Patents by Inventor Joachim Rheinheimer

Joachim Rheinheimer has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 7119097
    Abstract: A compound of the formula pharmaceutically acceptable salts and enantiomers thereof and pharmaceutical compositions containing this compound, its pharmaceutically acceptable salts and enantiomers are claimed.
    Type: Grant
    Filed: March 16, 2006
    Date of Patent: October 10, 2006
    Assignee: Abbott GmbH & Co. KG
    Inventors: Hartmut Riechers, Dagmar Klinge, Wilhelm Amberg, Andreas Kling, Stefan Muller, Ernst Baumann, Joachim Rheinheimer, Uwe Josef Vogelbacher, Wolfgang Wernet, Liliane Unger, Manfred Raschack
  • Publication number: 20060217400
    Abstract: Triazolopyrimidines of the formula I in which the index n and the substituents R1, R2 and R3 are as defined in the description, and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
    Type: Application
    Filed: December 17, 2003
    Publication date: September 28, 2006
    Inventors: Bernd Müller, Jordi Blasco, Thomas Grote, Carsten Blettner, Markus Gewehr, Wassilios Grammenos, Andreas Gypser, Joachim Rheinheimer, Peter Schäfer, Frank Schieweck, Anja Schwögler, Eberhard Ammermann, Siegfried Strathmann, Ulrich Schöfl, Reinhard Stierl
  • Publication number: 20060211573
    Abstract: 7-(Alkenylamino)triazolopyrimidines of the formula I wherein the substituents have the following meanings: L is halogen, alkyl, haloalkyl, alkoxy, amino, NHR or NR2; R is alkyl or alkyl-carbonyl; m is 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl or alkoxy; R1 is alkyl or haloalkyl; R2 is hydrogen, alkyl or haloalkyl; R3 is alkenyl, which can be unsubstituted or partially or completely halogenated or can be substituted according to the Description; R4 is hydrogen or alkyl, R3 and R4 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered unsaturated ring which can be interrupted by an atom from the group consisting of O, N and S and/or can carry one or more sub-stituents. Processes for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.
    Type: Application
    Filed: March 24, 2004
    Publication date: September 21, 2006
    Inventors: Jordi Blasco, Carsten Blettner, Bernd Muller, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Peter Schalfer, Frank Schieweck, Anja Schwogler, Maria Scherer, Siegfried Strathmann, Ulrich Schofl, Reinhard Stierl
  • Publication number: 20060211711
    Abstract: 7-alkinylamino-triazolopyrimidins of formula (I), wherein the substituents have the following meanings: L=halogen, alkyl, halogenalkyl, alkoxy, amino, NHR, NR2, cyano, S(O)nA1 or C(O)A2; R=alkyl or alkylcarbonyl, A1=hydrogen, hydroxy, alkyl, alkylamino or aialkylamino; n=0, 1 or 2; A2=alkenyl, alkoxy, halogenalkoxy or one of the groups cited in A1; m=1, 2, 3, 4 or 5, whereby at least one group L is present in an ortho-position to the bond with the triazolopyrimidine skeleton; X=halogen, cyano, alkyl, halogenalkyl or alkoxy; R1=hydrogen or alkyl; R2=alkinyl which can be unsubstituted or substituted according to the description. The invention also relates to methods for the production of said compounds, agents containing said compounds and the use thereof to combat harmful phytopathogenic fungi.
    Type: Application
    Filed: March 30, 2004
    Publication date: September 21, 2006
    Inventors: Jordi Blasco, Carsten Blettner, Bernd Müller, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Peter Schäfer, Frank Schieweck, Anja Schwögler, Maria Scherer, Siegfried Strathmann, Ulrich Schöfl, Reinhard Stierl
  • Patent number: 7109205
    Abstract: Carboxylic acid derivatives where R–R6, X, Y and Z have the meanings stated in the description, and the preparation thereof, are described. The novel compounds are suitable for controlling diseases.
    Type: Grant
    Filed: June 24, 2003
    Date of Patent: September 19, 2006
    Assignee: Abbott GmbH & Co. KG
    Inventors: Hartmut Riechers, Dagmar Klinge, Wilhelm Amberg, Andreas Kling, Stefan Müller, Ernst Baumann, Joachim Rheinheimer, Uwe Josef Vogelbacher, Wolfgang Wernet, Liliane Unger, Manfred Raschack
  • Publication number: 20060199801
    Abstract: Bicyclic compounds of the formula I in which A1 or A5 is C and the other of the two variables A1, A5 is N, C or C—R3; A2, A3, A4 independently of one another are N or C—R3a, where one of the variables A2, A3 or A4 may also be S or a group N—R4 if A1 and A5 are both C, and where A4 is not N or C—R3a if A1 is N, A3 is C—R3a and A5 is C, and where A1 is attached to A2 and A3 to A4 or A2 is attached to A3 and A4 to A5 or A1 is attached to A5 and A2 to A3 or A1 is attached to A5 and A3 to A4 or A1 is attached to A2 and A4 to A5 by double bonds; n is 0, 1, 2, 3, 4 or 5; Ra is halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkyl, C1-C6-haloalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R5; R1 is halogen, cyano, C1-C10-alkyl, where a carbon atom of the C1-C10-alkyl radical may be replaced by a silicium atom, C1-C6-haloalkyl, C2-C10-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C4-alkyl, where the cycloalkyl moiety of the two last-mentioned groups may be unsu
    Type: Application
    Filed: April 16, 2004
    Publication date: September 7, 2006
    Inventors: Jordi i Blasco, Carsten Blettner, Bernd Muller, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Peter Schafer, Frank Schieweck, Anja Schwogler, Oliver Wagner, Eberhard Ammermann, Siegfried Strathmann, Ulrich Schofl, Maria Scherer, Reinhard Stierl
  • Patent number: 7101900
    Abstract: Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described. In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1–C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1–C6-alkyl, C1–C6-alkoxy, C1–C4-haloalkyl, C1–C4-haloalkoxy, C1–C4-alkylthio, C1–C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1–C6-alkyl, thienyl-C1–C4-alkyl, or pyrazolyl-C1–C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1–C6-alkyl, C1–C6-alkoxy, C1–C4-haloalkyl, C1–C4-haloalkoxy, C1–C4-alkylthio, C1–C4-alkoxyalkoxy, C1–C6-alkylcarbonyl; n is 0–5; p is, depending on the number of free valencies, 0–4.
    Type: Grant
    Filed: February 22, 2005
    Date of Patent: September 5, 2006
    Assignee: BASF Aktiengesellschaft
    Inventors: Joachim Rheinheimer, Karl Eicken, Ingo Rose, Thomas Grote, Eberhard Ammermann, John-Bryan Speakman, Siegfried Strathmann, Gisela Lorenz
  • Patent number: 7094894
    Abstract: Disclosed are a method for producing fungicidal triazolopyrimidine compounds, agents containing said compounds, and the use thereof for controlling harmful fungi. Also disclosed are triazolopyrimidines of formula (I), in which the substituents have the following meaning: L1 represents alkyl; L2 represents halogen; L3represents hydrogen or halogen; X represents halogen, cyano, alkyl, alkoxy, or haloalkoxy; R1, R2 represent hydrogen, alkyl, haloalkyl, cycloalkyl, alkenyl, alkadienyl, alkinyl, or cycloalkinyl, phenyl, naphthyl, or a five-unit to ten-unit saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group O, N, or S, R1 and R2 can also form a five-unit or six-unit ring along with the nitrogen atom to which they are linked. Said ring can be interrupted and/or substituted by an atom from the group O, N, and S while R1 and/or R2 can be substituted according to the description.
    Type: Grant
    Filed: April 30, 2003
    Date of Patent: August 22, 2006
    Assignee: BASF Aktiengesellschaft
    Inventors: Jordi Tormo i Blasco, Carsten Blettner, Bernd Müller, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Peter Schäfer, Frank Schieweck, Anja Schwögler, Eberhard Ammermann, Siegfried Strathmann, Gisela Lorenz, Reinhard Stierl
  • Publication number: 20060172891
    Abstract: The invention relates to novel biphenyl carboxamides of formula (I), wherein A, R, Z, X, Y, m and n have the meanings given in the description, to multiple methods for producing these substances, to their use for combating unwanted micro-organisms and to novel intermediate products and the production thereof.
    Type: Application
    Filed: March 20, 2004
    Publication date: August 3, 2006
    Inventors: Markus Gewehr, Bernd Muller, Thomas Grote, Wassilios Grammenos, Andreas Gypser, Jordi Blasco, Anja Schwogler, Joachim Rheinheimer, Carsten Blettner, Frank Schieweck, Michael Rack, Ulrich Schofl, Siegfried Strathmann, Reinhard Stierl, Jan Rether
  • Publication number: 20060167017
    Abstract: Triazolopyrimidines of the formula I where the index and the substituents are as defined below: R1 is C1-C10-alkyl, C2-C10-alkenyl, C2-C10-alkynyl, C3-C10-cycloalkyl, C3-C10-cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon to the triazolopyrimidine and contains one to four heteroatoms from the group consisting of N, O and S; R2 is C1-C4-alkyl which may be substituted by halogen, cyano, nitro or C1-C2-alkoxy; n is 0 or an integer from 1 to 4; R is as defined in the description; X is SOm—Rx, NRxRy or NRx—(C?O)—Ry; m is 0 or an integer from 1 to 3; and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
    Type: Application
    Filed: December 16, 2003
    Publication date: July 27, 2006
    Applicant: BASF Aktiengesellschaft
    Inventors: Bernd Muller, Jordi Blasco, Thomas Grote, Carsten Blettner, Markus Gewehr, Wassilios Grammenos, Andreas Gypser, Joachim Rheinheimer, Peter Schafer, Frank Schieweck, Anja Schwogler, Eberhard Ammermann, Siegfried Strathmann, Ulrich Schofl, Reinhard Stierl
  • Publication number: 20060160811
    Abstract: The present invention relates to bicyclic compounds of general formula I, in which X, Y independently of one another are N or C—R4; n is 1, 2, 3, 4 or 5; Ra is halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkyl, C1-C6-haloalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R5; R1 is halogen, cyano, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl which is optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl which is optionally mono- or polysubstituted by alkyl and/or halogen, OR6, SR6 or NR7R8; R2 is halogen, cyano, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl which is optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl which is optionally mono- or polysubstituted by alkyl and/or halogen, OR6, SR6 or NR7R8; R3 is hydrogen, C1-C6-alkyl, C1-C6-haloalkyl or C3-C6-cycloalkyl which is optionally mono- or polysubstituted by alkyl and/or halogen; and the agriculturally acceptable salts of co
    Type: Application
    Filed: July 15, 2004
    Publication date: July 20, 2006
    Inventors: Oliver Wagner, Thomas Grote, Carsten Blettner, Markus Gewehr, Wassilios Grammenos, Andreas Gypser, Bernd Muller, Joachim Rheinheimer, Peter Schafer, Frank Schieweck, Anja Schwogler, Jordi Blasco, Alan Akers, John-Bryan Speakman, Michael Rack, Reinhard Stierl, Maria Scherer, Siegfried Strathmann, Ulrich Schofl
  • Publication number: 20060160808
    Abstract: A compound of the formula pharmaceutically acceptable salts and enantiomers thereof and pharmaceutical compositions containing this compound, its pharmaceutically acceptable salts and enantiomers are claimed.
    Type: Application
    Filed: March 16, 2006
    Publication date: July 20, 2006
    Inventors: Hartmut Riechers, Dagmar Klinge, Wilhelm Amberg, Andreas Kling, Stefan Muller, Ernst Baumann, Joachim Rheinheimer, Owe Vogelbacher, Wolfgang Wernet, Liliane Unger, Manfred Rashack
  • Patent number: 7071334
    Abstract: 6-(2-Chloro-6-fluoro-phenyl)-triazolopyrimidines of formula (I), in which R1 and R2 independently denote hydrogen or alkyl, alkenyl, alkynyl, alkadienyl, or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R1 and R2 radicals may be unsubstituted or partially or fully halogenated or may be substituted as defined in the description.
    Type: Grant
    Filed: April 6, 2002
    Date of Patent: July 4, 2006
    Assignee: BASF Aktiengesellschaft
    Inventors: Jordi Tormo i Blasco, Hubert Sauter, Bernd Müller, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Ingo Rose, Peter Schäfer, Frank Schieweck, Eberhard Ammermann, Siegfried Strathmann, Gisela Lorenz, Reinhard Stierl
  • Publication number: 20060135538
    Abstract: 7-(R)-Aminotriazolopyrimidines of the formula I where the substituents and the index are as defined below: R1 is hydrogen or methyl; R2 is methyl; R3 is C2-C1o-alkyl, C1-C4-alkoxymethyl, C3-C1o-cycloalkyl; R4 is halogen, Cl-C4-alkyl, C1-C4-haloalkyl or Cl-C4-alkoxy; n is a number from 1 to 5; Y is halogen, cyano, Cl-C4-alkyl or Cl-C4-alkoxy; where * is a center of chirality in the R configuration, processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
    Type: Application
    Filed: January 30, 2006
    Publication date: June 22, 2006
    Inventors: Jordi Tormo Blasco, Klaus Ditrich, Hubert Sauter, Oliver Cullmann, Markus Gewehr, Wassilios Grammenos, Bernd Muller, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Ingo Rose, Peter Schafer, Frank Schieweck, Eberhard Ammermann, Siegfried Strathmann, Gisela Lorenz, Reinhard Stierl
  • Patent number: 7038047
    Abstract: Substituted 6-(2-methoxy-phenyl)-triazolopyrimidines of formula I in which R1 and R2 independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R1 and R2 radicals may be unsubstituted or substituted as defined in the description, or R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; L1, L2 independently denote hydrogen or halogen, provided that at least one from L1 or L2 is halogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositi
    Type: Grant
    Filed: July 8, 2002
    Date of Patent: May 2, 2006
    Assignee: BASF Aktiengesellschaft
    Inventors: Jordi Tormo i Blasco, Hubert Sauter, Bernd Müller, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Ingo Rose, Peter Schäfer, Frank Schieweck, Michael Rack, Eberhard Ammermann, Siegfried Strathmann, Gisela Lorenz, Reinhard Stierl
  • Publication number: 20060079537
    Abstract: 2-Substituted triazolopyrimidines of the formula I, in which the substituents are as defined below: L are halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, —C(?O)-A or S(?O)pA?; A and A? are as defined in the description; p is 0, 1 or 2; m is 0, 1, 2, 3, 4 or 5; X is cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S, where R1 and/or R2 may be substituted as defined in the description; and R3 is cyano, hydroxyl, alkoxy, alkeny
    Type: Application
    Filed: November 14, 2003
    Publication date: April 13, 2006
    Inventors: Jordi Blasco, Carsten Blettner, Bernd Muller, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Peter Schafer, Frank Schieweck, Anja Schwogler, Eberhard Ammermann, Siegfried Strathmann, Ulrich Schofl, Reinhard Stierl
  • Publication number: 20060058326
    Abstract: Pyrimidines of the formula I in which Ln is as defined in the description and the substituents R1, R2 and R3 are as defined below: R1 is C1-C10-alkyl, C2-C10-alkenyl, C2-C10-alkynyl, C3-C12-cycloalkyl, C3-C10-cycloalkenyl, phenyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon and contains one to four heteroatoms from the group consisting of O, N and S; R2 is halogen, cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-alkoxy, C3-C4-alkenyloxy or C3-C4-alkynyloxy, where the alkyl, alkenyl and alkynyl radicals of R2 may be substituted by halogen, cyano, nitro, C1-C2-alkoxy or C1-C4-alkoxycarbonyl; R3 is a five- or six-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S; and processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are
    Type: Application
    Filed: January 28, 2004
    Publication date: March 16, 2006
    Applicant: BASF AKTIENGESLLSCHAFT
    Inventors: Bernd Muller, Thomas Grote, Carsten Blettner, Markus Gewehr, Wassilios Grammenos, Andreas Gypser, Joachim Rheinheimer, Peter Schafer, Frank Schieweck, Anja Schwogler, Jordi Tormo I Blasco, Oliver Wagner, Maria Scherer, Siegfried Strathmann, Ulrich Schofl, Reinhard Stierl
  • Publication number: 20050272748
    Abstract: 2-Mercapto-substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy or —C(?O)-A; A is hydrogen, hydroxyl, alkyl, alkenyl, alkoxy, haloalkoxy, alkylamino or dialkylamino; m is 0, 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four hetero atoms from the group consisting of O, N and S; R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S; where R1 and/or R2 may be substituted as stated in the description; processes
    Type: Application
    Filed: November 14, 2003
    Publication date: December 8, 2005
    Applicant: BASF Aktiengesellschaft
    Inventors: Jordi Tormo Blasco, Carsten Blettner, Bernd Muller, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Peter Schafer, Frank Schieweck, Anja Schwogler, Eberhard Ammermann, Siegfried Strathmann, Ulrich Schofl, Reinhard Stierl
  • Publication number: 20050272749
    Abstract: 5-Alkyl-7-aminotriazolopyrimidines of the formula I, where: R1, R2 are hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cycloalkyl, phenyl, naphthyl; 5- or 6-membered saturated, unsaturated or aromatic heterocyclyl which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or R1 and R2 together with the bridging nitrogen atom can form a 5- or 6-membered ring which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 is cycloalkyl or bicycloalkyl; where R1, R2 and R3 may be substituted as outlined in the description; X is alkyl or haloalkyl; and their salts; processes and intermediates for their preparation, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.
    Type: Application
    Filed: November 4, 2003
    Publication date: December 8, 2005
    Applicant: BASF Aktiengesellschaft
    Inventors: Jordi Tormo Blasco, Carsten Bletner, Bernd Muller, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Peter Schafer, Frank Schieweck, Anja Schwogler, Eberhard Ammermann, Siegfried Strathmann, Ulrich Schofl, Reinhard Stierl
  • Publication number: 20050261314
    Abstract: The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R1, R2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R3 and R2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by Ra.
    Type: Application
    Filed: July 16, 2002
    Publication date: November 24, 2005
    Inventors: Jordi i Blasco, Hubert Sauter, Bernd Muller, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Andreas Gypser, Joachim Rheinheimer, Ingo Rose, Peter Schafer, Frank Schieweck, Eberhard Ammermann, Siegfried Strathmann, Gisela Lorenz, Reinhard Stierl