, Jean-Pierre Tarayre, Bernard Vacher
  • Publication number: 20050065348
    Abstract: The invention concerns compounds of general formula (I) for treating opioid drug dependence.
    Type: Application
    Filed: July 11, 2002
    Publication date: March 24, 2005
    Inventors: Francis Colpaert, Liesbeth Slot, Wouter Koek, Jean-Pierre Tarayre, Bernard Vacher
  • Patent number: 5633255
    Abstract: 1,2-dihydro-2-oxo-3-amino-quinoxaline derivatives of general formula (I) in which R.sub.1 and R.sub.2 are independently hydrogen or a straight or branched C.sub.1 -C.sub.4 alkyl radical, R.sub.3 is a straight or branched C.sub.3 -C.sub.6 alkyl, alkenyl or hydroxy-alkyl grouping, their salts with pharmaceutically-acceptable acids, and a method for preparing them and their use in therapy are disclosed.
    Type: Grant
    Filed: April 6, 1995
    Date of Patent: May 27, 1997
    Assignee: Pierre Fabre Medicament
    Inventors: Dennis Bigg, Jean-Francois Patoiseau, Jean-Marie Autin, Jean-Pierre Tarayre
  • Patent number: 5198441
    Abstract: New derivatives of 1,2-dihydro 2-oxo quinoxalines corresponding to the general formula I: ##STR1## in which: R is a hydrogen or halogen atomR.sub.1 is a hydrogen atom or a straight or branched C.sub.1 -C.sub.4 alkyl radicalR.sub.2 is:a hydrogen atoma C(O)R.sub.4 radical in which R.sub.4 is a straight or branched C.sub.1 -C.sub.4 alkyl groupa C(O)NHR.sub.5 radical in which R.sub.5 is a straight or branched C.sub.1 -C.sub.4 alkyl radical or a phenyl groupA is a C.sub.1 -C.sub.4 alkaline chainR.sub.3 represents:a hydrogen atom, a C.sub.1 -C.sub.4 alkyl radical, a C.sub.3 -C.sub.6 cycloalkyl radical, an alcynyl, nitrile, hydroxyl, carboxamido, pyridyl, phenyl group, or a phenyl group substituted by a halogen atom, a C.sub.1 -C.sub.4 alkyl group, a C.sub.1 -C.sub.4 alkoxy group or a nitro groupan alkenyl radical of the formula: ##STR2## in which R.sub.6, R.sub.7 may, independently of each other, be a hydrogen atom, a C.sub.1 -C.sub.
    Type: Grant
    Filed: June 17, 1991
    Date of Patent: March 30, 1993
    Assignee: Pierre Fabre Medicament
    Inventors: Guy Pitet, Christian Faure, Francoise Couret, Dennis Bigg, Jean-Pierre Tarayre
  • Patent number: 4510142
    Abstract: This invention relates to new derivatives of biphenyl alkyl carboxylates, to a process for the preparation thereof and the use thereof as medicaments.The new derivatives according to the present invention correspond to general formula (I): ##STR1## wherein X represents a hydrogen atom or a halogen atom,R represents a hydrogen atom or an alkyl group, andR.sub.1 represents the following groups: ##STR2## These compounds will notably be used in the treatment of obstinate pains and inflammatory syndromes.
    Type: Grant
    Filed: October 12, 1982
    Date of Patent: April 9, 1985
    Assignee: Pierre Fabre S.A.
    Inventors: Henry Cousse, Gilbert Mouzin, Jean-Pierre Tarayre, Jean-Pierre Rieu
  • Patent number: 4246271
    Abstract: The present invention relates to new derivatives of 4-phenyl-2-thiazolyl oxamates having the formula: ##STR1## in which: X represents hydrogen, halogen, lower-alkyl, or lower-alkoxy.R is lower-alkyl or phenyllower-alkyl, e.g., benzyl.These compounds, which have inhibiting properties on the passive cutaneous anaphylactic reaction, are useful in the treatment of asthma. Pharmaceutical compositions thereof and method of treating therewith.
    Type: Grant
    Filed: June 14, 1979
    Date of Patent: January 20, 1981
    Inventors: Henri Cousse, Gilbert Mouzin, Jean-Pierre Tarayre, Silvano Casadio
  • Patent number: 4225610
    Abstract: The present invention concerns new derivatives of 4-phenyl 2-amino thiazole of the formula ##STR1## in which X represents a hydrogen atom, a halogen, a lower alkyl or an alkoxy,R is a hydrogen, a haloalkoxy, a substituted or unsubstituted aryl, a pyridyl, an aryloxy or a carboxy alkyl, having immunomodulating properties, useful in the treatment of rheumatoid arthritis and other ailments requiring immunotherapy.
    Type: Grant
    Filed: October 19, 1978
    Date of Patent: September 30, 1980
    Assignee: Pierre Fabre, S.A.
    Inventors: Jean-Pierre Tarayre, Henri Cousse, Gilbert Mouzin, Henri Lauressergues, Silvano Casadio
  • Patent number: 4192883
    Abstract: New chemical compounds, which are pyrrolidinoethylamine amides, in the form of free bases and salts thereof, which are useful as antitussives, pharmaceutical compositions thereof, and method of treating therewith.In the form of their salts, the compounds have the formula: ##STR1## wherein ##STR2## is an acyl radical of a phenylacetic,.alpha.-phenyl-.alpha.-ethylacetic, diphenylacetic, benzilic, .alpha.-lower-alkoxy-.alpha.,.alpha.-diphenylacetic, 10-phenothiazinecarboxylic, benzoic, halobenzoic, 3-coumarincarboxylic, 9-xanthenecarboxylic, salicylic, cresotic, halocresotic, lower-alkoxybenzoic, phenoxyacetic, phenoxyisobutyric, halophenoxyisobutyric, cinnamic, or 9-fluorene carboxylic acid, and wherein R'H represents an inorganic or organic acid, and wherein R may be, for example, a substituted aromatic ring of the formula: ##STR3## wherein R.sub.1 and R.sub.2 may independently be lower-alkyl, lower-alkoxy, hydrogen, lower-alkenyloxy, or lower-alkynyloxy, and X may be hydrogen or halogen.
    Type: Grant
    Filed: August 7, 1978
    Date of Patent: March 11, 1980
    Assignee: Pierre Fabre, S.A.
    Inventors: Henri Cousse, Bernard Bonnaud, Jean-Pierre Tarayre, Silvano Casadio
  • Patent number: 4122199
    Abstract: New chemical compounds, which are pyrrolidinoethylamine amides, in the form of free bases and salts thereof, which are useful as antitussives, pharmaceutical compositions thereof, and method of treating therewith.In the form of their salts, the compounds have the formula: ##STR1## wherein ##STR2## is an acyl radical of a phenylacetic, 60 -phenyl-.alpha.-(1 to 5 C atoms) acetic, (1 to 5 C atoms) diphenylacetic, benzilic, diphenyl-.alpha.-chloroacetic, .alpha.-lower-alkoxy-.alpha.,.alpha.-diphenylacetic, 3-coumarincarboxylic, 9-xanthenecarboxylic, phenoxyacetic, phenoxyisobutyric, halophenoxyisobutyric, or 9-flourene carboxylic acid, and wherein R'H represents an inorganic or organic acid.Medicaments containing these active principles may be used, inter alia, in the treatment of coughs and respiratory complaints.
    Type: Grant
    Filed: August 16, 1976
    Date of Patent: October 24, 1978
    Assignee: Pierre Fabre S.A.
    Inventors: Henri Cousse, Bernard Bonnaud, Jean-Pierre Tarayre, Silvano Casadio